Mutation

Kinetic parameters

Tree Display

AceDB Schema

XML Display

Feedback

Kinetic parameters for mutation F329Q_human-BCHE

Substrate

MoleculeKmKcatExp. conditionsReference
Butyrylthiocholine 0.88 mM - 100mM Na phosphate pH7.4 T22C Gnatt_1994_J.Neurochem_62_749

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
DFP - - 0.006 uM 100mM Na phosphate pH7.4 T22C Butyrylthiocholine Gnatt_1994_J.Neurochem_62_749
Echothiophate - - 3.7 uM 100mM Na phosphate pH7.4 T22C Butyrylthiocholine Gnatt_1994_J.Neurochem_62_749
Iso-OMPA - - 2 uM 100mM Na phosphate pH7.4 T22C Butyrylthiocholine Gnatt_1994_J.Neurochem_62_749

Send your questions or comments to :
Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
For technical information about these pages see:
ESTHER Home Page and ACEDB Home Page
AcePerl Lincoln Stein Home Page
webmaster

Acknowledgements and disclaimer