Lenina OA, Zueva IV, Zobov VV, Semenov VE, Masson P, Petrov KA (2020)
Slow-binding reversible inhibitor of acetylcholinesterase with long-lasting action for prophylaxis of organophosphate poisoning
Sci Rep 10: 16611
Petrov KA, Zueva IV, Kovyazina IV, Sedov I, Lushchekina SV, Kharlamova AD, Lenina O, Koshkin S, Shtyrlin Y, Nikolsky EE, Masson P (2018)
C-547, a 6-methyluracil derivative with long-lasting binding and rebinding on acetylcholinesterase: Pharmacokinetic and pharmacodynamic studies
Neuropharmacology 131: 304
Kharlamova AD, Lushchekina SV, Petrov KA, Kots ED, Nachon F, Villard-Wandhammer M, Zueva IV, Krejci E, Reznik VS, Zobov VV, Nikolsky EE, Masson P (2016)
Slow-binding inhibition of acetylcholinesterase by an alkylammonium derivative of 6-methyluracil: mechanism and possible advantages for myasthenia gravis treatment
Biochemical Journal 473: 1225
Semenov VE, Zueva IV, Mukhamedyarov MA, Lushchekina SV, Kharlamova AD, Petukhova EO, Mikhailov AS, Podyachev SN, Saifina LF, Petrov KA, Minnekhanova OA, Zobov VV, Nikolsky EE, Masson P, Reznik VS (2015)
6-Methyluracil Derivatives as Bifunctional Acetylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease
ChemMedChem 10: 1863
Lindovsky J, Petrov KA, Krusek J, Reznik VS, Nikolsky EE, Vyskocil F (2012)
Effect of tissue-specific acetylcholinesterase inhibitor C-547 on alpha3beta4 and alphabetaepsilondelta acetylcholine receptors in COS cells
European Journal of Pharmacology 688: 22
Petrov KA, Yagodina LO, Valeeva GR, Lannik NI, Nikitashina AD, Rizvanov AA, Zobov VV, Bukharaeva EA, Reznik VS, Nikolsky EE, Vyskocil F (2011)
Different sensitivities of rat skeletal muscles and brain to novel anti-cholinesterase agents, alkylammonium derivatives of 6-methyluracil (ADEMS)
British Journal of Pharmacology 163: 732
Abramochkin DV, Petrov KA, Zobov VV, Yagodina LO, Nikolsky EE, Rosenshtraukh LV (2009)
Mechanisms of cardiac muscle insensitivity to a novel acetylcholinesterase inhibitor C-547
J Cardiovasc Pharmacol 53: 162
Petrov KA, Kovyazina IV, Zobov VV, Bukharaeva EA, Nikolsky EE, Vyskocil F (2009)
Different sensitivity of miniature endplate currents in rat external and internal intercostal muscles to the acetylcholinesterase inhibitor C-547 as compared with diaphragm and extensor digitorum longus
Physiol Res 58: 149
Anikienko KA, Bychikhin EA, Reznik VS, Akamsin D, Galyametdinova IV (2008)
Compounds with the dioxopyrimidine cycle inhibit cholinesterases from different groups of animals
Chemico-Biological Interactions 175: 286
Petrov KA, Kovyazina LV, Zobov VV, Bukharaeva EA, Nikolsky EE, Vyskocil F (2006)
Different sensitivity of miniature endplate currents of the rat extensor digitorum longus, soleus and diaphragm muscles to a novel acetylcholinesterase inhibitor C-547
Physiol Res 55: 585
Gorshkova OV, Zobov VV, Bukharaeva EA, Nikolsky EE, Akamsin VD, Galyametdinova IV, Reznik VS (2001)
Effect of tetraalkylammonium derivative of 6-methyluracil on amplitude and temporal parameters of miniature endplate potentials in frog neuromuscular junction
Bulletin of Experimental Biology & Medicine 131: 446