Barelier S, Avellan R, Gnawali GR, Fourquet P, Roig-Zamboni V, Poncin I, Point V, Bourne Y, Audebert S, Camoin L, Spilling CD, Canaan S, Cavalier JF, Sulzenbacher G (2022) <br />Direct capture, inhibition and crystal structure of HsaD (Rv3569c) from M. tuberculosis<br /><i>Febs J</i> <br /><br />Cavalier JF, Spilling CD, Durand T, Camoin L, Canaan S (2021) <br />Lipolytic enzymes inhibitors: A new way for antibacterial drugs discovery<br /><i>Eur Journal of Medicinal Chemistry</i> <b>209</b>: 112908<br /><br />Nguyen PC, Madani A, Santucci P, Martin BP, Paudel RR, Delattre S, Herrmann JL, Spilling CD, Kremer L, Canaan S, Cavalier JF (2018) <br />Cyclophostin and Cyclipostins analogues, new promising molecules to treat mycobacterial-related diseases<br /><i>Int J Antimicrob Agents</i> <b>51</b>: 651<br /><br />Nguyen PC, Nguyen VS, Martin BP, Fourquet P, Camoin L, Spilling CD, Cavalier JF, Cambillau C, Canaan S (2018) <br />Biochemical and Structural Characterization of TesA, a Major Thioesterase Required for Outer-Envelope Lipid Biosynthesis in Mycobacterium tuberculosis<br /><i>Journal of Molecular Biology</i> <b>430</b>: 5120<br /><br />Viljoen A, Richard M, Nguyen PC, Fourquet P, Camoin L, Paudal RR, Gnawali GR, Spilling CD, Cavalier JF, Canaan S, Blaise M, Kremer L (2018) <br />Cyclipostins and cyclophostin analogs inhibit the antigen 85C from Mycobacterium tuberculosis both in vitro and in vivo<br /><i>Journal of Biological Chemistry</i> <b>293</b>: 2755<br /><br />Nguyen PC, Delorme V, Benarouche A, Martin BP, Paudel R, Gnawali GR, Madani A, Puppo R, Landry V, Kremer L, Brodin P, Spilling CD, Cavalier JF, Canaan S (2017) <br />Cyclipostins and Cyclophostin analogs as promising compounds in the fight against tuberculosis<br /><i>Sci Rep</i> <b>7</b>: 11751<br /><br />Martin BP, Vasilieva E, Dupureur CM, Spilling CD (2015) <br />Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin<br /><i>Bioorganic & Medicinal Chemistry</i> <b>23</b>: 7529<br /><br />Vasilieva E, Dutta S, Malla RK, Martin BP, Spilling CD, Dupureur CM (2015) <br />Rat hormone sensitive lipase inhibition by cyclipostins and their analogs<br /><i>Bioorganic & Medicinal Chemistry</i> <b>23</b>: 944<br /><br />Point V, Malla RK, Carriere F, Canaan S, Spilling CD, Cavalier JF (2013) <br />Enantioselective inhibition of microbial lipolytic enzymes by nonracemic monocyclic enolphosphonate analogues of cyclophostin<br /><i>Journal of Medicinal Chemistry</i> <b>56</b>: 4393<br /><br />Point V, Malla RK, Diomande S, Martin BP, Delorme V, Carriere F, Canaan S, Rath NP, Spilling CD, Cavalier JF (2012) <br />Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases<br /><i>Journal of Medicinal Chemistry</i> <b>55</b>: 10204<br /><br />Malla RK, Bandyopadhyay S, Spilling CD, Dutta S, Dupureur CM (2011) <br />The first total synthesis of (+/-)-cyclophostin and (+/-)-cyclipostin P: inhibitors of the serine hydrolases acetyl cholinesterase and hormone sensitive lipase<br /><i>Org Lett</i> <b>13</b>: 3094<br /><br />Dutta S, Malla RK, Bandyopadhyay S, Spilling CD, Dupureur CM (2010) <br />Synthesis and kinetic analysis of some phosphonate analogs of cyclophostin as inhibitors of human acetylcholinesterase<br /><i>Bioorganic & Medicinal Chemistry</i> <b>18</b>: 2265<br /><br />Bandyopadhyay S, Dutta S, Spilling CD, Dupureur CM, Rath NP (2008) <br />Synthesis and biological evaluation of a phosphonate analog of the natural acetyl cholinesterase inhibitor cyclophostin<br /><i>J Org Chem</i> <b>73</b>: 8386<br /><br />