Report for Lapillo M

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References (4)

Title : Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors - Poli_2019_J.Enzyme.Inhib.Med.Chem_34_589
Author(s) : Poli G , Lapillo M , Jha V , Mouawad N , Caligiuri I , Macchia M , Minutolo F , Rizzolio F , Tuccinardi T , Granchi C
Ref : J Enzyme Inhib Med Chem , 34 :589 , 2019
Abstract : Poli_2019_J.Enzyme.Inhib.Med.Chem_34_589
ESTHER : Poli_2019_J.Enzyme.Inhib.Med.Chem_34_589
PubMedSearch : Poli_2019_J.Enzyme.Inhib.Med.Chem_34_589
PubMedID: 30696302
Gene_locus related to this paper: human-MGLL

Title : Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors - Bononi_2018_Eur.J.Med.Chem_157_817
Author(s) : Bononi G , Granchi C , Lapillo M , Giannotti M , Nieri D , Fortunato S , Boustani ME , Caligiuri I , Poli G , Carlson KE , Kim SH , Macchia M , Martinelli A , Rizzolio F , Chicca A , Katzenellenbogen JA , Minutolo F , Tuccinardi T
Ref : Eur Journal of Medicinal Chemistry , 157 :817 , 2018
Abstract : Bononi_2018_Eur.J.Med.Chem_157_817
ESTHER : Bononi_2018_Eur.J.Med.Chem_157_817
PubMedSearch : Bononi_2018_Eur.J.Med.Chem_157_817
PubMedID: 30144699

Title : Polypharmacological profile of 1,2-dihydro-2-oxo-pyridine-3-carboxamides in the endocannabinoid system - Chicca_2018_Eur.J.Med.Chem_154_155
Author(s) : Chicca A , Arena C , Bertini S , Gado F , Ciaglia E , Abate M , Digiacomo M , Lapillo M , Poli G , Bifulco M , Macchia M , Tuccinardi T , Gertsch J , Manera C
Ref : Eur Journal of Medicinal Chemistry , 154 :155 , 2018
Abstract : Chicca_2018_Eur.J.Med.Chem_154_155
ESTHER : Chicca_2018_Eur.J.Med.Chem_154_155
PubMedSearch : Chicca_2018_Eur.J.Med.Chem_154_155
PubMedID: 29793210

Title : Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors - Aghazadeh Tabrizi_2018_J.Med.Chem_61_1340
Author(s) : Aghazadeh Tabrizi M , Baraldi PG , Baraldi S , Ruggiero E , De Stefano L , Rizzolio F , Di Cesare Mannelli L , Ghelardini C , Chicca A , Lapillo M , Gertsch J , Manera C , Macchia M , Martinelli A , Granchi C , Minutolo F , Tuccinardi T
Ref : Journal of Medicinal Chemistry , 61 :1340 , 2018
Abstract : Aghazadeh Tabrizi_2018_J.Med.Chem_61_1340
ESTHER : Aghazadeh Tabrizi_2018_J.Med.Chem_61_1340
PubMedSearch : Aghazadeh Tabrizi_2018_J.Med.Chem_61_1340
PubMedID: 29309142