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Structure Report for: 5HQ3

Name Class
5HQ3NameHuman acetylcholinesterase designed variant expressed in bacteria
Gene_locushuman-ACHE
PaperGoldenzweig_2016_Mol.Cell_63_337
Mutation (51)
PDB_file5hq3-pdb
InhibitorVX
FamilyACHE
CommentGoldenzweig, A., Goldsmith, M., Hill, S.E., Gertman, O., Laurino, P.,
Ashani, Y., Dym, O., Albeck, S., Unger, T., Prilusky, J., Lieberman, R.L.,
Aharoni, A., Silman, I., Sussman, J.L., Tawfik, D.S., Fleishman, S.J. (51 substitutions)
(V12T,K23T,M42V,L48R,V60W,S67N,E91N,T109K,S110N,T112A,L115M,A127S,Q140R,A141T,
T144V,V187I,V226I,G234A,T238Y,G240S,M241R,G242E,T249L,H253K,T275N,A278P,
V280E,S309P,A318N,H322K,V331N,Q325D,A357E,A361E,V378I,R393K,L394N,E396D,V408I,
L414F,G416Q,L418Y,Q421N,A434S,S438P,L441E,A467K,Q474R,G506D,A507E,Q509K)
>5HQ3
MEGREDAELLVTTRGGRLRGIRLTTPGGPVSAFLGIPFAEPPVGPRRFRPPEPKQPWSGVWDATTFQNVCYQYVDTLYPG
FEGTEMWNPNRNLSEDCLYLNVWTPYPRPKNPAPVMVWIYGGGFYSGSSSLDVYDGRFLVRTERVVLVSMNYRVGAFGFL
ALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAILQSGAPNAPWAYV
SREEARRRALQLAKLVGCPPGGTGGNDTELVACLRNRPPQELVNHEWHVLPQESVFRFSFVPVVDGDFLPDTPEALINNG
DFKGLDVLVGVNKDEGSYFLVYGAPGFSKDNESLISREEFLEGVRVGVPQVSDLAAEAIVLHYTDWLHPEDPAKNRDALS
DVVGDHNVICPVAQFAQRYAANGARVYAYVFEHRSSTLPWPEWMGVPHGYEIEFIFGIPLDPSRNYTKEEKIFARRLMRY
WANFARTGDPNEPRDPKAPQWPPYTADEQKYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSATDTLD
Revelation_date27-Jul-2016
NewsJULY-27-2016

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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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