Title : Confirming target engagement for reversible inhibitors in vivo by kinetically tuned activity-based probes - Adibekian_2012_J.Am.Chem.Soc_134_10345 |
Author(s) : Adibekian A , Martin BR , Chang JW , Hsu KL , Tsuboi K , Bachovchin DA , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Hodder PS , Rosen H , Cravatt BF |
Ref : J Am Chem Soc , 134 :10345 , 2012 |
Abstract : Adibekian_2012_J.Am.Chem.Soc_134_10345 |
ESTHER : Adibekian_2012_J.Am.Chem.Soc_134_10345 |
PubMedSearch : Adibekian_2012_J.Am.Chem.Soc_134_10345 |
PubMedID: 22690931 |
Adibekian A, Martin BR, Chang JW, Hsu KL, Tsuboi K, Bachovchin DA, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Hodder PS, Rosen H, Cravatt BF (2012)
Confirming target engagement for reversible inhibitors in vivo by kinetically tuned activity-based probes
J Am Chem Soc
134 :10345
Adibekian A, Martin BR, Chang JW, Hsu KL, Tsuboi K, Bachovchin DA, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Hodder PS, Rosen H, Cravatt BF (2012)
J Am Chem Soc
134 :10345