Barelier S, Avellan R, Gnawali GR, Fourquet P, Roig-Zamboni V, Poncin I, Point V, Bourne Y, Audebert S, Camoin L, Spilling CD, Canaan S, Cavalier JF, Sulzenbacher G (2022)
Direct capture, inhibition and crystal structure of HsaD (Rv3569c) from M. tuberculosis
Febs J

Cavalier JF, Spilling CD, Durand T, Camoin L, Canaan S (2021)
Lipolytic enzymes inhibitors: A new way for antibacterial drugs discovery
Eur Journal of Medicinal Chemistry 209: 112908

Nguyen PC, Madani A, Santucci P, Martin BP, Paudel RR, Delattre S, Herrmann JL, Spilling CD, Kremer L, Canaan S, Cavalier JF (2018)
Cyclophostin and Cyclipostins analogues, new promising molecules to treat mycobacterial-related diseases
Int J Antimicrob Agents 51: 651

Nguyen PC, Nguyen VS, Martin BP, Fourquet P, Camoin L, Spilling CD, Cavalier JF, Cambillau C, Canaan S (2018)
Biochemical and Structural Characterization of TesA, a Major Thioesterase Required for Outer-Envelope Lipid Biosynthesis in Mycobacterium tuberculosis
Journal of Molecular Biology 430: 5120

Viljoen A, Richard M, Nguyen PC, Fourquet P, Camoin L, Paudal RR, Gnawali GR, Spilling CD, Cavalier JF, Canaan S, Blaise M, Kremer L (2018)
Cyclipostins and cyclophostin analogs inhibit the antigen 85C from Mycobacterium tuberculosis both in vitro and in vivo
Journal of Biological Chemistry 293: 2755

Nguyen PC, Delorme V, Benarouche A, Martin BP, Paudel R, Gnawali GR, Madani A, Puppo R, Landry V, Kremer L, Brodin P, Spilling CD, Cavalier JF, Canaan S (2017)
Cyclipostins and Cyclophostin analogs as promising compounds in the fight against tuberculosis
Sci Rep 7: 11751

Martin BP, Vasilieva E, Dupureur CM, Spilling CD (2015)
Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin
Bioorganic & Medicinal Chemistry 23: 7529

Vasilieva E, Dutta S, Malla RK, Martin BP, Spilling CD, Dupureur CM (2015)
Rat hormone sensitive lipase inhibition by cyclipostins and their analogs
Bioorganic & Medicinal Chemistry 23: 944

Point V, Malla RK, Carriere F, Canaan S, Spilling CD, Cavalier JF (2013)
Enantioselective inhibition of microbial lipolytic enzymes by nonracemic monocyclic enolphosphonate analogues of cyclophostin
Journal of Medicinal Chemistry 56: 4393

Point V, Malla RK, Diomande S, Martin BP, Delorme V, Carriere F, Canaan S, Rath NP, Spilling CD, Cavalier JF (2012)
Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases
Journal of Medicinal Chemistry 55: 10204

Malla RK, Bandyopadhyay S, Spilling CD, Dutta S, Dupureur CM (2011)
The first total synthesis of (+/-)-cyclophostin and (+/-)-cyclipostin P: inhibitors of the serine hydrolases acetyl cholinesterase and hormone sensitive lipase
Org Lett 13: 3094

Dutta S, Malla RK, Bandyopadhyay S, Spilling CD, Dupureur CM (2010)
Synthesis and kinetic analysis of some phosphonate analogs of cyclophostin as inhibitors of human acetylcholinesterase
Bioorganic & Medicinal Chemistry 18: 2265

Bandyopadhyay S, Dutta S, Spilling CD, Dupureur CM, Rath NP (2008)
Synthesis and biological evaluation of a phosphonate analog of the natural acetyl cholinesterase inhibitor cyclophostin
J Org Chem 73: 8386