Mutation

Kinetic parameters

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Kinetic parameters for mutation V132A_human-ACHE

Substrate

MoleculeKmKcatExp. conditionsReference
3,3-dimethylbutylthioacetate 210 & 30 uM 58000 & 9000/min 50mM NaPhosphate pH8 Kronman_1994_J.Biol.Chem_269_27819
Acetylthiocholine 120 & 10 uM 340000 & 40000/min 50mM NaPhosphate pH8 Kronman_1994_J.Biol.Chem_269_27819

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
Edrophonium 1.2 & 0.1 uM - - 50mM NaPhosphate pH8 3.3-dimethylbutylthioacetate Kronman_1994_J.Biol.Chem_269_27819
Edrophonium 1.2 & 0.1 uM - - 50mM NaPhosphate pH8 Acetylthiocholine Kronman_1994_J.Biol.Chem_269_27819

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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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