Report for Terstappen GC

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References (8)

Title : Preclinical assessment of an adjunctive treatment approach for cognitive impairment associated with schizophrenia using the alpha7 nicotinic acetylcholine receptor agonist WYE-103914\/SEN34625 - Marquis_2011_Psychopharmacology.(Berl)_218_635
Author(s) : Marquis KL , Comery TA , Jow F , Navarra RL , Grauer SM , Pulicicchio C , Kelley C , Brennan JA , Roncarati R , Scali C , Haydar S , Ghiron C , Terstappen GC , Dunlop J
Ref : Psychopharmacology (Berl) , 218 :635 , 2011
Abstract : Marquis_2011_Psychopharmacology.(Berl)_218_635
ESTHER : Marquis_2011_Psychopharmacology.(Berl)_218_635
PubMedSearch : Marquis_2011_Psychopharmacology.(Berl)_218_635
PubMedID: 21643676

Title : Novel alpha-7 nicotinic acetylcholine receptor agonists containing a urea moiety: identification and characterization of the potent, selective, and orally efficacious agonist 1-[6-(4-fluorophenyl)pyridin-3-yl]-3-(4-piperidin-1-ylbutyl) urea (SEN34625\/WYE-103914) - Ghiron_2010_J.Med.Chem_53_4379
Author(s) : Ghiron C , Haydar SN , Aschmies S , Bothmann H , Castaldo C , Cocconcelli G , Comery TA , Di L , Dunlop J , Lock T , Kramer A , Kowal D , Jow F , Grauer S , Harrison B , La Rosa S , Maccari L , Marquis KL , Micco I , Nencini A , Quinn J , Robichaud AJ , Roncarati R , Scali C , Terstappen GC , Turlizzi E , Valacchi M , Varrone M , Zanaletti R , Zanelli U
Ref : Journal of Medicinal Chemistry , 53 :4379 , 2010
Abstract : Ghiron_2010_J.Med.Chem_53_4379
ESTHER : Ghiron_2010_J.Med.Chem_53_4379
PubMedSearch : Ghiron_2010_J.Med.Chem_53_4379
PubMedID: 20465311

Title : Poster: In vitro pharmacological characterization and pro-cognitive effects of the selective alpha-7 nicotinic agonist WYE-103914 -
Author(s) : Dunlop J , Comery TA , Lock T , Kramer A , Kowal D , Yeola S , Jow F , Aschmies S , Lin Q , Beyer CE , Brennan J , Kelley C , Roncarati R , Scali C , Haydar S , Ghiron C , Marquis KL , Harrison B , Robichaud A , Terstappen GC
Ref : Biochemical Pharmacology , 78 :911 , 2009
PubMedID:

Title : Procognitive and neuroprotective activity of a novel alpha7 nicotinic acetylcholine receptor agonist for treatment of neurodegenerative and cognitive disorders - Roncarati_2009_J.Pharmacol.Exp.Ther_329_459
Author(s) : Roncarati R , Scali C , Comery TA , Grauer SM , Aschmi S , Bothmann H , Jow B , Kowal D , Gianfriddo M , Kelley C , Zanelli U , Ghiron C , Haydar S , Dunlop J , Terstappen GC
Ref : Journal of Pharmacology & Experimental Therapeutics , 329 :459 , 2009
Abstract : Roncarati_2009_J.Pharmacol.Exp.Ther_329_459
ESTHER : Roncarati_2009_J.Pharmacol.Exp.Ther_329_459
PubMedSearch : Roncarati_2009_J.Pharmacol.Exp.Ther_329_459
PubMedID: 19223665

Title : Poster: Characterization of the alpha-7 nicotinic receptor agonist WYE-103914 in models relevant to schizophrenia and interaction with antipsychotics -
Author(s) : Marquis KL , Comery TA , Navarra RL , Leiser S , Grauer SM , Pulicicchio C , Kelley C , Roncarati R , Scali C , Haydar S , Ghiron C , Harrison B , Robichaud A , Terstappen GC , Dunlop J
Ref : Biochemical Pharmacology , 78 :911 , 2009
PubMedID:

Title : Functional screening of alpha7 nicotinic receptor ligands - Dunlop_2008_Expert.Opin.Drug.Discov_3_623
Author(s) : Dunlop J , Peri R , Terstappen GC , Bowlby M
Ref : Expert Opin Drug Discov , 3 :623 , 2008
Abstract : Dunlop_2008_Expert.Opin.Drug.Discov_3_623
ESTHER : Dunlop_2008_Expert.Opin.Drug.Discov_3_623
PubMedSearch : Dunlop_2008_Expert.Opin.Drug.Discov_3_623
PubMedID: 23506144

Title : Functional properties of alpha7 nicotinic acetylcholine receptors co-expressed with RIC-3 in a stable recombinant CHO-K1 cell line - Roncarati_2008_Assay.Drug.Dev.Technol_6_181
Author(s) : Roncarati R , Seredenina T , Jow B , Jow F , Papini S , Kramer A , Bothmann H , Dunlop J , Terstappen GC
Ref : Assay Drug Dev Technol , 6 :181 , 2008
Abstract : Roncarati_2008_Assay.Drug.Dev.Technol_6_181
ESTHER : Roncarati_2008_Assay.Drug.Dev.Technol_6_181
PubMedSearch : Roncarati_2008_Assay.Drug.Dev.Technol_6_181
PubMedID: 18471073

Title : In vitro screening strategies for nicotinic receptor ligands - Dunlop_2007_Biochem.Pharmacol_74(8)_1172
Author(s) : Dunlop J , Roncarati R , Jow B , Bothmann H , Lock T , Kowal D , Bowlby M , Terstappen GC
Ref : Biochemical Pharmacology , 74 :1172 , 2007
Abstract : Dunlop_2007_Biochem.Pharmacol_74(8)_1172
ESTHER : Dunlop_2007_Biochem.Pharmacol_74(8)_1172
PubMedSearch : Dunlop_2007_Biochem.Pharmacol_74(8)_1172
PubMedID: 17706607