Kharlamova AD, Lushchekina SV, Petrov KA, Kots ED, Nachon F, Villard-Wandhammer M, Zueva IV, Krejci E, Reznik VS, Zobov VV, Nikolsky EE, Masson P (2016)
Slow-binding inhibition of acetylcholinesterase by an alkylammonium derivative of 6-methyluracil: mechanism and possible advantages for myasthenia gravis treatment
Biochemical Journal 473: 1225
Semenov VE, Zueva IV, Mukhamedyarov MA, Lushchekina SV, Kharlamova AD, Petukhova EO, Mikhailov AS, Podyachev SN, Saifina LF, Petrov KA, Minnekhanova OA, Zobov VV, Nikolsky EE, Masson P, Reznik VS (2015)
6-Methyluracil Derivatives as Bifunctional Acetylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease
ChemMedChem 10: 1863
Zueva IV, Semenov VE, Mukhamedyarov MA, Lushchekina SV, Kharlamova AD, Petukhova EO, Mikhailov AS, Podyachev SN, Saifina LF, Petrov KA, Minnekhanova OA, Zobov VV, Nikolsky EE, Masson P, Reznik VS (2015)
6-Methyluracil derivatives as acetylcholinesterase inhibitors for treatment of Alzheimer's disease
Int J Risk Saf Med 27 Suppl 1: S69
Nikitashina AD, Petrov KA, Zobov VV, Reznik VS, Nikolsky EE (2013)
Specific inhibitory effects of the alkylammonium derivative 6-methyluracil on acetylcholinesterase of smooth and striated muscles in rats
Dokl Biol Sci 449: 82
Lindovsky J, Petrov KA, Krusek J, Reznik VS, Nikolsky EE, Vyskocil F (2012)
Effect of tissue-specific acetylcholinesterase inhibitor C-547 on alpha3beta4 and alphabetaepsilondelta acetylcholine receptors in COS cells
European Journal of Pharmacology 688: 22
Petrov KA, Yagodina LO, Valeeva GR, Lannik NI, Nikitashina AD, Rizvanov AA, Zobov VV, Bukharaeva EA, Reznik VS, Nikolsky EE, Vyskocil F (2011)
Different sensitivities of rat skeletal muscles and brain to novel anti-cholinesterase agents, alkylammonium derivatives of 6-methyluracil (ADEMS)
British Journal of Pharmacology 163: 732
Anikienko KA, Bychikhin EA, Reznik VS, Akamsin D, Galyametdinova IV (2008)
Compounds with the dioxopyrimidine cycle inhibit cholinesterases from different groups of animals
Chemico-Biological Interactions 175: 286
Petrov KA, Kovyazina IV, Zobov VV, Bukharaeva EA, Reznik VS, Nikolsky EE (2007)
Effect of a tetraalkylammonium derivative of 6-methyluracil from a new class of acetylcholinesterase inhibitors on the endplate potential amplitude in muscles of different function types under high-frequency nerve stimulation
Dokl Biol Sci 415: 261
Zobov VV, Berezinskii LA, Aslyamova AA, Reznik VS (2005)
Delayed effects of daphnia intoxication with selective and nonselective inhibitors of acetylcholinesterase
Bulletin of Experimental Biology & Medicine 139: 68
Zobov VV, Petrov KA, Asliamova AA, Beresinskii LA, Akamsin VD, Galiametdinova IV, Reznik VS (2005)
Selective blockade of locomotor muscles by uracil-containing tetraalkylammonium acetylcholinesterase inhibitors
Dokl Biol Sci 401: 77
Anikienko KA, Bychikhin EA, Kurochkin VK, Reznik VS, Akamsin VD, Galyametdinova IV (2001)
Tetraalkylammonium derivatives of 6-methyluracil, a new class of cholinesterase inhibitors: characteristics of interaction with cholinesterases from different groups of animals
Dokl Biochem Biophys 376: 39
Gorshkova OV, Zobov VV, Bukharaeva EA, Nikolsky EE, Akamsin VD, Galyametdinova IV, Reznik VS (2001)
Effect of tetraalkylammonium derivative of 6-methyluracil on amplitude and temporal parameters of miniature endplate potentials in frog neuromuscular junction
Bulletin of Experimental Biology & Medicine 131: 446