Mutation

Kinetic parameters

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Kinetic parameters for mutation F329D_human-BCHE

Substrate

MoleculeKmKcatExp. conditionsReference
Butyrylthiocholine 2.2 mM - 100mM Na phosphate pH7.4 T22C Gnatt_1994_J.Neurochem_62_749

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
DFP - - 0.03 uM 100mM Na phosphate pH7.4 T22C Butyrylthiocholine Gnatt_1994_J.Neurochem_62_749
Echothiophate - - 2 uM 100mM Na phosphate pH7.4 T22C Butyrylthiocholine Gnatt_1994_J.Neurochem_62_749
Iso-OMPA - - 30 uM 100mM Na phosphate pH7.4 T22C Butyrylthiocholine Gnatt_1994_J.Neurochem_62_749

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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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