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Title : Combining Experimental and Computational Methods to Produce Conjugates of Anticholinesterase and Antioxidant Pharmacophores with Linker Chemistries Affecting Biological Activities Related to Treatment of Alzheimer's Disease - Makhaeva_2024_Molecules_29_321 |
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serkov IV , Proshin AN , Soldatova YV , Poletaeva DA , Faingold, II , Mumyatova VA , Terentiev AA , Radchenko EV , Palyulin VA , Bachurin SO , Richardson RJ |
Ref : Molecules , 29 :321 , 2024 |
Abstract : Makhaeva_2024_Molecules_29_321 |
ESTHER : Makhaeva_2024_Molecules_29_321 |
PubMedSearch : Makhaeva_2024_Molecules_29_321 |
PubMedID: 38257233 |
Title : Bis-Amiridines as Acetylcholinesterase and Butyrylcholinesterase Inhibitors: N-Functionalization Determines the Multitarget Anti-Alzheimer's Activity Profile - Makhaeva_2022_Molecules_27_ |
Author(s) : Makhaeva GF , Kovaleva NV , Boltneva NP , Rudakova EV , Lushchekina SV , Astakhova TY , Serkov IV , Proshin AN , Radchenko EV , Palyulin VA , Korabecny J , Soukup O , Bachurin SO , Richardson RJ |
Ref : Molecules , 27 : , 2022 |
Abstract : Makhaeva_2022_Molecules_27_ |
ESTHER : Makhaeva_2022_Molecules_27_ |
PubMedSearch : Makhaeva_2022_Molecules_27_ |
PubMedID: 35164325 |
Title : Amiridine-piperazine hybrids as cholinesterase inhibitors and potential multitarget agents for Alzheimer's disease treatment - Makhaeva_2021_Bioorg.Chem_112_104974 |
Author(s) : Makhaeva GF , Lushchekina SV , Kovaleva NV , Yu Astakhova T , Boltneva NP , Rudakova EV , Serebryakova OG , Proshin AN , Serkov IV , Trofimova TP , Tafeenko VA , Radchenko EV , Palyulin VA , Fisenko VP , Korabecny J , Soukup O , Richardson RJ |
Ref : Bioorg Chem , 112 :104974 , 2021 |
Abstract : Makhaeva_2021_Bioorg.Chem_112_104974 |
ESTHER : Makhaeva_2021_Bioorg.Chem_112_104974 |
PubMedSearch : Makhaeva_2021_Bioorg.Chem_112_104974 |
PubMedID: 34029971 |
Title : New Multifunctional Agents Based on Conjugates of 4-Amino-2,3-polymethylenequinoline and Butylated Hydroxytoluene for Alzheimer's Disease Treatment - Makhaeva_2020_Molecules_25_5891 |
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Faingold, II , Poletaeva DA , Soldatova YV , Kotelnikova RA , Serkov IV , Ustinov AK , Proshin AN , Radchenko EV , Palyulin VA , Richardson RJ |
Ref : Molecules , 25 :5891 , 2020 |
Abstract : Makhaeva_2020_Molecules_25_5891 |
ESTHER : Makhaeva_2020_Molecules_25_5891 |
PubMedSearch : Makhaeva_2020_Molecules_25_5891 |
PubMedID: 33322783 |
Title : Arachidonoylcholine and Other Unsaturated Long-Chain Acylcholines Are Endogenous Modulators of the Acetylcholine Signaling System - Akimov_2020_Biomolecules_10_ |
Author(s) : Akimov MG , Kudryavtsev DS , Kryukova EV , Fomina-Ageeva EV , Zakharov SS , Gretskaya NM , Zinchenko GN , Serkov IV , Makhaeva GF , Boltneva NP , Kovaleva NV , Serebryakova OG , Lushchekina SV , Palikov VA , Palikova Y , Dyachenko IA , Kasheverov IE , Tsetlin VI , Bezuglov VV |
Ref : Biomolecules , 10 : , 2020 |
Abstract : Akimov_2020_Biomolecules_10_ |
ESTHER : Akimov_2020_Biomolecules_10_ |
PubMedSearch : Akimov_2020_Biomolecules_10_ |
PubMedID: 32059521 |
Title : New Hybrids of 4-Amino-2,3-polymethylene-quinoline and p-Tolylsulfonamide as Dual Inhibitors of Acetyl- and Butyrylcholinesterase and Potential Multifunctional Agents for Alzheimer's Disease Treatment - Makhaeva_2020_Molecules_25_3915 |
Author(s) : Makhaeva GF , Kovaleva NV , Boltneva NP , Lushchekina SV , Astakhova TY , Rudakova EV , Proshin AN , Serkov IV , Radchenko EV , Palyulin VA , Bachurin SO , Richardson RJ |
Ref : Molecules , 25 :3915 , 2020 |
Abstract : Makhaeva_2020_Molecules_25_3915 |
ESTHER : Makhaeva_2020_Molecules_25_3915 |
PubMedSearch : Makhaeva_2020_Molecules_25_3915 |
PubMedID: 32867324 |
Title : Conjugates of tacrine and 1,2,4-thiadiazole derivatives as new potential multifunctional agents for Alzheimer's disease treatment: Synthesis, quantum-chemical characterization, molecular docking, and biological evaluation - Makhaeva_2019_Bioorg.Chem__103387 |
Author(s) : Makhaeva GF , Kovaleva NV , Boltneva NP , Lushchekina SV , Rudakova EV , Stupina TS , Terentiev AA , Serkov IV , Proshin AN , Radchenko EV , Palyulin VV , Bachurin SO , Richardson RJ |
Ref : Bioorg Chem , :103387 , 2019 |
Abstract : Makhaeva_2019_Bioorg.Chem__103387 |
ESTHER : Makhaeva_2019_Bioorg.Chem__103387 |
PubMedSearch : Makhaeva_2019_Bioorg.Chem__103387 |
PubMedID: 31735356 |
Title : Conjugates of Tacrine and Its Cyclic Homologues with p-Toluenesulfonamide as Novel Acetylcholinesterase and Butyrylcholinesterase Inhibitors - Makhaeva_2018_Dokl.Biochem.Biophys_483_369 |
Author(s) : Makhaeva GF , Kovaleva NV , Lushchekina SV , Rudakova EV , Boltneva NP , Proshin AN , Lednev BV , Serkov IV , Bachurin SO |
Ref : Dokl Biochem Biophys , 483 :369 , 2018 |
Abstract : Makhaeva_2018_Dokl.Biochem.Biophys_483_369 |
ESTHER : Makhaeva_2018_Dokl.Biochem.Biophys_483_369 |
PubMedSearch : Makhaeva_2018_Dokl.Biochem.Biophys_483_369 |
PubMedID: 30607741 |
Title : Novel conjugates of tacrine with 1,2,4,-thiadiazole as highly effective cholinesterase inhibitors, blockers of NMDA receptors, and antioxidants - Makhaeva_2017_Dokl.Biochem.Biophys_477_405 |
Author(s) : Makhaeva GF , Grigoriev VV , Proshin AN , Kovaleva NV , Rudakova EV , Boltneva NP , Serkov IV , Bachurin SO |
Ref : Dokl Biochem Biophys , 477 :405 , 2017 |
Abstract : Makhaeva_2017_Dokl.Biochem.Biophys_477_405 |
ESTHER : Makhaeva_2017_Dokl.Biochem.Biophys_477_405 |
PubMedSearch : Makhaeva_2017_Dokl.Biochem.Biophys_477_405 |
PubMedID: 29297118 |
Title : Synthesis, molecular docking and biological evaluation of N,N-disubstituted 2-aminothiazolines as a new class of butyrylcholinesterase and carboxylesterase inhibitors - Makhaeva_2016_Bioorg.Med.Chem_24_1050 |
Author(s) : Makhaeva GF , Boltneva NP , Lushchekina SV , Serebryakova OG , Stupina TS , Terentiev AA , Serkov IV , Proshin AN , Bachurin SO , Richardson RJ |
Ref : Bioorganic & Medicinal Chemistry , 24 :1050 , 2016 |
Abstract : Makhaeva_2016_Bioorg.Med.Chem_24_1050 |
ESTHER : Makhaeva_2016_Bioorg.Med.Chem_24_1050 |
PubMedSearch : Makhaeva_2016_Bioorg.Med.Chem_24_1050 |
PubMedID: 26827140 |
Title : N,N-disubstituted 2-aminothiazolines as new inhibitors of serine esterases - |
Author(s) : Boltneva NP , Serebryakova OG , Makhaeva GF , Serkov IV , Proshin AN , Bachurin SO |
Ref : Dokl Biochem Biophys , 451 :209 , 2013 |
PubMedID: 23975403 |