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Structure Report for: 2OQI

Name|Human Dipeptidyl Peptidase IV (DPP4) with Piperidinone-constrained phenethylamine
Revelation date|03-Apr-2007
Family|DPP4N_Peptidase_S9: there are 829 genes in this family, 179 structure(s)
PDB File|ESTHER: header of PDB entry RCSB: Full entry
Pei, Z., Li, X., von Geldern, T. W., Longenecker, K.L., Pireh, D., Stewart, K.D., Backes, B.J., Lai, C., Lubben, T.H., Ballaron, S.J., Beno, D.W., Kempf-Grote, A.J., Sham, H.L., Trevillyan, J.M.
Ligand|Inhibitor: Piperidinone-constrained-phenethylamine-31 Ligand in structure: Ligplot


    Title: Discovery and structure-activity relationships of piperidinone- and piperidine-constrained phenethylamines as novel, potent, and selective dipeptidyl peptidase IV inhibitors
    Pei Z, Li X, von Geldern TW, Longenecker K, Pireh D, Stewart KD, Backes BJ, Lai C, Lubben TH and Trevillyan JM <4 more author(s)>
    Ref: Journal of Medicinal Chemistry, 50:1983, 2007 : PubMed


Representative scheme of DPP4N_Peptidase_S9 structure and an image from PDBsum server

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PDB-Sum2OQI Previously Class, Architecture, Topology and Homologous superfamily - PDB-Sum server
FSSP2OQI Fold classification based on Structure-Structure alignment of Proteins - FSSP server
SCOP2OQI Structural Classification Of Protein - SCOP server
PROTEOPEDIA2oqi 3D, interactive encyclopedia of proteins - PROTEOPEDIA server

Send your questions or comments to :
Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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