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Mutation Report for: Q119G_human-BCHE

Q119G_human-BCHE
Gene_Locus|human-BCHE
Mode of mutation|Site directed mutagenesis
Amino Acid change|Q119G
Torpedo number|121
Summary|
Comment|p.Q119G Gln119Gly (p.Q147G Gln147Gly in primary sequence with 28 amino-acids signal peptide) no significant changes in Km and kcat for esters
Kinetic parameters|BW284C51_Q119G_human-BCHE,
Butyrylthiocholine_Q119G_human-BCHE,
Dibucaine_Q119G_human-BCHE,
Solanine_Q119G_human-BCHE,
Succinylcholine~Suxamethonium_Q119G_human-BCHE,
Tacrine_Q119G_human-BCHE


References:
    Title: Overlapping drug interaction sites of human butyrylcholinesterase dissected by site-directed mutagenesis
    Loewenstein-Lichtenstein Y, Glick D, Gluzman N, Sternfeld M, Zakut H, Soreq H
    Ref: Molecular Pharmacology, 50:1423, 1996 : PubMed

            




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Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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