Mutation

Kinetic parameters

Tree Display

AceDB Schema

XML Display

Feedback

Kinetic parameters for mutation F295L/F297V/Y337A_human-ACHE

Substrate

MoleculeKmKcatExp. conditionsReference
Acetylthiocholine 2900 uM 0.8 10+5/min IS 50mM phosphate pH8 T27C Kaplan_2001_Biochemistry_40_7433
Butyrylthiocholine 0.90 mM 0.55 10+5/min IS 50mM phosphate pH8 T27C Kaplan_2001_Biochemistry_40_7433

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
Decamethonium 210 uM - - T25C IS 50 mM phosphate Acetylthiocholine Kaplan_2001_Biochemistry_40_7433
Decamethonium 260 uM - - T25C IS 50 mM phosphate Acetylthiocholine Kaplan_2001_Biochemistry_40_7433
Edrophonium 53 uM - - T25C IS 50 mM phosphate Acetylthiocholine Kaplan_2001_Biochemistry_40_7433
HuperzineA 20000 nM - - T25C IS 50 mM phosphate Acetylthiocholine Kaplan_2001_Biochemistry_40_7433
Tacrine 9 nM - - T25C IS 50 mM phosphate Acetylthiocholine Kaplan_2001_Biochemistry_40_7433

Send your questions or comments to :
Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
For technical information about these pages see:
ESTHER Home Page and ACEDB Home Page
AcePerl Lincoln Stein Home Page
webmaster

Acknowledgements and disclaimer