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| Title : Disentangling the formation, mechanism, and evolvement of the covalent methanesulfonyl fluoride acetylcholinesterase adduct: Insights into an aged-like inactive complex susceptible to reactivation by a combination of nucleophiles - Stojan_2024_Protein.Sci_33_e4977 |
| Author(s) : Stojan J , Pesaresi A , Meden A , Lamba D |
| Ref : Protein Science , 33 :e4977 , 2024 |
| Abstract : Stojan_2024_Protein.Sci_33_e4977 |
| ESTHER : Stojan_2024_Protein.Sci_33_e4977 |
| PubMedSearch : Stojan_2024_Protein.Sci_33_e4977 |
| PubMedID: 38591646 |
| Title : Kinetic and structural studies on the inhibition of acetylcholinesterase and butyrylcholinesterase by a series of multitarget-directed galantamine-peptide derivatives - Pesaresi_2022_Chem.Biol.Interact__110092 |
| Author(s) : Pesaresi A , Lamba D , Vezenkov L , Tsekova D , Lozanov V |
| Ref : Chemico-Biological Interactions , :110092 , 2022 |
| Abstract : Pesaresi_2022_Chem.Biol.Interact__110092 |
| ESTHER : Pesaresi_2022_Chem.Biol.Interact__110092 |
| PubMedSearch : Pesaresi_2022_Chem.Biol.Interact__110092 |
| PubMedID: 35987277 |
| Title : Kinetic Modeling of Time-Dependent Enzyme Inhibition by Pre-Steady-State Analysis of Progress Curves: The Case Study of the Anti-Alzheimer's Drug Galantamine - Lamba_2022_Int.J.Mol.Sci_23_ |
| Author(s) : Lamba D , Pesaresi A |
| Ref : Int J Mol Sci , 23 : , 2022 |
| Abstract : Lamba_2022_Int.J.Mol.Sci_23_ |
| ESTHER : Lamba_2022_Int.J.Mol.Sci_23_ |
| PubMedSearch : Lamba_2022_Int.J.Mol.Sci_23_ |
| PubMedID: 35563466 |
| Title : Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease - Chalupova_2019_Eur.J.Med.Chem_168_491 |
| Author(s) : Chalupova K , Korabecny J , Bartolini M , Monti B , Lamba D , Caliandro R , Pesaresi A , Brazzolotto X , Gastellier AJ , Nachon F , Pejchal J , Jarosova M , Hepnarova V , Jun D , Hrabinova M , Dolezal R , Karasova JZ , Mzik M , Kristofikova Z , Misik J , Muckova L , Jost P , Soukup O , Benkova M , Setnicka V , Habartova L , Chvojkova M , Kleteckova L , Vales K , Mezeiova E , Uliassi E , Valis M , Nepovimova E , Bolognesi ML , Kuca K |
| Ref : Eur Journal of Medicinal Chemistry , 168 :491 , 2019 |
| Abstract : Chalupova_2019_Eur.J.Med.Chem_168_491 |
| ESTHER : Chalupova_2019_Eur.J.Med.Chem_168_491 |
| PubMedSearch : Chalupova_2019_Eur.J.Med.Chem_168_491 |
| PubMedID: 30851693 |
| Gene_locus related to this paper: torca-ACHE |
| Title : Kinetic and structural studies on the interactions of Torpedo californica acetylcholinesterase with two donepezil-like rigid analogues - Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
| Author(s) : Caliandro R , Pesaresi A , Cariati L , Procopio A , Oliverio M , Lamba D |
| Ref : J Enzyme Inhib Med Chem , 33 :794 , 2018 |
| Abstract : Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
| ESTHER : Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
| PubMedSearch : Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
| PubMedID: 29651884 |
| Gene_locus related to this paper: torca-ACHE |
| Title : Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and X-ray Crystallography - Zha_2016_J.Med.Chem_59_114 |
| Author(s) : Zha X , Lamba D , Zhang L , Lou Y , Xu C , Kang D , Chen L , Xu Y , De Simone A , Samez S , Pesaresi A , Stojan J , Lopez MG , Egea J , Andrisano V , Bartolini M |
| Ref : Journal of Medicinal Chemistry , 59 :114 , 2016 |
| Abstract : Zha_2016_J.Med.Chem_59_114 |
| ESTHER : Zha_2016_J.Med.Chem_59_114 |
| PubMedSearch : Zha_2016_J.Med.Chem_59_114 |
| PubMedID: 26632651 |
| Gene_locus related to this paper: torca-ACHE |
| Title : Multitarget Drug Design Strategy: Quinone-Tacrine Hybrids Designed To Block Amyloid-beta Aggregation and To Exert Anticholinesterase and Antioxidant Effects - Nepovimova_2014_J.Med.Chem_57_8576 |
| Author(s) : Nepovimova E , Uliassi E , Korabecny J , Pena-Altamira LE , Samez S , Pesaresi A , Garcia GE , Bartolini M , Andrisano V , Bergamini C , Fato R , Lamba D , Roberti M , Kuca K , Monti B , Bolognesi ML |
| Ref : Journal of Medicinal Chemistry , 57 :8576 , 2014 |
| Abstract : Nepovimova_2014_J.Med.Chem_57_8576 |
| ESTHER : Nepovimova_2014_J.Med.Chem_57_8576 |
| PubMedSearch : Nepovimova_2014_J.Med.Chem_57_8576 |
| PubMedID: 25259726 |
| Gene_locus related to this paper: torca-ACHE |
| Title : Evaluation and computational characterization of the facilitated transport of Glc carbon C-1 oxime reactivators across a blood brain barrier model - Bhonsle_2013_Chem.Biol.Interact_203_129 |
| Author(s) : Bhonsle JB , Causey R , Oyler BL , Bartolucci C , Lamba D , Pesaresi A , Bhamare NK , Soojhawon I , Garcia GE |
| Ref : Chemico-Biological Interactions , 203 :129 , 2013 |
| Abstract : Bhonsle_2013_Chem.Biol.Interact_203_129 |
| ESTHER : Bhonsle_2013_Chem.Biol.Interact_203_129 |
| PubMedSearch : Bhonsle_2013_Chem.Biol.Interact_203_129 |
| PubMedID: 23073172 |
| Title : Insights into the fatty acid chain length specificity of the carboxylesterase PA3859 from Pseudomonas aeruginosa: A combined structural, biochemical and computational study - Pesaresi_2010_Biochimie_92_1787 |
| Author(s) : Pesaresi A , Lamba D |
| Ref : Biochimie , 92 :1787 , 2010 |
| Abstract : Pesaresi_2010_Biochimie_92_1787 |
| ESTHER : Pesaresi_2010_Biochimie_92_1787 |
| PubMedSearch : Pesaresi_2010_Biochimie_92_1787 |
| PubMedID: 20850500 |
| Gene_locus related to this paper: pseae-PA3859 |
| Title : Isolation, characterization, and heterologous expression of a carboxylesterase of Pseudomonas aeruginosa PAO1 - Pesaresi_2005_Curr.Microbiol_50_102 |
| Author(s) : Pesaresi A , Devescovi G , Lamba D , Venturi V , Degrassi G |
| Ref : Curr Microbiol , 50 :102 , 2005 |
| Abstract : Pesaresi_2005_Curr.Microbiol_50_102 |
| ESTHER : Pesaresi_2005_Curr.Microbiol_50_102 |
| PubMedSearch : Pesaresi_2005_Curr.Microbiol_50_102 |
| PubMedID: 15717224 |
| Gene_locus related to this paper: pseae-PA3859 |
| Title : Crystallization, X-ray diffraction analysis and phasing of carboxylesterase PA3859 from Pseudomonas aeruginosa - Pesaresi_2005_Biochim.Biophys.Acta_1752_197 |
| Author(s) : Pesaresi A , Lamba D |
| Ref : Biochimica & Biophysica Acta , 1752 :197 , 2005 |
| Abstract : Pesaresi_2005_Biochim.Biophys.Acta_1752_197 |
| ESTHER : Pesaresi_2005_Biochim.Biophys.Acta_1752_197 |
| PubMedSearch : Pesaresi_2005_Biochim.Biophys.Acta_1752_197 |
| PubMedID: 16120484 |
| Gene_locus related to this paper: pseae-PA3859 |