Mutation

Kinetic parameters

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Kinetic parameters for mutation Y72N/Y124Q/W286R_mouse-ACHE

Substrate

MoleculeKmKcatExp. conditionsReference
Acetylthiocholine 850 & 130 uM 210000 & 60000/min 100mM NaP pH7 T22C eq3 sch3 Radic_1993_Biochemistry_32_12074

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
BW284C51 1600 & 200 nM 52000 & 20000 nM - 100mM NaP pH7.0 T22C eq3.gif sch3.gif Acetylthiocholine Radic_1993_Biochemistry_32_12074
Decamethonium 4000 & 1000 uM 10000 & 7000 uM - 100mM NaP pH7.0 T22C eq3.gif sch3.gif Acetylthiocholine Radic_1993_Biochemistry_32_12074
Edrophonium 2.1 & 0.8 uM 12 & 6 uM - 100mM NaP pH7.0 T22C eq3.gif sch3.gif Acetylthiocholine Radic_1993_Biochemistry_32_12074
Propidium 230 & 84 uM 470 & 210 uM - 100mM NaP pH7.0 T22C eq3.gif sch3.gif Acetylthiocholine Radic_1993_Biochemistry_32_12074
WT-fasciculin2 - 270000 & 20000 nM - 100mM NaP pH7.0 T37C eq4 sch4 meth6 Acetylthiocholine Radic_1994_J.Biol.Chem_269_11233

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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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