Report for Jeppesen L

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References (19)

Title : The muscarinic receptor agonist BuTAC, a novel potential antipsychotic, does not impair learning and memory in mouse passive avoidance - Rasmussen_2001_Schizophr.Res_49_193
Author(s) : Rasmussen T , Fink-Jensen A , Sauerberg P , Swedberg MD , Thomsen C , Sheardown MJ , Jeppesen L , Calligaro DO , DeLapp NW , Whitesitt CA , Ward JS , Shannon HE , Bymaster FP
Ref : Schizophr Res , 49 :193 , 2001
Abstract : Rasmussen_2001_Schizophr.Res_49_193
ESTHER : Rasmussen_2001_Schizophr.Res_49_193
PubMedSearch : Rasmussen_2001_Schizophr.Res_49_193
PubMedID: 11343877

Title : Synthesis and pharmacological evaluation of dimeric muscarinic acetylcholine receptor agonists - Christopoulos_2001_J.Pharmacol.Exp.Ther_298_1260
Author(s) : Christopoulos A , Grant MK , Ayoubzadeh N , Kim ON , Sauerberg P , Jeppesen L , El-Fakahany EE
Ref : Journal of Pharmacology & Experimental Therapeutics , 298 :1260 , 2001
Abstract : Christopoulos_2001_J.Pharmacol.Exp.Ther_298_1260
ESTHER : Christopoulos_2001_J.Pharmacol.Exp.Ther_298_1260
PubMedSearch : Christopoulos_2001_J.Pharmacol.Exp.Ther_298_1260
PubMedID: 11504829

Title : Xanomeline, an M(1)\/M(4) preferring muscarinic cholinergic receptor agonist, produces antipsychotic-like activity in rats and mice - Shannon_2000_Schizophr.Res_42_249
Author(s) : Shannon HE , Rasmussen K , Bymaster FP , Hart JC , Peters SC , Swedberg MD , Jeppesen L , Sheardown MJ , Sauerberg P , Fink-Jensen A
Ref : Schizophr Res , 42 :249 , 2000
Abstract : Shannon_2000_Schizophr.Res_42_249
ESTHER : Shannon_2000_Schizophr.Res_42_249
PubMedSearch : Shannon_2000_Schizophr.Res_42_249
PubMedID: 10785583

Title : Muscarinic receptor agonists decrease cocaine self-administration rates in drug-naive mice - Rasmussen_2000_Eur.J.Pharmacol_402_241
Author(s) : Rasmussen T , Sauerberg P , Nielsen EB , Swedberg MD , Thomsen C , Sheardown MJ , Jeppesen L , Calligaro DO , DeLapp NW , Whitesitt CA , Ward JS , Shannon HE , Bymaster FP , Fink-Jensen A
Ref : European Journal of Pharmacology , 402 :241 , 2000
Abstract : Rasmussen_2000_Eur.J.Pharmacol_402_241
ESTHER : Rasmussen_2000_Eur.J.Pharmacol_402_241
PubMedSearch : Rasmussen_2000_Eur.J.Pharmacol_402_241
PubMedID: 10958890

Title : Poster: Muscarinic receptor characterization and neurochemical effects of the antipsychotic-like muscarinic agonist PTAC -
Author(s) : Bymaster FP , Shannon HE , DeLapp NW , Calligaro DO , Perry KW , Zhang W , Rasmussen K , Ward JS , Fink-Jensen A , Olesen PH , Rasmussen T , Sheardown M , Swedberg MD , Jeppesen L , Sauerberg P
Ref : Life Sciences , 64 :579 , 1999
PubMedID:

Title : Poster: Behavioral and electrophysiological effects of the antipsychotic-like muscarinic agonist PTAC -
Author(s) : Shannon HE , Bymaster FP , Rasmussen K , DeLapp NW , Calligaro DO , Perry KW , Mitch CH , Ward JS , Fink-Jensen A , Olesen PH , Rasmussen T , Sheardown M , Swedberg MD , Jeppesen L , Sauerberg P
Ref : Life Sciences , 64 :587 , 1999
PubMedID:

Title : Potential role of muscarinic receptors in schizophrenia - Bymaster_1999_Life.Sci_64(6-7)_527
Author(s) : Bymaster FP , Shannon HE , Rasmussen K , DeLapp NW , Ward JS , Calligaro DO , Mitch CH , Whitesitt CA , Ludvigsen TS , Sheardown MJ , Swedberg MD , Rasmussen T , Olesen PH , Jeppesen L , Sauerberg P , Fink-Jensen A
Ref : Life Sciences , 64 :527 , 1999
Abstract : Bymaster_1999_Life.Sci_64(6-7)_527
ESTHER : Bymaster_1999_Life.Sci_64(6-7)_527
PubMedSearch : Bymaster_1999_Life.Sci_64(6-7)_527
PubMedID: 10069519

Title : Poster: Determination of the intrinsic functional muscarinic activity of xanomeline -
Author(s) : Falcone JF , Bymaster FP , Butler T , Thomsen C , Calligaro DO , Shannon HE , Whitesitt C , Ward J , Sheardown M , Fink-Jensen A , Jeppesen L , Sauerberg P , DeLapp NC
Ref : Life Sciences , 64 :579 , 1999
PubMedID:

Title : Muscarinic receptor agonists, like dopamine receptor antagonist antipsychotics, inhibit conditioned avoidance response in rats - Shannon_1999_J.Pharmacol.Exp.Ther_290_901
Author(s) : Shannon HE , Hart JC , Bymaster FP , Calligaro DO , DeLapp NW , Mitch CH , Ward JS , Fink-Jensen A , Sauerberg P , Jeppesen L , Sheardown MJ , Swedberg MD
Ref : Journal of Pharmacology & Experimental Therapeutics , 290 :901 , 1999
Abstract : Shannon_1999_J.Pharmacol.Exp.Ther_290_901
ESTHER : Shannon_1999_J.Pharmacol.Exp.Ther_290_901
PubMedSearch : Shannon_1999_J.Pharmacol.Exp.Ther_290_901
PubMedID: 10411607

Title : Poster: Muscarinic agonists with antipsychotic-like activity. Structure activity-relationships of 1,2,5-thiadiazole analogues with functioally dopamine antagonist activity -
Author(s) : Sauerberg P , Jeppesen L , Olesen PH , Rasmussen T , Swedberg MD , Sheardown MJ , Fink-Jensen A , Thomsen C , Thogersen H , Ward JS , Calligaro DO , DeLapp NW , Bymaster FP , Shannon HE
Ref : Life Sciences , 64 :555 , 1999
PubMedID:

Title : 1-(1,2,5-Thiadiazol-4-yl)-4-azatricyclo[2.2.1.0(2,6)]heptanes as new potent muscarinic M1 agonists: structure-activity relationship for 3-aryl-2-propyn-1-yloxy and 3-aryl-2-propyn-1-ylthio derivatives - Jeppesen_1999_J.Med.Chem_42_1999
Author(s) : Jeppesen L , Olesen PH , Hansen L , Sheardown MJ , Thomsen C , Rasmussen T , Jensen AF , Christensen MS , Rimvall K , Ward JS , Whitesitt CA , Calligaro DO , Bymaster FP , DeLapp NW , Felder CC , Shannon HE , Sauerberg P
Ref : Journal of Medicinal Chemistry , 42 :1999 , 1999
Abstract : Jeppesen_1999_J.Med.Chem_42_1999
ESTHER : Jeppesen_1999_J.Med.Chem_42_1999
PubMedSearch : Jeppesen_1999_J.Med.Chem_42_1999
PubMedID: 10354408

Title : Poster: New potent muscarinic 1,2,5-thiadiazole-azacycles and dimers hereof -
Author(s) : Jeppesen L , Sauerberg P , Olesen PH , Sheardown MJ , Thomsen C , Rasmussen T , Fink-Jensen A , Christensen MS , Ward JS , Whitesitt C , Calligaro DO , Bymaster FP , DeLapp NW , Felder CC , Shannon HE
Ref : Life Sciences , 64 :555 , 1999
PubMedID:

Title : Poster: Reversal of pertussis toxin-induced thermal allodynia by muscarinic cholinergic agonists in mice -
Author(s) : Zhang L , Shannon HE , Bymaster FP , DeLapp NW , Womer DE , Mitch CH , Ward JS , Olesen PH , Sheardown M , Swedberg MD , Jeppesen L , Sauerberg P
Ref : Life Sciences , 64 :587 , 1999
PubMedID:

Title : Muscarinic agonists with antipsychotic-like activity: structure-activity relationships of 1,2,5-thiadiazole analogues with functional dopamine antagonist activity - Sauerberg_1998_J.Med.Chem_41_4378
Author(s) : Sauerberg P , Jeppesen L , Olesen PH , Rasmussen T , Swedberg MD , Sheardown MJ , Fink-Jensen A , Thomsen C , Thogersen H , Rimvall K , Ward JS , Calligaro DO , DeLapp NW , Bymaster FP , Shannon HE
Ref : Journal of Medicinal Chemistry , 41 :4378 , 1998
Abstract : Sauerberg_1998_J.Med.Chem_41_4378
ESTHER : Sauerberg_1998_J.Med.Chem_41_4378
PubMedSearch : Sauerberg_1998_J.Med.Chem_41_4378
PubMedID: 9784113

Title : Identification of side chains on 1,2,5-thiadiazole-azacycles optimal for muscarinic m1 receptor activation - Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897
Author(s) : Sauerberg P , Jeppesen L , Olesen PH , Sheardown MJ , Fink-Jensen A , Rasmussen T , Rimvall K , Shannon HE , Bymaster FP , DeLapp NW , Calligaro DO , Ward JS , Whitesitt CA , Thomsen C
Ref : Bioorganic & Medicinal Chemistry Lett , 8 :2897 , 1998
Abstract : Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897
ESTHER : Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897
PubMedSearch : Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897
PubMedID: 9873644

Title : Xanomeline compared to other muscarinic agents on stimulation of phosphoinositide hydrolysis in vivo and other cholinomimetic effects - Bymaster_1998_Brain.Res_795_179
Author(s) : Bymaster FP , Carter PA , Peters SC , Zhang W , Ward JS , Mitch CH , Calligaro DO , Whitesitt CA , DeLapp NC , Shannon HE , Rimvall K , Jeppesen L , Sheardown MJ , Fink-Jensen A , Sauerberg P
Ref : Brain Research , 795 :179 , 1998
Abstract : Bymaster_1998_Brain.Res_795_179
ESTHER : Bymaster_1998_Brain.Res_795_179
PubMedSearch : Bymaster_1998_Brain.Res_795_179
PubMedID: 9622623

Title : 1,2,5-Thiadiazole analogues of aceclidine as potent m1 muscarinic agonists - Ward_1998_J.Med.Chem_41_379
Author(s) : Ward JS , Merritt L , Calligaro DO , Bymaster FP , Shannon HE , Mitch CH , Whitesitt CA , Brunsting D , Sheardown MJ , Olesen PH , Swedberg MD , Jeppesen L , Sauerberg P
Ref : Journal of Medicinal Chemistry , 41 :379 , 1998
Abstract : Ward_1998_J.Med.Chem_41_379
ESTHER : Ward_1998_J.Med.Chem_41_379
PubMedSearch : Ward_1998_J.Med.Chem_41_379
PubMedID: 9464368

Title : Muscarinic agonists exhibit functional dopamine antagonism in unilaterally 6-OHDA lesioned rats - Fink-Jensen_1998_Neuroreport_9_3481
Author(s) : Fink-Jensen A , Kristensen P , Shannon HE , Calligaro DO , DeLapp NW , Whitesitt CA , Ward JS , Thomsen C , Rasmusseen T , Sheardown MJ , Jeppesen L , Sauerberg P , Bymaster FP
Ref : Neuroreport , 9 :3481 , 1998
Abstract : Fink-Jensen_1998_Neuroreport_9_3481
ESTHER : Fink-Jensen_1998_Neuroreport_9_3481
PubMedSearch : Fink-Jensen_1998_Neuroreport_9_3481
PubMedID: 9855303

Title : Poster: Stimulation of phosphoinositide hydrolysis in vivo by xanomeline and other muscarinic agents -
Author(s) : Bymaster FP , Carter PA , Shannon HE , DeLapp NC , Whitesitt CA , Ward JS , Calligaro DO , Mitch CH , Sheardown MJ , Swedberg MD , Rimvall K , Fink-Jensen A , Jeppesen L , Sauerberg P
Ref : Life Sciences , 60 :1165 , 1997
PubMedID: