Barelier S, Avellan R, Gnawali GR, Fourquet P, Roig-Zamboni V, Poncin I, Point V, Bourne Y, Audebert S, Camoin L, Spilling CD, Canaan S, Cavalier JF, Sulzenbacher G (2022)
Direct capture, inhibition and crystal structure of HsaD (Rv3569c) from M. tuberculosis
Febs J

Li M, Patel HV, Cognetta AB, 3rd, Smith TC, 2nd, Mallick I, Cavalier JF, Previti ML, Canaan S, Aldridge BB, Cravatt BF, Seeliger JC (2022)
Identification of cell wall synthesis inhibitors active against Mycobacterium tuberculosis by competitive activity-based protein profiling
Cell Chemical Biology 29: 883

Cavalier JF, Spilling CD, Durand T, Camoin L, Canaan S (2021)
Lipolytic enzymes inhibitors: A new way for antibacterial drugs discovery
Eur Journal of Medicinal Chemistry 209: 112908

Madani A, Mallick I, Guy A, Crauste C, Durand T, Fourquet P, Audebert S, Camoin L, Canaan S, Cavalier JF (2020)
Dissecting the antibacterial activity of oxadiazolone-core derivatives against Mycobacterium abscessus
PLoS ONE 15: e0238178

Nguyen PC, Madani A, Santucci P, Martin BP, Paudel RR, Delattre S, Herrmann JL, Spilling CD, Kremer L, Canaan S, Cavalier JF (2018)
Cyclophostin and Cyclipostins analogues, new promising molecules to treat mycobacterial-related diseases
Int J Antimicrob Agents 51: 651

Nguyen PC, Nguyen VS, Martin BP, Fourquet P, Camoin L, Spilling CD, Cavalier JF, Cambillau C, Canaan S (2018)
Biochemical and Structural Characterization of TesA, a Major Thioesterase Required for Outer-Envelope Lipid Biosynthesis in Mycobacterium tuberculosis
Journal of Molecular Biology 430: 5120

Nguyen PC, Delorme V, Benarouche A, Guy A, Landry V, Audebert S, Pophillat M, Camoin L, Crauste C, Galano JM, Durand T, Brodin P, Canaan S, Cavalier JF (2018)
Oxadiazolone derivatives, new promising multi-target inhibitors against M. tuberculosis
Bioorg Chem 81: 414

Viljoen A, Richard M, Nguyen PC, Fourquet P, Camoin L, Paudal RR, Gnawali GR, Spilling CD, Cavalier JF, Canaan S, Blaise M, Kremer L (2018)
Cyclipostins and cyclophostin analogs inhibit the antigen 85C from Mycobacterium tuberculosis both in vitro and in vivo
Journal of Biological Chemistry 293: 2755

Aouani I, Sellami B, Lahbib K, Cavalier JF, Touil S (2017)
Efficient synthesis of novel dialkyl-3-cyanopropylphosphate derivatives and evaluation of their anticholinesterase activity
Bioorg Chem 72: 301

Benarouche A, Sams L, Bourlieu C, Vie V, Point V, Cavalier JF, Carriere F (2017)
Studying Gastric Lipase Adsorption Onto Phospholipid Monolayers by Surface Tensiometry, Ellipsometry, and Atomic Force Microscopy
Methods Enzymol 583: 255

Nguyen PC, Delorme V, Benarouche A, Martin BP, Paudel R, Gnawali GR, Madani A, Puppo R, Landry V, Kremer L, Brodin P, Spilling CD, Cavalier JF, Canaan S (2017)
Cyclipostins and Cyclophostin analogs as promising compounds in the fight against tuberculosis
Sci Rep 7: 11751

Bourlieu C, Paboeuf G, Chever S, Pezennec S, Cavalier JF, Guyomarc'h F, Deglaire A, Bouhallab S, Dupont D, Carriere F, Vie V (2016)
Adsorption of gastric lipase onto multicomponent model lipid monolayers with phase separation
Colloids Surf B Biointerfaces 143: 97

Lemarie F, Cavalier JF, Garcia C, Boissel F, Point V, Catheline D, Legrand P, Carriere F, Rioux V (2016)
Effect of preduodenal lipase inhibition in suckling rats on dietary octanoic acid (C8:0) gastric absorption and plasma octanoylated ghrelin concentration
Biochimica & Biophysica Acta 1861: 1111

Point V, Benarouche A, Zarrillo J, Guy A, Magnez R, Fonseca L, Raux B, Leclaire J, Buono G, Fotiadu F, Durand T, Carriere F, Vaysse C, Couedelo L, Cavalier JF (2016)
Slowing down fat digestion and absorption by an oxadiazolone inhibitor targeting selectively gastric lipolysis
Eur Journal of Medicinal Chemistry 123: 834

Ulker S, Placidi C, Point V, Gadenne B, Serveau-Avesque C, Canaan S, Carriere F, Cavalier JF (2016)
New lipase assay using Pomegranate oil coating in microtiter plates
Biochimie 120: 110

Kamoun J, Schue M, Messaoud W, Baignol J, Point V, Mateos-Diaz E, Mansuelle P, Gargouri Y, Parsiegla G, Cavalier JF, Carriere F, Aloulou A (2015)
Biochemical characterization of Yarrowia lipolytica LIP8, a secreted lipase with a cleavable C-terminal region
Biochimica & Biophysica Acta 1851: 129

Benarouche A, Point V, Carriere F, Cavalier JF (2014)
An interfacial and comparative in vitro study of gastrointestinal lipases and Yarrowia lipolytica LIP2 lipase, a candidate for enzyme replacement therapy
Biochimie 102: 145

Benarouche A, Point V, Carriere F, Cavalier JF (2014)
Using the reversible inhibition of gastric lipase by Orlistat for investigating simultaneously lipase adsorption and substrate hydrolysis at the lipid-water interface
Biochimie 101: 221

Delorme V, Raux B, Puppo R, Leclaire J, Cavalier JF, Marc S, Kamarajugadda PK, Buono G, Fotiadu F, Canaan S, Carriere F (2014)
Supported inhibitor for fishing lipases in complex biological media and mass spectrometry identification
Biochimie 107 Pt A: 124

Aloulou A, Benarouche A, Puccinelli D, Spinelli S, Cavalier JF, Cambillau C, Carriere F (2013)
Biochemical and structural characterization of non-glycosylated Yarrowia lipolytica LIP2 lipase
Eur.J.Lipid.Sci.Tech 115: 429

Benarouche A, Point V, Parsiegla G, Carriere F, Cavalier JF (2013)
New insights into the pH-dependent interfacial adsorption of dog gastric lipase using the monolayer technique
Colloids Surf B Biointerfaces 111: 306

Point V, Malla RK, Carriere F, Canaan S, Spilling CD, Cavalier JF (2013)
Enantioselective inhibition of microbial lipolytic enzymes by nonracemic monocyclic enolphosphonate analogues of cyclophostin
Journal of Medicinal Chemistry 56: 4393

Point V, Benarouche A, Jemel I, Parsiegla G, Lambeau G, Carriere F, Cavalier JF (2013)
Effects of the propeptide of group X secreted phospholipase A(2) on substrate specificity and interfacial activity on phospholipid monolayers
Biochimie 95: 51

Delorme V, Diomande SV, Dedieu L, Cavalier JF, Carriere F, Kremer L, Leclaire J, Fotiadu F, Canaan S (2012)
MmPPOX inhibits Mycobacterium tuberculosis lipolytic enzymes belonging to the hormone-sensitive lipase family and alters mycobacterial growth
PLoS ONE 7: e46493

Point V, Malla RK, Diomande S, Martin BP, Delorme V, Carriere F, Canaan S, Rath NP, Spilling CD, Cavalier JF (2012)
Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases
Journal of Medicinal Chemistry 55: 10204

Point V, Pavan Kumar KV, Marc S, Delorme V, Parsiegla G, Amara S, Carriere F, Buono G, Fotiadu F, Canaan S, Leclaire J, Cavalier JF (2012)
Analysis of the discriminative inhibition of mammalian digestive lipases by 3-phenyl substituted 1,3,4-oxadiazol-2(3H)-ones.
Eur Journal of Medicinal Chemistry 58: 452

Delorme V, Dhouib R, Canaan S, Fotiadu F, Carriere F, Cavalier JF (2011)
Effects of surfactants on lipase structure, activity, and inhibition
Pharm Res 28: 1831

Cavalier JF, Lafont D, Boullanger P, Houisse D, Giallo J, Ballester JM, Carriere F (2009)
Validation of lipolysis product extraction from aqueous/biological samples, separation and quantification by thin-layer chromatography with flame ionization detection analysis using O-cholesteryl ethylene glycol as a new internal standard
Journal of Chromatography A 1216: 6543

Miled N, Riviere M, Cavalier JF, Buono G, Berti L, Verger R (2005)
Discrimination between closed and open forms of lipases using electrophoretic techniques
Analytical Biochemistry 338: 171

Cavalier JF, Buono G, Verger R (2000)
Covalent inhibition of digestive lipases by chiral phosphonates
Acc Chem Res 33: 579

Cavalier JF, Ransac S, Verger R, Buono G (1999)
Inhibition of human gastric and pancreatic lipases by chiral alkylphosphonates. A kinetic study with 1,2-didecanoyl-sn-glycerol monolayer
Chemistry & Physic of Lipids 100: 3