Report for Pavia MR

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References (6)

Title : Design and synthesis of m1-selective muscarinic agonists: (R)-(-)-(Z)-1-Azabicyclo[2.2.1]heptan-3-one, O-(3-(3'-methoxyphenyl)-2-propynyl)oxime maleate (CI-1017), a functionally m1-selective muscarinic agonist - Tecle_1998_J.Med.Chem_41_2524
Author(s) : Tecle H , Barrett SD , Lauffer DJ , Augelli-Szafran C , Brann MR , Callahan MJ , Caprathe BW , Davis RE , Doyle PD , Eubanks D , Lipiniski W , Mirzadegan T , Moos WH , Moreland DW , Nelson CB , Pavia MR , Raby C , Schwarz RD , Spencer CJ , Thomas AJ , Jaen JC
Ref : Journal of Medicinal Chemistry , 41 :2524 , 1998
Abstract : Tecle_1998_J.Med.Chem_41_2524
ESTHER : Tecle_1998_J.Med.Chem_41_2524
PubMedSearch : Tecle_1998_J.Med.Chem_41_2524
PubMedID: 9651157

Title : Synthesis and SAR of bulky 1-azabicyclo[2.2.1]-3-one oximes as muscarinic receptor subtype selective agonists - Tecle_1993_Life.Sci_52(5-6)_505
Author(s) : Tecle H , Lauffer DJ , Mirzadegan T , Moos WH , Moreland DW , Pavia MR , Schwarz RD , Davis RE
Ref : Life Sciences , 52 :505 , 1993
Abstract : Tecle_1993_Life.Sci_52(5-6)_505
ESTHER : Tecle_1993_Life.Sci_52(5-6)_505
PubMedSearch : Tecle_1993_Life.Sci_52(5-6)_505
PubMedID: 8382765

Title : A silica gel plate-based qualitative assay for acetylcholinesterase activity: a mass method to screen for potential inhibitors - Kiely_1991_Anal.Biochem_196_439
Author(s) : Kiely JS , Moos WH , Pavia MR , Schwarz RD , Woodard GL
Ref : Analytical Biochemistry , 196 :439 , 1991
Abstract : Kiely_1991_Anal.Biochem_196_439
ESTHER : Kiely_1991_Anal.Biochem_196_439
PubMedSearch : Kiely_1991_Anal.Biochem_196_439
PubMedID: 1663710

Title : Poster: Inhibition of rat acetyl- and butyrylcholinesterase activity by tacrine and related aminoacridines -
Author(s) : Schwarz RD , Spencer CJ , Davis RE , Moos WH , Pavia MR , Thomas AJ
Ref : In: Cholinesterases: Structure, Function, Mechanism, Genetics, and Cell Biology , (Massoulie J, Barnard EA, Chatonnet A, Bacou F, Doctor BP, Quinn DM) American Chemical Society, Washington, DC :343 , 1991
PubMedID:

Title : Next generation tacrine -
Author(s) : Schwarz RD , Davis RE , Gracon S , Hoover T , Moos WH , Pavia MR
Ref : Neurobiology of Aging , 12 :185 , 1991
PubMedID: 2052133

Title : Poster: CI-969: An orally active muscarinic receptor agonist related to arecoline -
Author(s) : Pavia MR , Schwarz AD , Coughenour LL , Davis RE , Dudley DT , Moos WH , Pugsley TA , Tecle H , Clark CA
Ref : Trends in Pharmacological Sciences , Suppl :100 , 1989
PubMedID: