Full name :
First name :
Mail :
Zip Code :
City :
Country :
Email :
Phone :
Fax :
Website :
Directory :
| Title : Preclinical metabolism and disposition of TP0473292, a novel oral prodrug of the potent metabotropic glutamate 2\/3 receptor antagonist TP0178894 for the treatment of depression - Inatani_2023_Drug.Metab.Dispos__ |
| Author(s) : Inatani S , Ochi M , Kinoshita K , Yamaguchi JI , Endo H |
| Ref : Drug Metabolism & Disposition: The Biological Fate of Chemicals , : , 2023 |
| Abstract : Inatani_2023_Drug.Metab.Dispos__ |
| ESTHER : Inatani_2023_Drug.Metab.Dispos__ |
| PubMedSearch : Inatani_2023_Drug.Metab.Dispos__ |
| PubMedID: 36754836 |
| Title : Bottom-up physiologically based pharmacokinetic modeling for predicting the human pharmacokinetic profiles of the ester prodrug MGS0274 and its active metabolite MGS0008, a metabotropic glutamate 2\/3 receptor agonist - Ochi_2022_Xenobiotica__1 |
| Author(s) : Ochi M , Kinoshita K , Yamaguchi JI , Endo H |
| Ref : Xenobiotica , :1 , 2022 |
| Abstract : Ochi_2022_Xenobiotica__1 |
| ESTHER : Ochi_2022_Xenobiotica__1 |
| PubMedSearch : Ochi_2022_Xenobiotica__1 |
| PubMedID: 35296225 |
| Title : Discovery of MGS0274, an ester prodrug of a metabotropic glutamate receptor 2\/3 agonist with improved oral bioavailability - Urabe_2020_Eur.J.Med.Chem_203_112521 |
| Author(s) : Urabe H , Miyakoshi N , Ohtake N , Nozoe A , Ochi M , Fukasawa M , Kinoshita K , Yamaguchi JI , Marumo T , Hikichi H , Chaki S , Hashihayata T |
| Ref : Eur Journal of Medicinal Chemistry , 203 :112521 , 2020 |
| Abstract : Urabe_2020_Eur.J.Med.Chem_203_112521 |
| ESTHER : Urabe_2020_Eur.J.Med.Chem_203_112521 |
| PubMedSearch : Urabe_2020_Eur.J.Med.Chem_203_112521 |
| PubMedID: 32698110 |