Name : Crystal structure of human lipoprotein-associated phospholipase A2 in complex with a [1.1.1]bicyclopentane- containing inhibitor at 1.91 A resolution
Revelation date : 01-Feb-2017
Family : PAF-Acetylhydrolase
Gene_locus : human-PLA2G7
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Somers DO
Ligand :
Title : Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replacement within an LpPLA2 Inhibitor - Measom_2017_ACS.Med.Chem.Lett_8_43 |
Author(s) : Measom ND , Down KD , Hirst DJ , Jamieson C , Manas ES , Patel VK , Somers DO |
Ref : ACS Med Chem Lett , 8 :43 , 2017 |
Abstract : Measom_2017_ACS.Med.Chem.Lett_8_43 |
ESTHER : Measom_2017_ACS.Med.Chem.Lett_8_43 |
PubMedSearch : Measom_2017_ACS.Med.Chem.Lett_8_43 |
PubMedID: 28105273 |
Gene_locus related to this paper: human-PLA2G7 |