Name : Crystal structure of human butyrylcholinesterase in complex with N-((1-benzylpiperidin-3-yl)methyl)-N-methylnaphthalene-2-sulfonamide
Revelation date : 05-Oct-2016
Family : BCHE
Gene_locus : human-BCHE
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Kosak, U., Brus, B., Knez, D., Gobec, M., Sink, R., Zivin, M., Salat, K., Podkowa, A., Filipek, B., Wieckowska, A., Malawska, B., Stojan, J., Coquelle, N., Colletier, J.P., Gobec, S
Ligand :
Title : Development of an in-vivo active reversible butyrylcholinesterase inhibitor - Kosak_2016_Sci.Rep_6_39495 |
Author(s) : Kosak U , Brus B , Knez D , Sink R , Zakelj S , Trontelj J , Pislar A , Slenc J , Gobec M , Zivin M , Tratnjek L , Perse M , Salat K , Podkowa A , Filipek B , Nachon F , Brazzolotto X , Wieckowska A , Malawska B , Stojan J , Rascan IM , Kos J , Coquelle N , Colletier JP , Gobec S |
Ref : Sci Rep , 6 :39495 , 2016 |
Abstract : Kosak_2016_Sci.Rep_6_39495 |
ESTHER : Kosak_2016_Sci.Rep_6_39495 |
PubMedSearch : Kosak_2016_Sci.Rep_6_39495 |
PubMedID: 28000737 |
Gene_locus related to this paper: human-BCHE |
Title : Development of an in-vivo active reversible butyrylcholinesterase inhibitor - Kosak_2016_Sci.Rep_6_39495 |
Author(s) : Kosak U , Brus B , Knez D , Sink R , Zakelj S , Trontelj J , Pislar A , Slenc J , Gobec M , Zivin M , Tratnjek L , Perse M , Salat K , Podkowa A , Filipek B , Nachon F , Brazzolotto X , Wieckowska A , Malawska B , Stojan J , Rascan IM , Kos J , Coquelle N , Colletier JP , Gobec S |
Ref : Sci Rep , 6 :39495 , 2016 |
Abstract : Kosak_2016_Sci.Rep_6_39495 |
ESTHER : Kosak_2016_Sci.Rep_6_39495 |
PubMedSearch : Kosak_2016_Sci.Rep_6_39495 |
PubMedID: 28000737 |
Gene_locus related to this paper: human-BCHE |