Full name : Nikolsky Evgeny E
First name : Evgeny E
Mail : Kazan State Medical University\; Department of Medical and Biological Physics\; 15\; Butlerova st.\; 420053
Zip Code :
City :
Country : Russia
Email : eenik1947@mail.ru
Phone : +78432387547
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Title : C-547, a 6-methyluracil derivative with long-lasting binding and rebinding on acetylcholinesterase: Pharmacokinetic and pharmacodynamic studies - Petrov_2018_Neuropharmacol_131_304 |
Author(s) : Petrov KA , Zueva IV , Kovyazina IV , Sedov I , Lushchekina SV , Kharlamova AD , Lenina O , Koshkin S , Shtyrlin Y , Nikolsky EE , Masson P |
Ref : Neuropharmacology , 131 :304 , 2018 |
Abstract : Petrov_2018_Neuropharmacol_131_304 |
ESTHER : Petrov_2018_Neuropharmacol_131_304 |
PubMedSearch : Petrov_2018_Neuropharmacol_131_304 |
PubMedID: 29277489 |
Title : Autoregulation of Acetylcholine Release and Micro-Pharmacodynamic Mechanisms at Neuromuscular Junction: Selective Acetylcholinesterase Inhibitors for Therapy of Myasthenic Syndromes - Petrov_2018_Front.Pharmacol_9_766 |
Author(s) : Petrov KA , Nikolsky EE , Masson P |
Ref : Front Pharmacol , 9 :766 , 2018 |
Abstract : Petrov_2018_Front.Pharmacol_9_766 |
ESTHER : Petrov_2018_Front.Pharmacol_9_766 |
PubMedSearch : Petrov_2018_Front.Pharmacol_9_766 |
PubMedID: 30050445 |
Title : Specific inhibition of acetylcholinesterase as an approach to decrease muscarinic side effects during myasthenia gravis treatment - Petrov_2018_Sci.Rep_8_304 |
Author(s) : Petrov KA , Kharlamova AD , Lenina OA , Nurtdinov AR , Sitdykova ME , Ilyin VI , Zueva IV , Nikolsky EE |
Ref : Sci Rep , 8 :304 , 2018 |
Abstract : Petrov_2018_Sci.Rep_8_304 |
ESTHER : Petrov_2018_Sci.Rep_8_304 |
PubMedSearch : Petrov_2018_Sci.Rep_8_304 |
PubMedID: 29321572 |
Title : Cholinergic Nociceptive Mechanisms in Rat Meninges and Trigeminal Ganglia: Potential Implications for Migraine Pain - Shelukhina_2017_Front.Neurol_8_163 |
Author(s) : Shelukhina I , Mikhailov N , Abushik P , Nurullin LF , Nikolsky EE , Giniatullin R |
Ref : Front Neurol , 8 :163 , 2017 |
Abstract : Shelukhina_2017_Front.Neurol_8_163 |
ESTHER : Shelukhina_2017_Front.Neurol_8_163 |
PubMedSearch : Shelukhina_2017_Front.Neurol_8_163 |
PubMedID: 28496430 |
Title : Nanoparticle-Delivered 2-PAM for Rat Brain Protection against Paraoxon Central Toxicity - Pashirova_2017_ACS.Appl.Mater.Interfaces_9_16922 |
Author(s) : Pashirova TN , Zueva IV , Petrov KA , Babaev VM , Lukashenko SS , Rizvanov IK , Souto EB , Nikolsky EE , Zakharova LY , Masson P , Sinyashin OG |
Ref : ACS Appl Mater Interfaces , 9 :16922 , 2017 |
Abstract : Pashirova_2017_ACS.Appl.Mater.Interfaces_9_16922 |
ESTHER : Pashirova_2017_ACS.Appl.Mater.Interfaces_9_16922 |
PubMedSearch : Pashirova_2017_ACS.Appl.Mater.Interfaces_9_16922 |
PubMedID: 28504886 |
Title : Slow-binding inhibition of acetylcholinesterase by an alkylammonium derivative of 6-methyluracil: mechanism and possible advantages for myasthenia gravis treatment - Kharlamova_2016_Biochem.J_473_1225 |
Author(s) : Kharlamova AD , Lushchekina SV , Petrov KA , Kots ED , Nachon F , Villard-Wandhammer M , Zueva IV , Krejci E , Reznik VS , Zobov VV , Nikolsky EE , Masson P |
Ref : Biochemical Journal , 473 :1225 , 2016 |
Abstract : Kharlamova_2016_Biochem.J_473_1225 |
ESTHER : Kharlamova_2016_Biochem.J_473_1225 |
PubMedSearch : Kharlamova_2016_Biochem.J_473_1225 |
PubMedID: 26929400 |
Gene_locus related to this paper: mouse-ACHE |
Title : Novel potent pyridoxine-based inhibitors of AChE and BChE, structural analogs of pyridostigmine, with improved in vivo safety profile - Strelnik_2016_Bioorg.Med.Chem.Lett_26_4092 |
Author(s) : Strelnik AD , Petukhov AS , Zueva IV , Zobov VV , Petrov KA , Nikolsky EE , Balakin KV , Bachurin SO , Shtyrlin YG |
Ref : Bioorganic & Medicinal Chemistry Lett , 26 :4092 , 2016 |
Abstract : Strelnik_2016_Bioorg.Med.Chem.Lett_26_4092 |
ESTHER : Strelnik_2016_Bioorg.Med.Chem.Lett_26_4092 |
PubMedSearch : Strelnik_2016_Bioorg.Med.Chem.Lett_26_4092 |
PubMedID: 27377327 |
Title : 6-Methyluracil Derivatives as Bifunctional Acetylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease - Semenov_2015_ChemMedChem_10_1863 |
Author(s) : Semenov VE , Zueva IV , Mukhamedyarov MA , Lushchekina SV , Kharlamova AD , Petukhova EO , Mikhailov AS , Podyachev SN , Saifina LF , Petrov KA , Minnekhanova OA , Zobov VV , Nikolsky EE , Masson P , Reznik VS |
Ref : ChemMedChem , 10 :1863 , 2015 |
Abstract : Semenov_2015_ChemMedChem_10_1863 |
ESTHER : Semenov_2015_ChemMedChem_10_1863 |
PubMedSearch : Semenov_2015_ChemMedChem_10_1863 |
PubMedID: 26412714 |
Title : 6-Methyluracil derivatives as acetylcholinesterase inhibitors for treatment of Alzheimer's disease - Zueva_2015_Int.J.Risk.Saf.Med_27 Suppl 1_S69 |
Author(s) : Zueva IV , Semenov VE , Mukhamedyarov MA , Lushchekina SV , Kharlamova AD , Petukhova EO , Mikhailov AS , Podyachev SN , Saifina LF , Petrov KA , Minnekhanova OA , Zobov VV , Nikolsky EE , Masson P , Reznik VS |
Ref : Int J Risk Saf Med , 27 Suppl 1 :S69 , 2015 |
Abstract : Zueva_2015_Int.J.Risk.Saf.Med_27 Suppl 1_S69 |
ESTHER : Zueva_2015_Int.J.Risk.Saf.Med_27 Suppl 1_S69 |
PubMedSearch : Zueva_2015_Int.J.Risk.Saf.Med_27 Suppl 1_S69 |
PubMedID: 26639718 |
Title : Schwann Cells Sense and Control Acetylcholine Spillover at the Neuromuscular Junction by alpha7 Nicotinic Receptors and Butyrylcholinesterase - Petrov_2014_J.Neurosci_34_11870 |
Author(s) : Petrov KA , Girard E , Nikitashina AD , Colasante C , Bernard V , Nurullin LF , Leroy J , Samigullin D , Colak O , Nikolsky EE , Plaud B , Krejci E |
Ref : Journal of Neuroscience , 34 :11870 , 2014 |
Abstract : Petrov_2014_J.Neurosci_34_11870 |
ESTHER : Petrov_2014_J.Neurosci_34_11870 |
PubMedSearch : Petrov_2014_J.Neurosci_34_11870 |
PubMedID: 25186736 |
Title : Specific inhibitory effects of the alkylammonium derivative 6-methyluracil on acetylcholinesterase of smooth and striated muscles in rats - |
Author(s) : Nikitashina AD , Petrov KA , Zobov VV , Reznik VS , Nikolsky EE |
Ref : Dokl Biol Sci , 449 :82 , 2013 |
PubMedID: 23652433 |
Title : Regulation of acetylcholinesterase activity by nitric oxide in rat neuromuscular junction via N-methyl-d-aspartate receptor activation - Petrov_2013_Eur.J.Neurosci_37_181 |
Author(s) : Petrov KA , Malomouzh AI , Kovyazina IV , Krejci E , Nikitashina AD , Proskurina SE , Zobov VV , Nikolsky EE |
Ref : European Journal of Neuroscience , 37 :181 , 2013 |
Abstract : Petrov_2013_Eur.J.Neurosci_37_181 |
ESTHER : Petrov_2013_Eur.J.Neurosci_37_181 |
PubMedSearch : Petrov_2013_Eur.J.Neurosci_37_181 |
PubMedID: 23121214 |
Title : Effect of tissue-specific acetylcholinesterase inhibitor C-547 on alpha3beta4 and alphabetaepsilondelta acetylcholine receptors in COS cells - Lindovsky_2012_Eur.J.Pharmacol_688_22 |
Author(s) : Lindovsky J , Petrov KA , Krusek J , Reznik VS , Nikolsky EE , Vyskocil F |
Ref : European Journal of Pharmacology , 688 :22 , 2012 |
Abstract : Lindovsky_2012_Eur.J.Pharmacol_688_22 |
ESTHER : Lindovsky_2012_Eur.J.Pharmacol_688_22 |
PubMedSearch : Lindovsky_2012_Eur.J.Pharmacol_688_22 |
PubMedID: 22634638 |
Title : Both neuronal and non-neuronal acetylcholine take part in non-quantal acetylcholine release in the rat atrium - Abramochkin_2012_Life.Sci_91_1023 |
Author(s) : Abramochkin DV , Borodinova AA , Rosenshtraukh LV , Nikolsky EE |
Ref : Life Sciences , 91 :1023 , 2012 |
Abstract : Abramochkin_2012_Life.Sci_91_1023 |
ESTHER : Abramochkin_2012_Life.Sci_91_1023 |
PubMedSearch : Abramochkin_2012_Life.Sci_91_1023 |
PubMedID: 23289117 |
Title : Different sensitivities of rat skeletal muscles and brain to novel anti-cholinesterase agents, alkylammonium derivatives of 6-methyluracil (ADEMS) - Petrov_2011_Br.J.Pharmacol_163_732 |
Author(s) : Petrov KA , Yagodina LO , Valeeva GR , Lannik NI , Nikitashina AD , Rizvanov AA , Zobov VV , Bukharaeva EA , Reznik VS , Nikolsky EE , Vyskocil F |
Ref : British Journal of Pharmacology , 163 :732 , 2011 |
Abstract : Petrov_2011_Br.J.Pharmacol_163_732 |
ESTHER : Petrov_2011_Br.J.Pharmacol_163_732 |
PubMedSearch : Petrov_2011_Br.J.Pharmacol_163_732 |
PubMedID: 21232040 |
Title : Non-quantal release of acetylcholine from parasympathetic nerve terminals in the right atrium of rats - Abramochkin_2010_Exp.Physiol_95_265 |
Author(s) : Abramochkin DV , Nurullin LF , Borodinova AA , Tarasova NV , Sukhova GS , Nikolsky EE , Rosenshtraukh LV |
Ref : Exp Physiol , 95 :265 , 2010 |
Abstract : Abramochkin_2010_Exp.Physiol_95_265 |
ESTHER : Abramochkin_2010_Exp.Physiol_95_265 |
PubMedSearch : Abramochkin_2010_Exp.Physiol_95_265 |
PubMedID: 19767403 |
Title : Mechanisms of cardiac muscle insensitivity to a novel acetylcholinesterase inhibitor C-547 - Abramochkin_2009_J.Cardiovasc.Pharmacol_53_162 |
Author(s) : Abramochkin DV , Petrov KA , Zobov VV , Yagodina LO , Nikolsky EE , Rosenshtraukh LV |
Ref : J Cardiovasc Pharmacol , 53 :162 , 2009 |
Abstract : Abramochkin_2009_J.Cardiovasc.Pharmacol_53_162 |
ESTHER : Abramochkin_2009_J.Cardiovasc.Pharmacol_53_162 |
PubMedSearch : Abramochkin_2009_J.Cardiovasc.Pharmacol_53_162 |
PubMedID: 19188831 |
Title : Different sensitivity of miniature endplate currents in rat external and internal intercostal muscles to the acetylcholinesterase inhibitor C-547 as compared with diaphragm and extensor digitorum longus - Petrov_2009_Physiol.Res_58_149 |
Author(s) : Petrov KA , Kovyazina IV , Zobov VV , Bukharaeva EA , Nikolsky EE , Vyskocil F |
Ref : Physiol Res , 58 :149 , 2009 |
Abstract : Petrov_2009_Physiol.Res_58_149 |
ESTHER : Petrov_2009_Physiol.Res_58_149 |
PubMedSearch : Petrov_2009_Physiol.Res_58_149 |
PubMedID: 19331513 |
Title : Effect of a tetraalkylammonium derivative of 6-methyluracil from a new class of acetylcholinesterase inhibitors on the endplate potential amplitude in muscles of different function types under high-frequency nerve stimulation - |
Author(s) : Petrov KA , Kovyazina IV , Zobov VV , Bukharaeva EA , Reznik VS , Nikolsky EE |
Ref : Dokl Biol Sci , 415 :261 , 2007 |
PubMedID: 17929660 |
Title : Different sensitivity of miniature endplate currents of the rat extensor digitorum longus, soleus and diaphragm muscles to a novel acetylcholinesterase inhibitor C-547 - Petrov_2006_Physiol.Res_55_585 |
Author(s) : Petrov KA , Kovyazina LV , Zobov VV , Bukharaeva EA , Nikolsky EE , Vyskocil F |
Ref : Physiol Res , 55 :585 , 2006 |
Abstract : Petrov_2006_Physiol.Res_55_585 |
ESTHER : Petrov_2006_Physiol.Res_55_585 |
PubMedSearch : Petrov_2006_Physiol.Res_55_585 |
PubMedID: 16792471 |
Title : Effect of N-acetylaspartylglutamate (NAAG) on non-quantal and spontaneous quantal release of acetylcholine at the neuromuscular synapse of rat - Malomouzh_2005_J.Neurochem_94_257 |
Author(s) : Malomouzh AI , Nikolsky EE , Lieberman EM , Sherman JA , Lubischer JL , Grossfeld RM , Urazaev A |
Ref : Journal of Neurochemistry , 94 :257 , 2005 |
Abstract : Malomouzh_2005_J.Neurochem_94_257 |
ESTHER : Malomouzh_2005_J.Neurochem_94_257 |
PubMedSearch : Malomouzh_2005_J.Neurochem_94_257 |
PubMedID: 15953368 |
Title : Dependence of miniature endplate current on kinetic parameters of acetylcholine receptors activation: a model study - Kovyazina_2003_Neurochem.Res_28_443 |
Author(s) : Kovyazina IV , Nikolsky EE , Giniatullin RA , Adamek S , Vyskocil F |
Ref : Neurochem Res , 28 :443 , 2003 |
Abstract : Kovyazina_2003_Neurochem.Res_28_443 |
ESTHER : Kovyazina_2003_Neurochem.Res_28_443 |
PubMedSearch : Kovyazina_2003_Neurochem.Res_28_443 |
PubMedID: 12675129 |
Title : Glutamate regulation of non-quantal release of acetylcholine in the rat neuromuscular junction - Malomouzh_2003_J.Neurochem_85_206 |
Author(s) : Malomouzh AI , Mukhtarov MR , Nikolsky EE , Vyskocil F , Lieberman EM , Urazaev AK |
Ref : Journal of Neurochemistry , 85 :206 , 2003 |
Abstract : Malomouzh_2003_J.Neurochem_85_206 |
ESTHER : Malomouzh_2003_J.Neurochem_85_206 |
PubMedSearch : Malomouzh_2003_J.Neurochem_85_206 |
PubMedID: 12641742 |
Title : Effect of tetraalkylammonium derivative of 6-methyluracil on amplitude and temporal parameters of miniature endplate potentials in frog neuromuscular junction - Gorshkova_2001_Bull.Exp.Biol.Med_131_446 |
Author(s) : Gorshkova OV , Zobov VV , Bukharaeva EA , Nikolsky EE , Akamsin VD , Galyametdinova IV , Reznik VS |
Ref : Bulletin of Experimental Biology & Medicine , 131 :446 , 2001 |
Abstract : Gorshkova_2001_Bull.Exp.Biol.Med_131_446 |
ESTHER : Gorshkova_2001_Bull.Exp.Biol.Med_131_446 |
PubMedSearch : Gorshkova_2001_Bull.Exp.Biol.Med_131_446 |
PubMedID: 11550049 |
Title : Modulation by nitric oxide (NO) of the intensity of non-quantum mediator secretion in neuromuscular junctions in rats - Mukhtarov_2001_Neurosci.Behav.Physiol_31_451 |
Author(s) : Mukhtarov MR , Urazaev AK , Nikolsky EE , Vyskocil F |
Ref : Neurosci Behav Physiol , 31 :451 , 2001 |
Abstract : Mukhtarov_2001_Neurosci.Behav.Physiol_31_451 |
ESTHER : Mukhtarov_2001_Neurosci.Behav.Physiol_31_451 |
PubMedSearch : Mukhtarov_2001_Neurosci.Behav.Physiol_31_451 |
PubMedID: 11508498 |
Title : Non-quantal acetylcholine release is increased after nitric oxide synthase inhibition - Mukhtarov_1999_Physiol.Res_48_315 |
Author(s) : Mukhtarov MR , Vyskocil F , Urazaev AK , Nikolsky EE |
Ref : Physiol Res , 48 :315 , 1999 |
Abstract : Mukhtarov_1999_Physiol.Res_48_315 |
ESTHER : Mukhtarov_1999_Physiol.Res_48_315 |
PubMedSearch : Mukhtarov_1999_Physiol.Res_48_315 |
PubMedID: 10638684 |
Title : The NO-mediated effect of carbachol and glutamate on postdenervation decrease of membrane potential in rat diaphragm is directed towards furosemide-sensitive chloride transport - |
Author(s) : Vyskocil F , Urazaev AK , Naumenko NV , Nikolsky EE |
Ref : Journal de Physiologie (Paris) , 92 :507 , 1998 |
PubMedID: |
Title : Role of non-quantal acetylcholine release in surplus polarization of mouse diaphragm fibres at the endplate zone - Nikolsky_1994_J.Physiol_477_497 |
Author(s) : Nikolsky EE , Zemkova H , Voronin VA , Vyskocil F |
Ref : The Journal of Physiology , 477 :497 , 1994 |
Abstract : Nikolsky_1994_J.Physiol_477_497 |
ESTHER : Nikolsky_1994_J.Physiol_477_497 |
PubMedSearch : Nikolsky_1994_J.Physiol_477_497 |
PubMedID: 7932237 |
Title : Functional role of cholinesterase in different types of neuro-muscular junction - |
Author(s) : Magazanik LG , Fedorov VV , Giniatullin RA , Nikolsky EE , Snetkov VA |
Ref : In: Cholinesterases, fundamental and applied aspects : proceedings of the Second International Meeting on Cholinesterases , (Brzin M, Barnard EA, Sket D, Eds) De Gruyter :229 , 1984 |
PubMedID: |