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Author Report for: Stepankova S

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    Title: Novel Inhibitors of Acetyl- and Butyrylcholinesterase Derived from Benzohydrazides: Synthesis, Evaluation and Docking Study
    Houngbedji NH, Stepankova S, Pflegr V, Svrckova K, Svarcova M, Vinsova J, Kratky M
    Ref: Pharmaceuticals (Basel), 16:, 2023 : PubMed

            

    Title: New 3-amino-2-thioxothiazolidin-4-one-based inhibitors of acetyl- and butyryl-cholinesterase: synthesis and activity
    Kratky M, Novackova K, Svrckova K, Svarcova M, Stepankova S
    Ref: Future Med Chem, :, 2023 : PubMed

            

    Title: Synthesis and neuroprotective activity of 3-aryl-3-azetidinyl acetic acid methyl ester derivatives
    Sachleviciute U, Gonzalez G, Kvasnicova M, Stepankova S, Kleizien N, Bieliauskas A, Zatloukal M, Strnad M, Slok FA and zukauskait A <2 more author(s)>
    Ref: Arch Pharm (Weinheim), :e2300378, 2023 : PubMed

            

    Title: Ring-fused 3beta-acetoxyandrost-5-enes as novel neuroprotective agents with cholinesterase inhibitory properties
    Gonzalez G, Kvasnica M, Svrckova K, Stepankova S, Santos JRC, Perina M, Jorda R, Lopes SMM, Melo T
    Ref: J Steroid Biochem Mol Biol, :106194, 2022 : PubMed

            

    Title: 5-Aryl-1,3,4-oxadiazol-2-amines Decorated with Long Alkyl and Their Analogues: Synthesis, Acetyl- and Butyrylcholinesterase Inhibition and Docking Study
    Pflegr V, Stepankova S, Svrckova K, Svarcova M, Vinsova J, Kratky M
    Ref: Pharmaceuticals (Basel), 15:400, 2022 : PubMed

            

    Title: Synthesis and Hybrid SAR Property Modeling of Novel Cholinesterase Inhibitors
    Kos J, Kozik V, Pindjakova D, Jankech T, Smolinski A, Stepankova S, Hosek J, Oravec M, Jampilek J, Bak A
    Ref: Int J Mol Sci, 22:, 2021 : PubMed

            

    Title: Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study
    Kratky M, Vu QA, Stepankova S, Maruca A, Silva TB, Ambroz M, Pflegr V, Rocca R, Svrckova K and Vinsova J <2 more author(s)>
    Ref: Bioorg Chem, 116:105301, 2021 : PubMed

            

    Title: Novel Aminoguanidine Hydrazone Analogues: From Potential Antimicrobial Agents to Potent Cholinesterase Inhibitors
    Kratky M, Stepankova S, Konecna K, Svrckova K, Maixnerova J, Svarcova M, Janourek O, Trejtnar F, Vinsova J
    Ref: Pharmaceuticals (Basel), 14:, 2021 : PubMed

            

    Title: Novel Sulfonamide-Based Carbamates as Selective Inhibitors of BChE
    Magar P, Parravicini O, Stepankova S, Svrckova K, Garro AD, Jendrzejewska I, Pauk K, Hosek J, Jampilek J and Imramovsky A <1 more author(s)>
    Ref: Int J Mol Sci, 22:, 2021 : PubMed

            

    Title: The synthesis and cholinesterase inhibitory activities of solasodine analogues with seven-membered F ring
    Kielczewska U, Jorda R, Gonzalez G, Morzycki JW, Ajani H, Svrckova K, Stepankova S, Wojtkielewicz A
    Ref: J Steroid Biochem Mol Biol, :105776, 2020 : PubMed

            

    Title: N-Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides and Their Analogues: Synthesis and Multitarget Biological Activity
    Kratky M, Baranyai Z, Stepankova S, Svrckova K, Svarcova M, Stolarikova J, Horvath L, Bosze S, Vinsova J
    Ref: Molecules, 25:, 2020 : PubMed

            

    Title: N-[3,5-Bis(trifluoromethyl)phenyl]-5-bromo-2-hydroxybenzamide Analogues: Novel Acetyl- and Butyrylcholinesterase Inhibitors
    Kratky M, Jaklova K, Stepankova S, Svrckova K, Pflegr V, Vinsova J
    Ref: Curr Top Med Chem, 20:2094, 2020 : PubMed

            

    Title: Novel Iodinated Hydrazide-hydrazones and their Analogues as Acetyl- and Butyrylcholinesterase Inhibitors
    Kratky M, Stepankova S, Brablikova M, Svrckova K, Svarcova M, Vinsova J
    Ref: Curr Top Med Chem, 20:2106, 2020 : PubMed

            

    Title: Novel Benzene-Based Carbamates for AChE/BChE Inhibition: Synthesis and Ligand/Structure-Oriented SAR Study
    Bak A, Kozik V, Kozakiewicz D, Gajcy K, Strub DJ, Swietlicka A, Stepankova S, Imramovsky A, Polanski J and Jampilek J <1 more author(s)>
    Ref: Int J Mol Sci, 20:1524, 2019 : PubMed

            

    Title: In Vitro and In Silico Acetylcholinesterase Inhibitory Activity of Thalictricavine and Canadine and Their Predicted Penetration across the Blood-Brain Barrier
    Chlebek J, Korabecny J, Dolezal R, Stepankova S, Perez DI, Hostalkova A, Opletal L, Cahlikova L, Macakova K and Jun D <2 more author(s)>
    Ref: Molecules, 24:, 2019 : PubMed

            

    Title: 2-Hydroxy-N-phenylbenzamides and Their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase
    Kratky M, Stepankova S, Houngbedji NH, Vosatka R, Vorcakova K, Vinsova J
    Ref: Biomolecules, 9:, 2019 : PubMed

            

    Title: Investigation of salicylanilide and 4-chlorophenol-based N-monosubstituted carbamates as potential inhibitors of acetyl- and butyrylcholinesterase
    Kratky M, Stepankova S, Vorcakova K, Vinsova J
    Ref: Bioorg Chem, 80:668, 2018 : PubMed

            

    Title: Synthesis and characterization of new inhibitors of cholinesterases based on N-phenylcarbamates: In vitro study of inhibitory effect, type of inhibition, lipophilicity and molecular docking
    Vorcakova K, Majekova M, Horakova E, Drabina P, Sedlak M, Stepankova S
    Ref: Bioorg Chem, 78:280, 2018 : PubMed

            

    Title: Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity
    Kratky M, Stepankova S, Vorcakova K, Navratilova L, Trejtnar F, Stolarikova J, Vinsova J
    Ref: Bioorg Chem, 71:244, 2017 : PubMed

            

    Title: Proline-Based Carbamates as Cholinesterase Inhibitors
    Pizova H, Havelkova M, Stepankova S, Bak A, Kauerova T, Kozik V, Oravec M, Imramovsky A, Kollar P and Jampilek J <1 more author(s)>
    Ref: Molecules, 22:, 2017 : PubMed

            

    Title: Synthesis, characterization and in vitro evaluation of substituted N-(2-phenylcyclopropyl)carbamates as acetyl- and butyrylcholinesterase inhibitors
    Horakova E, Drabina P, Broz B, Stepankova S, Vorcakova K, Kralovec K, Havelek R, Sedlak M
    Ref: J Enzyme Inhib Med Chem, :1, 2016 : PubMed

            

    Title: Novel Cholinesterase Inhibitors Based on O-Aromatic N,N-Disubstituted Carbamates and Thiocarbamates
    Kratky M, Stepankova S, Vorcakova K, Svarcova M, Vinsova J
    Ref: Molecules, 21:, 2016 : PubMed

            

    Title: Synthesis and in vitro evaluation of novel rhodanine derivatives as potential cholinesterase inhibitors
    Kratky M, Stepankova S, Vorcakova K, Vinsova J
    Ref: Bioorg Chem, 68:23, 2016 : PubMed

            

    Title: Synthesis, structural characterization, docking, lipophilicity and cytotoxicity of 1-[(1R)-1-(6-fluoro-1,3-benzothiazol-2-yl)ethyl]-3-alkyl carbamates, novel acetylcholinesterase and butyrylcholinesterase pseudo-irreversible inhibitors
    Pejchal V, Stepankova S, Pejchalova M, Kralovec K, Havelek R, Ruzickova Z, Ajani H, Lo R, Lepsik M
    Ref: Bioorganic & Medicinal Chemistry, 24:1560, 2016 : PubMed

            

    Title: Cholinesterase-based biosensors
    Stepankova S, Vorcakova K
    Ref: J Enzyme Inhib Med Chem, :1, 2016 : PubMed

            

    Title: In Vitro Inhibitory Effects of 8-O-Demethylmaritidine and Undulatine on Acetylcholinesterase and Their Predicted Penetration across the Blood-Brain Barrier
    Cahlikova L, Perez DI, Stepankova S, Chlebek J, Safratova M, Host'alkova A, Opletal L
    Ref: Journal of Natural Products, 78:1189, 2015 : PubMed

            

    Title: Chemical composition of bioactive alkaloid extracts from some Narcissus species and varieties and their biological activity
    Havlasova J, Safratova M, Siatka T, Stepankova S, Novak Z, Locarek M, Opletal L, Hrabinova M, Jun D and Cahlikova L <2 more author(s)>
    Ref: Nat Prod Commun, 9:1151, 2014 : PubMed

            

    Title: Salicylanilide diethyl phosphates as cholinesterases inhibitors
    Kratky M, Stepankova S, Vorcakova K, Vinsova J
    Ref: Bioorg Chem, 58C:48, 2014 : PubMed

            

    Title: Diethyl 2-(Phenylcarbamoyl)phenyl Phosphorothioates: Synthesis, Antimycobacterial Activity and Cholinesterase Inhibition
    Vinsova J, Kratky M, Komloova M, Dadapeer E, Stepankova S, Vorcakova K, Stolarikova J
    Ref: Molecules, 19:7152, 2014 : PubMed

            

    Title: Synthesis and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase inhibitors
    Imramovsky A, Pejchal V, Stepankova S, Vorcakova K, Jampilek J, Vanco J, Simunek P, Kralovec K, Bruckova L and Trejtnar F <1 more author(s)>
    Ref: Bioorganic & Medicinal Chemistry, 21:1735, 2013 : PubMed

            

    Title: New method for the determination of the half inhibition concentration (IC50) of cholinesterase inhibitors
    Kovarova M, Komers K, Stepankova S, Parik P, Cegan A
    Ref: Z Naturforsch C, 68:133, 2013 : PubMed

            

    Title: Acetylcholinesterase-inhibiting activity of salicylanilide N-alkylcarbamates and their molecular docking
    Imramovsky A, Stepankova S, Vanco J, Pauk K, Monreal-Ferriz J, Vinsova J, Jampilek J
    Ref: Molecules, 17:10142, 2012 : PubMed

            

    Title: 1,3-substituted imidazolidine-2,4,5-triones: synthesis and inhibition of cholinergic enzymes
    Pejchal V, Stepankova S, Padelkova Z, Imramovsky A, Jampilek J
    Ref: Molecules, 16:7565, 2011 : PubMed

            

    Title: Inhibition of acetylcholinesterase by 14 achiral and five chiral imidazole derivates
    Kovarova M, Komers K, Stepankova S, Cegan A
    Ref: Bioresour Technol, 101:6281, 2010 : PubMed

            

    Title: In vitro inhibition of cholinesterases by carbamates--a kinetic study
    Komersova A, Masopustova M, Komers K, Stepankova S, Cegan A
    Ref: Z Naturforsch C, 62:305, 2007 : PubMed

            

    Title: Inhibition of cholinesterase by dialkylcarbamates
    Stepankova S, Komers K, Komersova A, Masopustova M, Cegan A
    Ref: Z Naturforsch C, 62:308, 2007 : PubMed

            

    Title: Kinetics of 13 new cholinesterase inhibitors
    Zdrazilova P, Stepankova S, Komersova A, Vranova M, Komers K, Cegan A
    Ref: Z Naturforsch C, 61:611, 2006 : PubMed

            

    Title: Kinetics of total enzymatic hydrolysis of acetylcholine and acetylthiocholine
    Zdrazilova P, Stepankova S, Vranova M, Komers K, Komersova A, Cegan A
    Ref: Z Naturforsch C, 61:289, 2006 : PubMed

            

    Title: Two new methods monitoring kinetics of hydrolysis of acetylcholine and acetylthiocholine
    Stepankova S, Vranova M, Zdrazilova P, Komers K, Komersova A, Cegan A
    Ref: Z Naturforsch C, 60:943, 2005 : PubMed

            

    Title: Half-inhibition concentrations of new cholinesterase inhibitors
    Zdrazilova P, Stepankova S, Komers K, Ventura K, Cegan A
    Ref: Z Naturforsch C, 59:293, 2004 : PubMed

            


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