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Title : Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A\/CLK1 kinases - Tintas_2024_RSC.Med.Chem_15_963 |
Author(s) : Tintas ML , Peauger L , Barre A , Papamical C , Besson T , Sopkova-de Oliveira Santos J , Gembus V , Levacher V |
Ref : RSC Med Chem , 15 :963 , 2024 |
Abstract : Tintas_2024_RSC.Med.Chem_15_963 |
ESTHER : Tintas_2024_RSC.Med.Chem_15_963 |
PubMedSearch : Tintas_2024_RSC.Med.Chem_15_963 |
PubMedID: 38516603 |
Title : Development of Novel Potential Pleiotropic Compounds of Interest in Alzheimer's Disease Treatment through Rigidification Strategy - Lecoutey_2021_Molecules_26_ |
Author(s) : Lecoutey C , Legay R , Davis A , Sopkova-de Oliveira Santos J , Dallemagne P , Rochais C |
Ref : Molecules , 26 : , 2021 |
Abstract : Lecoutey_2021_Molecules_26_ |
ESTHER : Lecoutey_2021_Molecules_26_ |
PubMedSearch : Lecoutey_2021_Molecules_26_ |
PubMedID: 33926141 |
Title : Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT(6) receptor antagonist with therapeutic interest in Alzheimer's disease - Toublet_2020_Eur.J.Med.Chem_210_113059 |
Author(s) : Toublet FX , Lalut J , Hatat B , Lecoutey C , Davis A , Since M , Corvaisier S , Freret T , Sopkova-de Oliveira Santos J , Claeysen S , Boulouard M , Dallemagne P , Rochais C |
Ref : Eur Journal of Medicinal Chemistry , 210 :113059 , 2020 |
Abstract : Toublet_2020_Eur.J.Med.Chem_210_113059 |
ESTHER : Toublet_2020_Eur.J.Med.Chem_210_113059 |
PubMedSearch : Toublet_2020_Eur.J.Med.Chem_210_113059 |
PubMedID: 33310288 |
Title : Rational design of novel benzisoxazole derivatives with acetylcholinesterase inhibitory and serotoninergic 5-HT4 receptors activities for the treatment of Alzheimer's disease - Lalut_2020_Sci.Rep_10_3014 |
Author(s) : Lalut J , Payan H , Davis A , Lecoutey C , Legay R , Sopkova-de Oliveira Santos J , Claeysen S , Dallemagne P , Rochais C |
Ref : Sci Rep , 10 :3014 , 2020 |
Abstract : Lalut_2020_Sci.Rep_10_3014 |
ESTHER : Lalut_2020_Sci.Rep_10_3014 |
PubMedSearch : Lalut_2020_Sci.Rep_10_3014 |
PubMedID: 32080261 |
Title : In silico chemical library screening and experimental validation of novel compounds with potential varroacide activities - Riva_2019_Pestic.Biochem.Physiol_160_11 |
Author(s) : Riva C , Suzanne P , Charpentier G , Dulin F , Halm-Lemeille MP , Sopkova-de Oliveira Santos J |
Ref : Pestic Biochem Physiol , 160 :11 , 2019 |
Abstract : Riva_2019_Pestic.Biochem.Physiol_160_11 |
ESTHER : Riva_2019_Pestic.Biochem.Physiol_160_11 |
PubMedSearch : Riva_2019_Pestic.Biochem.Physiol_160_11 |
PubMedID: 31519244 |
Title : Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a Bio-Oxidizable Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation - Peauger_2017_J.Med.Chem_60_5909 |
Author(s) : Peauger L , Azzouz R , Gembus V , Tintas ML , Sopkova-de Oliveira Santos J , Bohn P , Papamicael C , Levacher V |
Ref : Journal of Medicinal Chemistry , 60 :5909 , 2017 |
Abstract : Peauger_2017_J.Med.Chem_60_5909 |
ESTHER : Peauger_2017_J.Med.Chem_60_5909 |
PubMedSearch : Peauger_2017_J.Med.Chem_60_5909 |
PubMedID: 28613859 |
Title : Benzylphenylpyrrolizinones with Anti-amyloid and Radical Scavenging Effects, Potentially Useful in Alzheimer's Disease Treatment - Jourdan_2017_ChemMedChem_12_913 |
Author(s) : Jourdan JP , Since M , El Kihel L , Lecoutey C , Corvaisier S , Legay R , Sopkova-de Oliveira Santos J , Cresteil T , Malzert-Freon A , Rochais C , Dallemagne P |
Ref : ChemMedChem , 12 :913 , 2017 |
Abstract : Jourdan_2017_ChemMedChem_12_913 |
ESTHER : Jourdan_2017_ChemMedChem_12_913 |
PubMedSearch : Jourdan_2017_ChemMedChem_12_913 |
PubMedID: 28342294 |
Title : Novel benzylidenephenylpyrrolizinones with pleiotropic activities potentially useful in Alzheimer's disease treatment - Jourdan_2016_Eur.J.Med.Chem_114_365 |
Author(s) : Jourdan JP , Since M , El Kihel L , Lecoutey C , Corvaisier S , Legay R , Sopkova-de Oliveira Santos J , Cresteil T , Malzert-Freon A , Rochais C , Dallemagne P |
Ref : Eur Journal of Medicinal Chemistry , 114 :365 , 2016 |
Abstract : Jourdan_2016_Eur.J.Med.Chem_114_365 |
ESTHER : Jourdan_2016_Eur.J.Med.Chem_114_365 |
PubMedSearch : Jourdan_2016_Eur.J.Med.Chem_114_365 |
PubMedID: 27046230 |
Title : Virtual screening discovery of new acetylcholinesterase inhibitors issued from CERMN chemical library - Sopkova-de_2010_J.Chem.Inf.Model_50_422 |
Author(s) : Sopkova-de Oliveira Santos J , Lesnard A , Agondanou JH , Dupont N , Godard AM , Stiebing S , Rochais C , Fabis F , Dallemagne P , Bureau R , Rault S |
Ref : J Chem Inf Model , 50 :422 , 2010 |
Abstract : Sopkova-de_2010_J.Chem.Inf.Model_50_422 |
ESTHER : Sopkova-de_2010_J.Chem.Inf.Model_50_422 |
PubMedSearch : Sopkova-de_2010_J.Chem.Inf.Model_50_422 |
PubMedID: 20196555 |