Biblio print

Tree Display

AceDB Schema

XML Display


Author Report for: Spilling CD

Contact information:

Spilling Christopher D
Department of Chemistry and Biochemistry and the Center for Nanoscience, University of Missouri-St. Louis, One University Boulevard, St. Louis, MO 63121
Phone :
Fax :
Send E-Mail to Spilling Christopher D

    Title: Direct capture, inhibition and crystal structure of HsaD (Rv3569c) from M. tuberculosis
    Barelier S, Avellan R, Gnawali GR, Fourquet P, Roig-Zamboni V, Poncin I, Point V, Bourne Y, Audebert S and Sulzenbacher G <4 more author(s)>
    Ref: Febs J, :, 2022 : PubMed


    Title: Lipolytic enzymes inhibitors: A new way for antibacterial drugs discovery
    Cavalier JF, Spilling CD, Durand T, Camoin L, Canaan S
    Ref: Eur Journal of Medicinal Chemistry, 209:112908, 2021 : PubMed


    Title: Cyclophostin and Cyclipostins analogues, new promising molecules to treat mycobacterial-related diseases
    Nguyen PC, Madani A, Santucci P, Martin BP, Paudel RR, Delattre S, Herrmann JL, Spilling CD, Kremer L and Cavalier JF <1 more author(s)>
    Ref: Int J Antimicrob Agents, 51:651, 2018 : PubMed


    Title: Biochemical and Structural Characterization of TesA, a Major Thioesterase Required for Outer-Envelope Lipid Biosynthesis in Mycobacterium tuberculosis
    Nguyen PC, Nguyen VS, Martin BP, Fourquet P, Camoin L, Spilling CD, Cavalier JF, Cambillau C, Canaan S
    Ref: Journal of Molecular Biology, 430:5120, 2018 : PubMed


    Title: Cyclipostins and cyclophostin analogs inhibit the antigen 85C from Mycobacterium tuberculosis both in vitro and in vivo
    Viljoen A, Richard M, Nguyen PC, Fourquet P, Camoin L, Paudal RR, Gnawali GR, Spilling CD, Cavalier JF and Kremer L <2 more author(s)>
    Ref: Journal of Biological Chemistry, 293:2755, 2018 : PubMed


    Title: Cyclipostins and Cyclophostin analogs as promising compounds in the fight against tuberculosis
    Nguyen PC, Delorme V, Benarouche A, Martin BP, Paudel R, Gnawali GR, Madani A, Puppo R, Landry V and Canaan S <4 more author(s)>
    Ref: Sci Rep, 7:11751, 2017 : PubMed


    Title: Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin
    Martin BP, Vasilieva E, Dupureur CM, Spilling CD
    Ref: Bioorganic & Medicinal Chemistry, 23:7529, 2015 : PubMed


    Title: Rat hormone sensitive lipase inhibition by cyclipostins and their analogs
    Vasilieva E, Dutta S, Malla RK, Martin BP, Spilling CD, Dupureur CM
    Ref: Bioorganic & Medicinal Chemistry, 23:944, 2015 : PubMed


    Title: Enantioselective inhibition of microbial lipolytic enzymes by nonracemic monocyclic enolphosphonate analogues of cyclophostin
    Point V, Malla RK, Carriere F, Canaan S, Spilling CD, Cavalier JF
    Ref: Journal of Medicinal Chemistry, 56:4393, 2013 : PubMed


    Title: Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases
    Point V, Malla RK, Diomande S, Martin BP, Delorme V, Carriere F, Canaan S, Rath NP, Spilling CD, Cavalier JF
    Ref: Journal of Medicinal Chemistry, 55:10204, 2012 : PubMed


    Title: The first total synthesis of (+/-)-cyclophostin and (+/-)-cyclipostin P: inhibitors of the serine hydrolases acetyl cholinesterase and hormone sensitive lipase
    Malla RK, Bandyopadhyay S, Spilling CD, Dutta S, Dupureur CM
    Ref: Org Lett, 13:3094, 2011 : PubMed


    Title: Synthesis and kinetic analysis of some phosphonate analogs of cyclophostin as inhibitors of human acetylcholinesterase
    Dutta S, Malla RK, Bandyopadhyay S, Spilling CD, Dupureur CM
    Ref: Bioorganic & Medicinal Chemistry, 18:2265, 2010 : PubMed


    Title: Synthesis and biological evaluation of a phosphonate analog of the natural acetyl cholinesterase inhibitor cyclophostin
    Bandyopadhyay S, Dutta S, Spilling CD, Dupureur CM, Rath NP
    Ref: J Org Chem, 73:8386, 2008 : PubMed


Send your questions or comments to :
Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
For technical information about these pages see:
ESTHER Home Page and ACEDB Home Page
AcePerl Lincoln Stein Home Page

Acknowledgements and disclaimer