Mutation

Kinetic parameters

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Kinetic parameters for mutation D349N_human-ACHE

Substrate

MoleculeKmKcatExp. conditionsReference
3,3-dimethylbutylthioacetate 220 & 30 uM 40000 & 5000/min IS 5mM Shafferman_1994_EMBO.J_13_3448
Acetylthiocholine 100 & 10 uM 390000 & 50000/min IS 5mM Shafferman_1994_EMBO.J_13_3448

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
Edrophonium 0.60 & 0.09 uM - - IS 150mM Acetylthiocholine Shafferman_1994_EMBO.J_13_3448

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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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