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Title : An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent - Willis_2019_Beilstein.J.Org.Chem_15_2790 |
Author(s) : Willis NJ , Bayle ED , Papageorgiou G , Steadman D , Atkinson BN , Mahy W , Fish PV |
Ref : Beilstein J Org Chem , 15 :2790 , 2019 |
Abstract : Willis_2019_Beilstein.J.Org.Chem_15_2790 |
ESTHER : Willis_2019_Beilstein.J.Org.Chem_15_2790 |
PubMedSearch : Willis_2019_Beilstein.J.Org.Chem_15_2790 |
PubMedID: 31807213 |
Gene_locus related to this paper: human-NOTUM |
Title : Scaffold-hopping identifies furano[2,3-d]pyrimidine amides as potent Notum inhibitors - Atkinson_2019_Bioorg.Med.Chem.Lett__126751 |
Author(s) : Atkinson BN , Steadman D , Mahy W , Zhao Y , Sipthorp J , Bayle ED , Svensson F , Papageorgiou G , Jeganathan F , Frew S , Monaghan A , Bictash M , Jones EY , Fish PV |
Ref : Bioorganic & Medicinal Chemistry Lett , :126751 , 2019 |
Abstract : Atkinson_2019_Bioorg.Med.Chem.Lett__126751 |
ESTHER : Atkinson_2019_Bioorg.Med.Chem.Lett__126751 |
PubMedSearch : Atkinson_2019_Bioorg.Med.Chem.Lett__126751 |
PubMedID: 31862412 |
Gene_locus related to this paper: human-NOTUM |