Title : Pyrrolidine-constrained phenethylamines: The design of potent, selective, and pharmacologically efficacious dipeptidyl peptidase IV (DPP4) inhibitors from a lead-like screening hit - Backes_2007_Bioorg.Med.Chem.Lett_17_2005 |
Author(s) : Backes BJ , Longenecker K , Hamilton GL , Stewart K , Lai C , Kopecka H , von Geldern TW , Madar DJ , Pei Z , Lubben TH , Zinker BA , Tian Z , Ballaron SJ , Stashko MA , Mika AK , Beno DW , Kempf-Grote AJ , Black-Schaefer C , Sham HL , Trevillyan JM |
Ref : Bioorganic & Medicinal Chemistry Lett , 17 :2005 , 2007 |
Abstract : Backes_2007_Bioorg.Med.Chem.Lett_17_2005 |
ESTHER : Backes_2007_Bioorg.Med.Chem.Lett_17_2005 |
PubMedSearch : Backes_2007_Bioorg.Med.Chem.Lett_17_2005 |
PubMedID: 17276063 |
Gene_locus related to this paper: ratno-dpp4 , human-DPP4 |
Gene_locus related to this paper: ratno-dpp4 , human-DPP4 |
Backes BJ, Longenecker K, Hamilton GL, Stewart K, Lai C, Kopecka H, von Geldern TW, Madar DJ, Pei Z, Lubben TH, Zinker BA, Tian Z, Ballaron SJ, Stashko MA, Mika AK, Beno DW, Kempf-Grote AJ, Black-Schaefer C, Sham HL, Trevillyan JM (2007)
Pyrrolidine-constrained phenethylamines: The design of potent, selective, and pharmacologically efficacious dipeptidyl peptidase IV (DPP4) inhibitors from a lead-like screening hit
Bioorganic & Medicinal Chemistry Lett
17 :2005
Backes BJ, Longenecker K, Hamilton GL, Stewart K, Lai C, Kopecka H, von Geldern TW, Madar DJ, Pei Z, Lubben TH, Zinker BA, Tian Z, Ballaron SJ, Stashko MA, Mika AK, Beno DW, Kempf-Grote AJ, Black-Schaefer C, Sham HL, Trevillyan JM (2007)
Bioorganic & Medicinal Chemistry Lett
17 :2005