Hrabinova M

General

Full name : Hrabinova Martina

First name : Martina

Mail : University of Defence\; Faculty of Military Health Sciences, Department of Toxicology and Military Pharmacy,Trebeska 1575, 50001, Hradec Kralove

Zip Code :

City :

Country : Czech Republic

Email : martina.hrabinova@unob.cz

Phone :

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Website :

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References (79)

Title : Morphing cholinesterase inhibitor amiridine into multipotent drugs for the treatment of Alzheimer's disease - Mezeiova_2024_Biomed.Pharmacother_173_116399
Author(s) : Mezeiova E , Prchal L , Hrabinova M , Muckova L , Pulkrabkova L , Soukup O , Misiachna A , Janousek J , Fibigar J , Kucera T , Horak M , Makhaeva GF , Korabecny J
Ref : Biomed Pharmacother , 173 :116399 , 2024
Abstract : Mezeiova_2024_Biomed.Pharmacother_173_116399
ESTHER : Mezeiova_2024_Biomed.Pharmacother_173_116399
PubMedSearch : Mezeiova_2024_Biomed.Pharmacother_173_116399
PubMedID: 38492439

Title : A-series agent A-234: initial in vitro and in vivo characterization - Hrabinova_2024_Arch.Toxicol__
Author(s) : Hrabinova M , Pejchal J , Hepnarova V , Muckova L , Junova L , Opravil J , Zdarova Karasova J , Rozsypal T , Dlabkova A , Rehulkova H , Kucera T , Vecera Z , Caisberger F , Schmidt M , Soukup O , Jun D
Ref : Archives of Toxicology , : , 2024
Abstract : Hrabinova_2024_Arch.Toxicol__
ESTHER : Hrabinova_2024_Arch.Toxicol__
PubMedSearch : Hrabinova_2024_Arch.Toxicol__
PubMedID: 38446233

Title : Carltonine-Derived Compounds for Targeted Butyrylcholinesterase Inhibition - Pidany_2024_RSC.Med.Chem__
Author(s) : Pidany F , Kroustkova J , Jenco J , Breiterova K , Muckovab L , Novakova L , Kunes J , Fibigar J , Kucera T , Novak M , Sorf A , Hrabinova M , Pulkrabkova L , Janousek J , Soukup O , Jun D , Korabecny J , Cahlikova L
Ref : RSC Med Chem , : , 2024
Abstract : Pidany_2024_RSC.Med.Chem__
ESTHER : Pidany_2024_RSC.Med.Chem__
PubMedSearch : Pidany_2024_RSC.Med.Chem__
PubMedID:

Title : Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition - Misiachna_2024_Eur.J.Med.Chem_266_116130
Author(s) : Misiachna A , Svobodova B , Netolicky J , Chvojkova M , Kleteckova L , Prchal L , Novak M , Hrabinova M , Kucera T , Muckova L , Moravcova Z , Karasova JZ , Pejchal J , Blazek F , Malinak D , Hakenova K , Krausova BH , Kolcheva M , Ladislav M , Korabecny J , Pahnke J , Vales K , Horak M , Soukup O
Ref : Eur Journal of Medicinal Chemistry , 266 :116130 , 2024
Abstract : Misiachna_2024_Eur.J.Med.Chem_266_116130
ESTHER : Misiachna_2024_Eur.J.Med.Chem_266_116130
PubMedSearch : Misiachna_2024_Eur.J.Med.Chem_266_116130
PubMedID: 38218127

Title : Uncharged mono- and bisoximes: In search of a zwitterion to countermeasure organophosphorus intoxication - Gorecki_2024_Chem.Biol.Interact__110941
Author(s) : Gorecki L , Markova A , Hepnarova V , Zivna N , Junova L , Hrabinova M , Janousek J , Kobrlova T , Prchal L , Jun D , Soukup O , Horn G , Worek F , Marek J , Korabecny J
Ref : Chemico-Biological Interactions , :110941 , 2024
Abstract : Gorecki_2024_Chem.Biol.Interact__110941
ESTHER : Gorecki_2024_Chem.Biol.Interact__110941
PubMedSearch : Gorecki_2024_Chem.Biol.Interact__110941
PubMedID: 38493910

Title : A-agents, misleadingly known as Novichoks: a narrative review - Opravil_2023_Arch.Toxicol__
Author(s) : Opravil J , Pejchal J , Finger V , Korabecny J , Rozsypal T , Hrabinova M , Muckova L , Hepnarova V , Konecny J , Soukup O , Jun D
Ref : Archives of Toxicology , : , 2023
Abstract : Opravil_2023_Arch.Toxicol__
ESTHER : Opravil_2023_Arch.Toxicol__
PubMedSearch : Opravil_2023_Arch.Toxicol__
PubMedID: 37612377

Title : Highly selective butyrylcholinesterase inhibitors related to Amaryllidaceae alkaloids - Design, synthesis, and biological evaluation - Pidany_2023_Eur.J.Med.Chem_252_115301
Author(s) : Pidany F , Kroustkova J , Al Mamun A , Suchankova D , Brazzolotto X , Nachon F , Chantegreil F , Dolezal R , Pulkrabkova L , Muckova L , Hrabinova M , Finger V , Kufa M , Soukup O , Jun D , Jenco J , Kunes J , Novakova L , Korabecny J , Cahlikova L
Ref : Eur Journal of Medicinal Chemistry , 252 :115301 , 2023
Abstract : Pidany_2023_Eur.J.Med.Chem_252_115301
ESTHER : Pidany_2023_Eur.J.Med.Chem_252_115301
PubMedSearch : Pidany_2023_Eur.J.Med.Chem_252_115301
PubMedID: 36996715
Gene_locus related to this paper: human-BCHE

Title : Differentiated SH-SY5Y neuroblastoma cells as a model for evaluation of nerve agent-associated neurotoxicity - Pulkrabkova_2023_Arch.Toxicol__
Author(s) : Pulkrabkova L , Muckova L , Hrabinova M , Sorf A , Kobrlova T , Jost P , Bezdekova D , Korabecny J , Jun D , Soukup O
Ref : Archives of Toxicology , : , 2023
Abstract : Pulkrabkova_2023_Arch.Toxicol__
ESTHER : Pulkrabkova_2023_Arch.Toxicol__
PubMedSearch : Pulkrabkova_2023_Arch.Toxicol__
PubMedID: 37221426

Title : Structure-Guided Design of N-Methylpropargylamino-Quinazoline Derivatives as Multipotent Agents for the Treatment of Alzheimer's Disease - Svobodova_2023_Int.J.Mol.Sci_24_
Author(s) : Svobodova B , Pulkrabkova L , Panek D , Misiachna A , Kolcheva M , Andrys R , Handl J , Capek J , Nyvltova P , Rousar T , Prchal L , Hepnarova V , Hrabinova M , Muckova L , Tosnerova D , Karabanovich G , Finger V , Soukup O , Horak M , Korabecny J
Ref : Int J Mol Sci , 24 : , 2023
Abstract : Svobodova_2023_Int.J.Mol.Sci_24_
ESTHER : Svobodova_2023_Int.J.Mol.Sci_24_
PubMedSearch : Svobodova_2023_Int.J.Mol.Sci_24_
PubMedID: 37298087

Title : Non-covalent acetylcholinesterase inhibitors: In vitro screening and molecular modeling for novel selective insecticides - Hepnarova_2022_Toxicol.In.Vitro__105463
Author(s) : Hepnarova V , Hrabinova M , Muckova L , Kucera T , Schmidt M , Dolezal R , Gorecki L , Hrabcova V , Korabecny J , Mezeiova E , Jun D , Pejchal J
Ref : Toxicol In Vitro , :105463 , 2022
Abstract : Hepnarova_2022_Toxicol.In.Vitro__105463
ESTHER : Hepnarova_2022_Toxicol.In.Vitro__105463
PubMedSearch : Hepnarova_2022_Toxicol.In.Vitro__105463
PubMedID: 36041654

Title : Design and synthesis of novel tacrine-indole hybrids as potential multitarget-directed ligands for the treatment of Alzheimer's disease - Hamulakova_2021_Future.Med.Chem__
Author(s) : Hamulakova S , Kudlickova Z , Janovec L , Mezencev R , Deckner ZJ , Chernoff YO , Janockova J , Ihnatova V , Bzonek P , Novakova N , Hepnarova V , Hrabinova M , Jun D , Korabecny J , Soukup O , Kuca K
Ref : Future Med Chem , : , 2021
Abstract : Hamulakova_2021_Future.Med.Chem__
ESTHER : Hamulakova_2021_Future.Med.Chem__
PubMedSearch : Hamulakova_2021_Future.Med.Chem__
PubMedID: 33829876

Title : Huprine Y - tryptophan heterodimers with potential implication to Alzheimer's disease treatment - Mezeiova_2021_Bioorg.Med.Chem.Lett__128100
Author(s) : Mezeiova E , Hrabinova M , Hepnarova V , Jun D , Janockova J , Muckova L , Prchal L , Kristofikova Z , Kucera T , Gorecki L , Chalupova K , Kunes J , Hroudova J , Soukup O , Korabecny J
Ref : Bioorganic & Medicinal Chemistry Lett , :128100 , 2021
Abstract : Mezeiova_2021_Bioorg.Med.Chem.Lett__128100
ESTHER : Mezeiova_2021_Bioorg.Med.Chem.Lett__128100
PubMedSearch : Mezeiova_2021_Bioorg.Med.Chem.Lett__128100
PubMedID: 33984470

Title : Development of versatile and potent monoquaternary reactivators of acetylcholinesterase - Gorecki_2021_Arch.Toxicol__
Author(s) : Gorecki L , Hepnarova V , Karasova JZ , Hrabinova M , Courageux C , Dias J , Kucera T , Kobrlova T , Muckova L , Prchal L , Malinak D , Jun D , Musilek K , Worek F , Nachon F , Soukup O , Korabecny J
Ref : Archives of Toxicology , : , 2021
Abstract : Gorecki_2021_Arch.Toxicol__
ESTHER : Gorecki_2021_Arch.Toxicol__
PubMedSearch : Gorecki_2021_Arch.Toxicol__
PubMedID: 33517499

Title : Monoterpene indole alkaloids from Vinca minor L. (Apocynaceae): Identification of new structural scaffold for treatment of Alzheimer's disease - Vrabec_2021_Phytochemistry_194_113017
Author(s) : Vrabec R , Marikova J , Locarek M , Korabecny J , Hulcova D , Hosalkova A , Kunes J , Chlebek J , Kucera T , Hrabinova M , Jun D , Soukup O , Andrisano V , Jenco J , Safratova M , Novakova L , Opletal L , Cahlikova L
Ref : Phytochemistry , 194 :113017 , 2021
Abstract : Vrabec_2021_Phytochemistry_194_113017
ESTHER : Vrabec_2021_Phytochemistry_194_113017
PubMedSearch : Vrabec_2021_Phytochemistry_194_113017
PubMedID: 34798410

Title : Amaryllidaceae Alkaloids of Norbelladine-Type as Inspiration for Development of Highly Selective Butyrylcholinesterase Inhibitors: Synthesis, Biological Activity Evaluation, and Docking Studies - Al Mamun_2021_Int.J.Mol.Sci_22_
Author(s) : Al Mamun A , Pidany F , Hulcova D , Marikova J , Kucera T , Schmidt M , Catapano MC , Hrabinova M , Jun D , Muckova L , Kunes J , Janousek J , Andrys R , Novakova L , Perinova R , Maafi N , Soukup O , Korabecny J , Cahlikova L
Ref : Int J Mol Sci , 22 : , 2021
Abstract : Al Mamun_2021_Int.J.Mol.Sci_22_
ESTHER : Al Mamun_2021_Int.J.Mol.Sci_22_
PubMedSearch : Al Mamun_2021_Int.J.Mol.Sci_22_
PubMedID: 34361074

Title : Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease - Gorecki_2021_ACS.Chem.Neurosci__
Author(s) : Gorecki L , Uliassi E , Bartolini M , Janockova J , Hrabinova M , Hepnarova V , Prchal L , Muckova L , Pejchal J , Karasova JZ , Mezeiova E , Benkova M , Kobrlova T , Soukup O , Petralla S , Monti B , Korabecny J , Bolognesi ML
Ref : ACS Chem Neurosci , : , 2021
Abstract : Gorecki_2021_ACS.Chem.Neurosci__
ESTHER : Gorecki_2021_ACS.Chem.Neurosci__
PubMedSearch : Gorecki_2021_ACS.Chem.Neurosci__
PubMedID: 33852284

Title : Amaryllidaceae Alkaloids of Belladine-Type from Narcissus pseudonarcissus cv. Carlton as New Selective Inhibitors of Butyrylcholinesterase - Al Mamun_2020_Biomolecules_10_
Author(s) : Al Mamun A , Marikova J , Hulcova D , Janousek J , Safratova M , Novakova L , Kucera T , Hrabinova M , Kunes J , Korabecny J , Cahlikova L
Ref : Biomolecules , 10 : , 2020
Abstract : Al Mamun_2020_Biomolecules_10_
ESTHER : Al Mamun_2020_Biomolecules_10_
PubMedSearch : Al Mamun_2020_Biomolecules_10_
PubMedID: 32455879

Title : Discovery of novel berberine derivatives with balanced cholinesterase and prolyl oligopeptidase inhibition profile - Sobolova_2020_Eur.J.Med.Chem_203_112593
Author(s) : Sobolova K , Hrabinova M , Hepnarova V , Kucera T , Kobrlova T , Benkova M , Janockova J , Dolezal R , Prchal L , Benek O , Mezeiova E , Jun D , Soukup O , Korabecny J
Ref : Eur Journal of Medicinal Chemistry , 203 :112593 , 2020
Abstract : Sobolova_2020_Eur.J.Med.Chem_203_112593
ESTHER : Sobolova_2020_Eur.J.Med.Chem_203_112593
PubMedSearch : Sobolova_2020_Eur.J.Med.Chem_203_112593
PubMedID: 32688201

Title : Donepezil and Rivastigmine: Pharmacokinetic Profile and Brain-targeting After Intramuscular Administration in Rats - Karasova_2020_Iran.J.Pharm.Res_19_95
Author(s) : Karasova JZ , Hrabinova M , Krejciova M , Jun D , Kuca K
Ref : Iran J Pharm Res , 19 :95 , 2020
Abstract : Karasova_2020_Iran.J.Pharm.Res_19_95
ESTHER : Karasova_2020_Iran.J.Pharm.Res_19_95
PubMedSearch : Karasova_2020_Iran.J.Pharm.Res_19_95
PubMedID: 33680013

Title : Alkaloids of Zephyranthes citrina (Amaryllidaceae) and their implication to Alzheimer's disease: Isolation, structural elucidation and biological activity - Kohelova_2020_Bioorg.Chem_107_104567
Author(s) : Kohelova E , Marikova J , Korabecny J , Hulcova D , Kucera T , Jun D , Chlebek J , Jenco J , Safratova M , Hrabinova M , Ritomska A , Malanik M , Perinova R , Breiterova K , Kunes J , Novakova L , Opletal L , Cahlikova L
Ref : Bioorg Chem , 107 :104567 , 2020
Abstract : Kohelova_2020_Bioorg.Chem_107_104567
ESTHER : Kohelova_2020_Bioorg.Chem_107_104567
PubMedSearch : Kohelova_2020_Bioorg.Chem_107_104567
PubMedID: 33387730

Title : Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists - Konecny_2020_Biomolecules_11_
Author(s) : Konecny J , Misiachna A , Hrabinova M , Pulkrabkova L , Benkova M , Prchal L , Kucera T , Kobrlova T , Finger V , Kolcheva M , Kortus S , Jun D , Valko M , Horak M , Soukup O , Korabecny J
Ref : Biomolecules , 11 : , 2020
Abstract : Konecny_2020_Biomolecules_11_
ESTHER : Konecny_2020_Biomolecules_11_
PubMedSearch : Konecny_2020_Biomolecules_11_
PubMedID: 33375115

Title : Derivatives of the beta-Crinane Amaryllidaceae Alkaloid Haemanthamine as Multi-Target Directed Ligands for Alzheimer's Disease - Kohelova_2019_Molecules_24_
Author(s) : Kohelova E , Perinova R , Maafi N , Korabecny J , Hulcova D , Marikova J , Kucera T , Martinez Gonzalez L , Hrabinova M , Vorcakova K , Novakova L , De Simone A , Havelek R , Cahlikova L
Ref : Molecules , 24 : , 2019
Abstract : Kohelova_2019_Molecules_24_
ESTHER : Kohelova_2019_Molecules_24_
PubMedSearch : Kohelova_2019_Molecules_24_
PubMedID: 30987121

Title : Exploring Structure-Activity Relationship in Tacrine-Squaramide Derivatives as Potent Cholinesterase Inhibitors - Svobodova_2019_Biomolecules_9_
Author(s) : Svobodova B , Mezeiova E , Hepnarova V , Hrabinova M , Muckova L , Kobrlova T , Jun D , Soukup O , Jimeno ML , Marco-Contelles J , Korabecny J
Ref : Biomolecules , 9 : , 2019
Abstract : Svobodova_2019_Biomolecules_9_
ESTHER : Svobodova_2019_Biomolecules_9_
PubMedSearch : Svobodova_2019_Biomolecules_9_
PubMedID: 31430943

Title : In Vitro and In Silico Acetylcholinesterase Inhibitory Activity of Thalictricavine and Canadine and Their Predicted Penetration across the Blood-Brain Barrier - Chlebek_2019_Molecules_24_
Author(s) : Chlebek J , Korabecny J , Dolezal R , Stepankova S , Perez DI , Hostalkova A , Opletal L , Cahlikova L , Macakova K , Kucera T , Hrabinova M , Jun D
Ref : Molecules , 24 : , 2019
Abstract : Chlebek_2019_Molecules_24_
ESTHER : Chlebek_2019_Molecules_24_
PubMedSearch : Chlebek_2019_Molecules_24_
PubMedID: 30959739

Title : Tacrine and its 7-methoxy derivate\; time-change concentration in plasma and brain tissue and basic toxicological profile in rats - Karasova_2019_Drug.Chem.Toxicol__1
Author(s) : Karasova JZ , Soukup O , Korabecny J , Hroch M , Krejciova M , Hrabinova M , Misik J , Novotny L , Hepnarova V , Kuca K
Ref : Drug & Chemical Toxicology , :1 , 2019
Abstract : Karasova_2019_Drug.Chem.Toxicol__1
ESTHER : Karasova_2019_Drug.Chem.Toxicol__1
PubMedSearch : Karasova_2019_Drug.Chem.Toxicol__1
PubMedID: 31257938

Title : Pharmacological and toxicological in vitro and in vivo effect of higher doses of oxime reactivators - Hepnarova_2019_Toxicol.Appl.Pharmacol__114776
Author(s) : Hepnarova V , Muckova L , Ring A , Pejchal J , Herman D , Misik J , Hrabinova M , Jun D , Soukup O
Ref : Toxicol Appl Pharmacol , :114776 , 2019
Abstract : Hepnarova_2019_Toxicol.Appl.Pharmacol__114776
ESTHER : Hepnarova_2019_Toxicol.Appl.Pharmacol__114776
PubMedSearch : Hepnarova_2019_Toxicol.Appl.Pharmacol__114776
PubMedID: 31629733

Title : Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease - Chalupova_2019_Eur.J.Med.Chem_168_491
Author(s) : Chalupova K , Korabecny J , Bartolini M , Monti B , Lamba D , Caliandro R , Pesaresi A , Brazzolotto X , Gastellier AJ , Nachon F , Pejchal J , Jarosova M , Hepnarova V , Jun D , Hrabinova M , Dolezal R , Karasova JZ , Mzik M , Kristofikova Z , Misik J , Muckova L , Jost P , Soukup O , Benkova M , Setnicka V , Habartova L , Chvojkova M , Kleteckova L , Vales K , Mezeiova E , Uliassi E , Valis M , Nepovimova E , Bolognesi ML , Kuca K
Ref : Eur Journal of Medicinal Chemistry , 168 :491 , 2019
Abstract : Chalupova_2019_Eur.J.Med.Chem_168_491
ESTHER : Chalupova_2019_Eur.J.Med.Chem_168_491
PubMedSearch : Chalupova_2019_Eur.J.Med.Chem_168_491
PubMedID: 30851693
Gene_locus related to this paper: torca-ACHE

Title : In vitro and in silico Evaluation of Non-Quaternary Reactivators of AChE as Antidotes of Organophosphorus Poisoning - a New Hope or a Blind Alley? - Soukup_2018_Med.Chem_14_281
Author(s) : Soukup O , Korabecny J , Malinak D , Nepovimova E , Pham NL , Musilek K , Hrabinova M , Hepnarova V , Dolezal R , Pavek P , Jost P , Kobrlova T , Jankockova J , Gorecki L , Psotka M , Nguyen TD , Box K , Outhwaite B , Ceckova M , Sorf A , Jun D , Kuca K
Ref : Med Chem , 14 :281 , 2018
Abstract : Soukup_2018_Med.Chem_14_281
ESTHER : Soukup_2018_Med.Chem_14_281
PubMedSearch : Soukup_2018_Med.Chem_14_281
PubMedID: 29332594

Title : A newly developed oxime K203 is the most effective reactivator of tabun-inhibited acetylcholinesterase - Kuca_2018_BMC.Pharmacol.Toxicol_19_8
Author(s) : Kuca K , Musilek K , Jun D , Karasova JZ , Nepovimova E , Soukup O , Hrabinova M , Mikler J , Franca TCC , da Cunha EFF , de Castro AA , Valis M , Ramalho TC
Ref : BMC Pharmacol Toxicol , 19 :8 , 2018
Abstract : Kuca_2018_BMC.Pharmacol.Toxicol_19_8
ESTHER : Kuca_2018_BMC.Pharmacol.Toxicol_19_8
PubMedSearch : Kuca_2018_BMC.Pharmacol.Toxicol_19_8
PubMedID: 29467029

Title : Development of small bisquaternary cholinesterase inhibitors as drugs for pre-treatment of nerve agent poisonings - Kuca_2018_Drug.Des.Devel.Ther_12_505
Author(s) : Kuca K , Karasova JZ , Soukup O , Kassa J , Novotna E , Sepsova V , Horova A , Pejchal J , Hrabinova M , Vodakova E , Jun D , Nepovimova E , Valis M , Musilek K
Ref : Drug Des Devel Ther , 12 :505 , 2018
Abstract : Kuca_2018_Drug.Des.Devel.Ther_12_505
ESTHER : Kuca_2018_Drug.Des.Devel.Ther_12_505
PubMedSearch : Kuca_2018_Drug.Des.Devel.Ther_12_505
PubMedID: 29563775

Title : Synthesis, Biological Evaluation, and Docking Studies of Novel Bisquaternary Aldoxime Reactivators on Acetylcholinesterase and Butyrylcholinesterase Inhibited by Paraoxon - Kuca_2018_Molecules_23_
Author(s) : Kuca K , Jun D , Junova L , Musilek K , Hrabinova M , da Silva JAV , Ramalho TC , Valko M , Wu Q , Nepovimova E , Franca TCC
Ref : Molecules , 23 : , 2018
Abstract : Kuca_2018_Molecules_23_
ESTHER : Kuca_2018_Molecules_23_
PubMedSearch : Kuca_2018_Molecules_23_
PubMedID: 29735900

Title : Tacrine-coumarin and Tacrine-7-chloroquinoline Hybrids with Thiourea Linkers: Cholinesterase Inhibition Properties, Kinetic Study, Molecular Docking and Permeability Assay for Blood-brain Barrier - Hamulakova_2018_Curr.Alzheimer.Res_15_1096
Author(s) : Hamulakova S , Janovec L , Soukup O , Jun D , Janockova J , Hrabinova M , Sepsova V , Kuca K
Ref : Curr Alzheimer Res , 15 :1096 , 2018
Abstract : Hamulakova_2018_Curr.Alzheimer.Res_15_1096
ESTHER : Hamulakova_2018_Curr.Alzheimer.Res_15_1096
PubMedSearch : Hamulakova_2018_Curr.Alzheimer.Res_15_1096
PubMedID: 29992880

Title : Alkaloids from Narcissus poeticus cv. Pink Parasol of various structural types and their biological activity - Safratova_2018_Arch.Pharm.Res_41_208
Author(s) : Safratova M , Hostalkova A , Hulcova D , Breiterova K , Hrabcova V , Machado M , Fontinha D , Prudencio M , Kunes J , Chlebek J , Jun D , Hrabinova M , Novakova L , Havelek R , Seifrtova M , Opletal L , Cahlikova L
Ref : Arch Pharm Res , 41 :208 , 2018
Abstract : Safratova_2018_Arch.Pharm.Res_41_208
ESTHER : Safratova_2018_Arch.Pharm.Res_41_208
PubMedSearch : Safratova_2018_Arch.Pharm.Res_41_208
PubMedID: 29243039

Title : The concept of hybrid molecules of tacrine and benzyl quinolone carboxylic acid (BQCA) as multifunctional agents for Alzheimer's disease - Hepnarova_2018_Eur.J.Med.Chem_150_292
Author(s) : Hepnarova V , Korabecny J , Matouskova L , Jost P , Muckova L , Hrabinova M , Vykoukalova N , Kerhartova M , Kucera T , Dolezal R , Nepovimova E , Spilovska K , Mezeiova E , Pham NL , Jun D , Staud F , Kaping D , Kuca K , Soukup O
Ref : Eur Journal of Medicinal Chemistry , 150 :292 , 2018
Abstract : Hepnarova_2018_Eur.J.Med.Chem_150_292
ESTHER : Hepnarova_2018_Eur.J.Med.Chem_150_292
PubMedSearch : Hepnarova_2018_Eur.J.Med.Chem_150_292
PubMedID: 29533874

Title : Novel Tacrine-Scutellarin Hybrids as Multipotent Anti-Alzheimer's Agents: Design, Synthesis and Biological Evaluation - Spilovska_2017_Molecules_22_
Author(s) : Spilovska K , Korabecny J , Sepsova V , Jun D , Hrabinova M , Jost P , Muckova L , Soukup O , Janockova J , Kucera T , Dolezal R , Mezeiova E , Kaping D , Kuca K
Ref : Molecules , 22 : , 2017
Abstract : Spilovska_2017_Molecules_22_
ESTHER : Spilovska_2017_Molecules_22_
PubMedSearch : Spilovska_2017_Molecules_22_
PubMedID: 28621747

Title : Cholinesterase and Prolyl Oligopeptidase Inhibitory Activities of Alkaloids from Argemone platyceras (Papaveraceae) - Siatka_2017_Molecules_22_
Author(s) : Siatka T , Adamcova M , Opletal L , Cahlikova L , Jun D , Hrabinova M , Kunes J , Chlebek J
Ref : Molecules , 22 : , 2017
Abstract : Siatka_2017_Molecules_22_
ESTHER : Siatka_2017_Molecules_22_
PubMedSearch : Siatka_2017_Molecules_22_
PubMedID: 28708094

Title : Development of 2-Methoxyhuprine as Novel Lead for Alzheimer's Disease Therapy - Mezeiova_2017_Molecules_22_
Author(s) : Mezeiova E , Korabecny J , Sepsova V , Hrabinova M , Jost P , Muckova L , Kucera T , Dolezal R , Misik J , Spilovska K , Pham NL , Pokrievkova L , Roh J , Jun D , Soukup O , Kaping D , Kuca K
Ref : Molecules , 22 : , 2017
Abstract : Mezeiova_2017_Molecules_22_
ESTHER : Mezeiova_2017_Molecules_22_
PubMedSearch : Mezeiova_2017_Molecules_22_
PubMedID: 28788095

Title : Isoquinoline Alkaloids from Fumaria officinalis L. and Their Biological Activities Related to Alzheimer's Disease - Chlebek_2016_Chem.Biodivers_13_91
Author(s) : Chlebek J , Novak Z , Kassemova D , Safratova M , Kostelnik J , Maly L , Locarek M , Opletal L , Host'alkova A , Hrabinova M , Kunes J , Novotna P , Urbanova M , Novakova L , Macakova K , Hulcova D , Solich P , Perez Martin C , Jun D , Cahlikova L
Ref : Chem Biodivers , 13 :91 , 2016
Abstract : Chlebek_2016_Chem.Biodivers_13_91
ESTHER : Chlebek_2016_Chem.Biodivers_13_91
PubMedSearch : Chlebek_2016_Chem.Biodivers_13_91
PubMedID: 26765356

Title : Design, Synthesis and in vitro Evaluation of Indolotacrine Analogues as Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease - Benek_2016_ChemMedChem_11_1264
Author(s) : Benek O , Soukup O , Pasdiorova M , Hroch L , Sepsova V , Jost P , Hrabinova M , Jun D , Kuca K , Zala D , Ramsay RR , Marco-Contelles J , Musilek K
Ref : ChemMedChem , 11 :1264 , 2016
Abstract : Benek_2016_ChemMedChem_11_1264
ESTHER : Benek_2016_ChemMedChem_11_1264
PubMedSearch : Benek_2016_ChemMedChem_11_1264
PubMedID: 26427608

Title : Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease - Jerabek_2016_Eur.J.Med.Chem_127_250
Author(s) : Jerabek J , Uliassi E , Guidotti L , Korabecny J , Soukup O , Sepsova V , Hrabinova M , Kuca K , Bartolini M , Pena-Altamira LE , Petralla S , Monti B , Roberti M , Bolognesi ML
Ref : Eur Journal of Medicinal Chemistry , 127 :250 , 2016
Abstract : Jerabek_2016_Eur.J.Med.Chem_127_250
ESTHER : Jerabek_2016_Eur.J.Med.Chem_127_250
PubMedSearch : Jerabek_2016_Eur.J.Med.Chem_127_250
PubMedID: 28064079

Title : Targeting copper(II)-induced oxidative stress and the acetylcholinesterase system in Alzheimer's disease using multifunctional tacrine-coumarin hybrid molecules - Hamulakova_2016_J.Inorg.Biochem_161_52
Author(s) : Hamulakova S , Poprac P , Jomova K , Brezova V , Lauro P , Drostinova L , Jun D , Sepsova V , Hrabinova M , Soukup O , Kristian P , Gazova Z , Bednarikova Z , Kuca K , Valko M
Ref : J Inorg Biochem , 161 :52 , 2016
Abstract : Hamulakova_2016_J.Inorg.Biochem_161_52
ESTHER : Hamulakova_2016_J.Inorg.Biochem_161_52
PubMedSearch : Hamulakova_2016_J.Inorg.Biochem_161_52
PubMedID: 27230386

Title : Universality of Oxime K203 for Reactivation of Nerve Agent-Inhibited AChE - Kuca_2015_Med.Chem_11_683
Author(s) : Kuca K , Hrabinova M , Jun D , Musilek K , Penhaker M , Krejcar O , Soukup O
Ref : Med Chem , 11 :683 , 2015
Abstract : Kuca_2015_Med.Chem_11_683
ESTHER : Kuca_2015_Med.Chem_11_683
PubMedSearch : Kuca_2015_Med.Chem_11_683
PubMedID: 25845909

Title : Alkaloids from hydrastidis canadensis and their cholinesterase and prolyl oligopeptidase inhibitory -
Author(s) : Hostalkova A , Kunes J , Macakova K , Hrabinova M , Opletal L
Ref : Ceska a Slovenska Farmacie , 64 :41 , 2015
PubMedID: 26084651

Title : Tacrine-Trolox Hybrids: A Novel Class of Centrally Active, Nonhepatotoxic Multi-Target-Directed Ligands Exerting Anticholinesterase and Antioxidant Activities with Low In Vivo Toxicity - Nepovimova_2015_J.Med.Chem_58_8985
Author(s) : Nepovimova E , Korabecny J , Dolezal R , Babkova K , Ondrejicek A , Jun D , Sepsova V , Horova A , Hrabinova M , Soukup O , Bukum N , Jost P , Muckova L , Kassa J , Malinak D , Andrs M , Kuca K
Ref : Journal of Medicinal Chemistry , 58 :8985 , 2015
Abstract : Nepovimova_2015_J.Med.Chem_58_8985
ESTHER : Nepovimova_2015_J.Med.Chem_58_8985
PubMedSearch : Nepovimova_2015_J.Med.Chem_58_8985
PubMedID: 26503905

Title : 7-Methoxytacrine-p-Anisidine Hybrids as Novel Dual Binding Site Acetylcholinesterase Inhibitors for Alzheimer's Disease Treatment - Korabecny_2015_Molecules_20_22084
Author(s) : Korabecny J , Andrs M , Nepovimova E , Dolezal R , Babkova K , Horova A , Malinak D , Mezeiova E , Gorecki L , Sepsova V , Hrabinova M , Soukup O , Jun D , Kuca K
Ref : Molecules , 20 :22084 , 2015
Abstract : Korabecny_2015_Molecules_20_22084
ESTHER : Korabecny_2015_Molecules_20_22084
PubMedSearch : Korabecny_2015_Molecules_20_22084
PubMedID: 26690394

Title : (+)-Chenabinol (Revised NMR Data) and Two New Alkaloids from Berberis vulgaris and their Biological Activity - Novak_2015_Nat.Prod.Commun_10_1695
Author(s) : Novak Z , Host'alkova A , Opletal L , Novakova L , Hrabinova M , Kunes J , Cahlikova L
Ref : Nat Prod Commun , 10 :1695 , 2015
Abstract : Novak_2015_Nat.Prod.Commun_10_1695
ESTHER : Novak_2015_Nat.Prod.Commun_10_1695
PubMedSearch : Novak_2015_Nat.Prod.Commun_10_1695
PubMedID: 26669104

Title : Alkaloids from Peumus boldus and their acetylcholinesterase, butyrylcholinesterase and prolyl oligopeptidase inhibition activity - Host'alkova_2015_Nat.Prod.Commun_10_577
Author(s) : Host'alkova A , Opletal L , Kunes J , Novak Z , Hrabinova M , Chlebek J , Cegan L , Cahlikova L
Ref : Nat Prod Commun , 10 :577 , 2015
Abstract : Host'alkova_2015_Nat.Prod.Commun_10_577
ESTHER : Host'alkova_2015_Nat.Prod.Commun_10_577
PubMedSearch : Host'alkova_2015_Nat.Prod.Commun_10_577
PubMedID: 25973480

Title : Impact of tacrine and 7-methoxytacrine on gastric myoelectrical activity assessed using electrogastrography in experimental pigs - Bures_2015_Neuro.Endocrinol.Lett_36_
Author(s) : Bures J , Jun D , Hrabinova M , Tacheci I , Kvetina J , Pavlik M , Rejchrt S , Douda T , Kunes M , Kuca K , Kopacova M
Ref : Neuro Endocrinol Lett , 36 : , 2015
Abstract : Bures_2015_Neuro.Endocrinol.Lett_36_
ESTHER : Bures_2015_Neuro.Endocrinol.Lett_36_
PubMedSearch : Bures_2015_Neuro.Endocrinol.Lett_36_
PubMedID: 26757120

Title : Synthesis and biological evaluation of novel tacrine derivatives and tacrine-coumarin hybrids as cholinesterase inhibitors - Hamulakova_2014_J.Med.Chem_57_7073
Author(s) : Hamulakova S , Janovec L , Hrabinova M , Spilovska K , Korabecny J , Kristian P , Kuca K , Imrich J
Ref : Journal of Medicinal Chemistry , 57 :7073 , 2014
Abstract : Hamulakova_2014_J.Med.Chem_57_7073
ESTHER : Hamulakova_2014_J.Med.Chem_57_7073
PubMedSearch : Hamulakova_2014_J.Med.Chem_57_7073
PubMedID: 25089370

Title : Chemical composition of bioactive alkaloid extracts from some Narcissus species and varieties and their biological activity - Havlasova_2014_Nat.Prod.Commun_9_1151
Author(s) : Havlasova J , Safratova M , Siatka T , Stepankova S , Novak Z , Locarek M , Opletal L , Hrabinova M , Jun D , Benesova N , Kunes J , Cahlikova L
Ref : Nat Prod Commun , 9 :1151 , 2014
Abstract : Havlasova_2014_Nat.Prod.Commun_9_1151
ESTHER : Havlasova_2014_Nat.Prod.Commun_9_1151
PubMedSearch : Havlasova_2014_Nat.Prod.Commun_9_1151
PubMedID: 25233595

Title : Revised NMR data for 9-O-demethylgalanthine: an alkaloid from Zephyranthes robusta (Amaryllidaceae) and its biological activity - Safratova_2014_Nat.Prod.Commun_9_787
Author(s) : Safratova M , Novak Z , Kulhankova A , Kunes J , Hrabinova M , Jun D , Macakova K , Opletal L , Cahlikova L
Ref : Nat Prod Commun , 9 :787 , 2014
Abstract : Safratova_2014_Nat.Prod.Commun_9_787
ESTHER : Safratova_2014_Nat.Prod.Commun_9_787
PubMedSearch : Safratova_2014_Nat.Prod.Commun_9_787
PubMedID: 25115079

Title : Impact of paraoxon followed by acetylcholinesterase reactivator HI-6 on gastric myoelectric activity in experimental pigs - Bures_2013_Neuro.Endocrinol.Lett_34_79
Author(s) : Bures J , Kvetina J , Pavlik M , Kunes M , Kopacova M , Rejchrt S , Jun D , Hrabinova M , Kuca K , Tacheci I
Ref : Neuro Endocrinol Lett , 34 :79 , 2013
Abstract : Bures_2013_Neuro.Endocrinol.Lett_34_79
ESTHER : Bures_2013_Neuro.Endocrinol.Lett_34_79
PubMedSearch : Bures_2013_Neuro.Endocrinol.Lett_34_79
PubMedID: 24362097

Title : Preparation, in vitro evaluation and molecular modelling of pyridinium-quinolinium\/isoquinolinium non-symmetrical bisquaternary cholinesterase inhibitors - Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
Author(s) : Komloova M , Horova A , Hrabinova M , Jun D , Dolezal M , Vinsova J , Kuca K , Musilek K
Ref : Bioorganic & Medicinal Chemistry Lett , 23 :6663 , 2013
Abstract : Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
ESTHER : Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
PubMedSearch : Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
PubMedID: 24220173

Title : Structure-activity relationship for the reactivators of acetylcholinesterase inhibited by nerve agent VX - Kuca_2013_Med.Chem_9_689
Author(s) : Kuca K , Musilek K , Jun D , Karasova J , Soukup O , Pejchal J , Hrabinova M
Ref : Med Chem , 9 :689 , 2013
Abstract : Kuca_2013_Med.Chem_9_689
ESTHER : Kuca_2013_Med.Chem_9_689
PubMedSearch : Kuca_2013_Med.Chem_9_689
PubMedID: 22779796

Title : Alkaloids from Chlidanthus fragrans and their acetylcholinesterase, butyrylcholinesterase and prolyl oligopeptidase activities - Cahlikova_2013_Nat.Prod.Commun_8_1541
Author(s) : Cahlikova L , Hrabinova M , Kulhankova A , Benesova N , Chlebek J , Jun D , Novak Z , Macakova K , Kunes J , Kuca K , Opletal L
Ref : Nat Prod Commun , 8 :1541 , 2013
Abstract : Cahlikova_2013_Nat.Prod.Commun_8_1541
ESTHER : Cahlikova_2013_Nat.Prod.Commun_8_1541
PubMedSearch : Cahlikova_2013_Nat.Prod.Commun_8_1541
PubMedID: 24427936

Title : Synthesis, design and biological evaluation of novel highly potent tacrine congeners for the treatment of Alzheimer's disease - Hamulakova_2012_Eur.J.Med.Chem_55_23
Author(s) : Hamulakova S , Janovec L , Hrabinova M , Kristian P , Kuca K , Banasova M , Imrich J
Ref : Eur Journal of Medicinal Chemistry , 55 :23 , 2012
Abstract : Hamulakova_2012_Eur.J.Med.Chem_55_23
ESTHER : Hamulakova_2012_Eur.J.Med.Chem_55_23
PubMedSearch : Hamulakova_2012_Eur.J.Med.Chem_55_23
PubMedID: 22818849

Title : Preparation, in vitro screening and molecular modelling of symmetrical 4-tert-butylpyridinium cholinesterase inhibitors--analogues of SAD-128 - Musilek_2011_Bioorg.Med.Chem.Lett_21_150
Author(s) : Musilek K , Roder J , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Opletalova V , Kuca K , Jung YS
Ref : Bioorganic & Medicinal Chemistry Lett , 21 :150 , 2011
Abstract : Musilek_2011_Bioorg.Med.Chem.Lett_21_150
ESTHER : Musilek_2011_Bioorg.Med.Chem.Lett_21_150
PubMedSearch : Musilek_2011_Bioorg.Med.Chem.Lett_21_150
PubMedID: 21144749

Title : On the universality of oxime Hl-7 - antidote for case of the nerve agent poisoning - Kuca_2011_Mil.Med.Sci.Lett_80_80
Author(s) : Kuca K , Musilek K , Karasova J , Jun D , Soukup O , Pohanka M , Ghosh KK , Hrabinova M
Ref : Military Medical Science Letters , 80 :80 , 2011
Abstract : Kuca_2011_Mil.Med.Sci.Lett_80_80
ESTHER : Kuca_2011_Mil.Med.Sci.Lett_80_80
PubMedSearch : Kuca_2011_Mil.Med.Sci.Lett_80_80
PubMedID:

Title : Assessment of acetylcholinesterase activity using indoxylacetate and comparison with the standard Ellman's method - Pohanka_2011_Int.J.Mol.Sci_12_2631
Author(s) : Pohanka M , Hrabinova M , Kuca K , Simonato JP
Ref : Int J Mol Sci , 12 :2631 , 2011
Abstract : Pohanka_2011_Int.J.Mol.Sci_12_2631
ESTHER : Pohanka_2011_Int.J.Mol.Sci_12_2631
PubMedSearch : Pohanka_2011_Int.J.Mol.Sci_12_2631
PubMedID: 21731462

Title : Preparation and in vitro screening of symmetrical bis-isoquinolinium cholinesterase inhibitors bearing various connecting linkage--implications for early Myasthenia gravis treatment - Musilek_2011_Eur.J.Med.Chem_46_811
Author(s) : Musilek K , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Nachon F , Dolezal M , Kuca K
Ref : Eur Journal of Medicinal Chemistry , 46 :811 , 2011
Abstract : Musilek_2011_Eur.J.Med.Chem_46_811
ESTHER : Musilek_2011_Eur.J.Med.Chem_46_811
PubMedSearch : Musilek_2011_Eur.J.Med.Chem_46_811
PubMedID: 21236521

Title : The preparation, in vitro screening and molecular docking of symmetrical bisquaternary cholinesterase inhibitors containing a but-(2E)-en-1,4-diyl connecting linkage - Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
Author(s) : Musilek K , Pavlikova R , Marek J , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Dolezal M , Gunn-Moore F , Kuca K
Ref : J Enzyme Inhib Med Chem , 26 :245 , 2011
Abstract : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
ESTHER : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
PubMedSearch : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
PubMedID: 21406034

Title : Preparation and in vitro screening of symmetrical bispyridinium cholinesterase inhibitors bearing different connecting linkage-initial study for Myasthenia gravis implications - Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
Author(s) : Musilek K , Komloova M , Zavadova V , Holas O , Hrabinova M , Pohanka M , Dohnal V , Nachon F , Dolezal M , Kuca K , Jung YS
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :1763 , 2010
Abstract : Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
ESTHER : Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
PubMedSearch : Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
PubMedID: 20138518

Title : Oxime K027: novel low-toxic candidate for the universal reactivator of nerve agent- and pesticide-inhibited acetylcholinesterase - Kuca_2010_J.Enzyme.Inhib.Med.Chem_25_509
Author(s) : Kuca K , Musilek K , Jun D , Pohanka M , Ghosh KK , Hrabinova M
Ref : J Enzyme Inhib Med Chem , 25 :509 , 2010
Abstract : Kuca_2010_J.Enzyme.Inhib.Med.Chem_25_509
ESTHER : Kuca_2010_J.Enzyme.Inhib.Med.Chem_25_509
PubMedSearch : Kuca_2010_J.Enzyme.Inhib.Med.Chem_25_509
PubMedID: 20192902

Title : Pralidoxime--the gold standard of acetylcholinesterase reactivators--reactivation in vitro efficacy - Kuca_2010_Bratisl.Lek.Listy_111_502
Author(s) : Kuca K , Hrabinova M , Soukup O , Tobin G , Karasova J , Pohanka M
Ref : Bratislavske Lekarske Listy , 111 :502 , 2010
Abstract : Kuca_2010_Bratisl.Lek.Listy_111_502
ESTHER : Kuca_2010_Bratisl.Lek.Listy_111_502
PubMedSearch : Kuca_2010_Bratisl.Lek.Listy_111_502
PubMedID: 21180265

Title : Testing of a Referential Method Based on Indoxylacetate as a Acetylcholinesterase Substrate for Identification of Reactivation Efficacy. - Pohanka_2010_Mil.Med.Sci.Lett_79_111
Author(s) : Pohanka M , Hrabinova M , Karasova JZ , Holas O , Kuca K , Cabal J
Ref : Military Medical Science Letters , 79 :111 , 2010
Abstract : Pohanka_2010_Mil.Med.Sci.Lett_79_111
ESTHER : Pohanka_2010_Mil.Med.Sci.Lett_79_111
PubMedSearch : Pohanka_2010_Mil.Med.Sci.Lett_79_111
PubMedID:

Title : Reactivation of human brain homogenate cholinesterases inhibited by Tabun using newly developed oximes K117 and K127 - Kuca_2009_Basic.Clin.Pharmacol.Toxicol_105_207
Author(s) : Kuca K , Cabal J , Jung YS , Musilek K , Soukup O , Jun D , Pohanka M , Musilova L , Karasova J , Novotny L , Hrabinova M
Ref : Basic Clin Pharmacol Toxicol , 105 :207 , 2009
Abstract : Kuca_2009_Basic.Clin.Pharmacol.Toxicol_105_207
ESTHER : Kuca_2009_Basic.Clin.Pharmacol.Toxicol_105_207
PubMedSearch : Kuca_2009_Basic.Clin.Pharmacol.Toxicol_105_207
PubMedID: 19473310

Title : Novel bisquaternary oximes--reactivation of acetylcholinesterase and butyrylcholinesterase inhibited by paraoxon - Kuca_2009_Molecules_14_4915
Author(s) : Kuca K , Musilova L , Palecek J , Cirkva V , Paar M , Musilek K , Hrabinova M , Pohanka M , Karasova JZ , Jun D
Ref : Molecules , 14 :4915 , 2009
Abstract : Kuca_2009_Molecules_14_4915
ESTHER : Kuca_2009_Molecules_14_4915
PubMedSearch : Kuca_2009_Molecules_14_4915
PubMedID: 20032868

Title : Diagnosis of Intoxication by the Organophosphate VX: Comparison Between an Electrochemical Sensor and Ellman s Photometric Method - Pohanka_2008_Sensors.(Basel)_8_5229
Author(s) : Pohanka M , Hrabinova M , Kuca K
Ref : Sensors (Basel) , 8 :5229 , 2008
Abstract : Pohanka_2008_Sensors.(Basel)_8_5229
ESTHER : Pohanka_2008_Sensors.(Basel)_8_5229
PubMedSearch : Pohanka_2008_Sensors.(Basel)_8_5229
PubMedID: 27873811

Title : Potency of five structurally different acetylcholinesterase reactivators to reactivate human brain cholinesterases inhibited by cyclosarin - Kuca_2007_Clin.Toxicol.(Phila)_45_512
Author(s) : Kuca K , Cabal J , Jun D , Hrabinova M
Ref : Clinical Toxicology (Phila) , 45 :512 , 2007
Abstract : Kuca_2007_Clin.Toxicol.(Phila)_45_512
ESTHER : Kuca_2007_Clin.Toxicol.(Phila)_45_512
PubMedSearch : Kuca_2007_Clin.Toxicol.(Phila)_45_512
PubMedID: 17503257

Title : Targeted synthesis of 1-(4-hydroxyiminomethylpyridinium)-3-pyridiniumpropane dibromide--a new nerve agent reactivator - Kuca_2007_Molecules_12_1964
Author(s) : Kuca K , Musilek K , Paar M , Jun D , Stodulka P , Hrabinova M , Marek J
Ref : Molecules , 12 :1964 , 2007
Abstract : Kuca_2007_Molecules_12_1964
ESTHER : Kuca_2007_Molecules_12_1964
PubMedSearch : Kuca_2007_Molecules_12_1964
PubMedID: 17960099

Title : In vitro evaluation of acetylcholinesterase reactivators as potential antidotes against tabun nerve agent poisonings - Kuca_2006_Drug.Chem.Toxicol_29_443
Author(s) : Kuca K , Cabal J , Jun D , Hrabinova M
Ref : Drug & Chemical Toxicology , 29 :443 , 2006
Abstract : Kuca_2006_Drug.Chem.Toxicol_29_443
ESTHER : Kuca_2006_Drug.Chem.Toxicol_29_443
PubMedSearch : Kuca_2006_Drug.Chem.Toxicol_29_443
PubMedID: 16931445

Title : Russian VX: inhibition and reactivation of acetylcholinesterase compared with VX agent - Kuca_2006_Basic.Clin.Pharmacol.Toxicol_98_389
Author(s) : Kuca K , Jun D , Cabal J , Hrabinova M , Bartosova L , Opletalova V
Ref : Basic Clin Pharmacol Toxicol , 98 :389 , 2006
Abstract : Kuca_2006_Basic.Clin.Pharmacol.Toxicol_98_389
ESTHER : Kuca_2006_Basic.Clin.Pharmacol.Toxicol_98_389
PubMedSearch : Kuca_2006_Basic.Clin.Pharmacol.Toxicol_98_389
PubMedID: 16623863

Title : Substituted monoquaternary oximes as reactivators of cyclosarin--and chlorpyrifos--inhibited acetylcholinesterase - Racakova_2006_Arh.Hig.Rada.Toksikol_57_387
Author(s) : Racakova V , Hrabinova M , Jun D , Kuca K
Ref : Arh Hig Rada Toksikol , 57 :387 , 2006
Abstract : Racakova_2006_Arh.Hig.Rada.Toksikol_57_387
ESTHER : Racakova_2006_Arh.Hig.Rada.Toksikol_57_387
PubMedSearch : Racakova_2006_Arh.Hig.Rada.Toksikol_57_387
PubMedID: 17265677

Title : Potency of new structurally different oximes to reactivate cyclosarin-inhibited human brain acetylcholinesterases - Kuca_2006_J.Enzyme.Inhib.Med.Chem_21_663
Author(s) : Kuca K , Cabal J , Jun D , Bajgar J , Hrabinova M
Ref : J Enzyme Inhib Med Chem , 21 :663 , 2006
Abstract : Kuca_2006_J.Enzyme.Inhib.Med.Chem_21_663
ESTHER : Kuca_2006_J.Enzyme.Inhib.Med.Chem_21_663
PubMedSearch : Kuca_2006_J.Enzyme.Inhib.Med.Chem_21_663
PubMedID: 17252938

Title : New group of xylene linker-containing acetylcholinesterase reactivators as antidotes against the nerve agent cyclosarin - Hrabinova_2006_J.Enzyme.Inhib.Med.Chem_21_515
Author(s) : Hrabinova M , Musilek K , Jun D , Kuca K
Ref : J Enzyme Inhib Med Chem , 21 :515 , 2006
Abstract : Hrabinova_2006_J.Enzyme.Inhib.Med.Chem_21_515
ESTHER : Hrabinova_2006_J.Enzyme.Inhib.Med.Chem_21_515
PubMedSearch : Hrabinova_2006_J.Enzyme.Inhib.Med.Chem_21_515
PubMedID: 17194020

Title : In vitro potency of H oximes (HI-6, HLo-7), the oxime BI-6, and currently used oximes (pralidoxime, obidoxime, trimedoxime) to reactivate nerve agent-inhibited rat brain acetylcholinesterase - Kuca_2006_J.Toxicol.Environ.Health.A_69_1431
Author(s) : Kuca K , Cabal J , Kassa J , Jun D , Hrabinova M
Ref : J Toxicol Environ Health A , 69 :1431 , 2006
Abstract : Kuca_2006_J.Toxicol.Environ.Health.A_69_1431
ESTHER : Kuca_2006_J.Toxicol.Environ.Health.A_69_1431
PubMedSearch : Kuca_2006_J.Toxicol.Environ.Health.A_69_1431
PubMedID: 16766478

Title : A comparison of the potency of the oxime HLo-7 and currently used oximes (HI-6, pralidoxime, obidoxime) to reactivate nerve agent-inhibited rat brain acetylcholinesterase by in vitro methods - Kuca_2005_Acta.Medica.(Hradec.Kralove)_48_81
Author(s) : Kuca K , Cabal J , Kassa J , Jun D , Hrabinova M
Ref : Acta Medica (Hradec Kralove) , 48 :81 , 2005
Abstract : Kuca_2005_Acta.Medica.(Hradec.Kralove)_48_81
ESTHER : Kuca_2005_Acta.Medica.(Hradec.Kralove)_48_81
PubMedSearch : Kuca_2005_Acta.Medica.(Hradec.Kralove)_48_81
PubMedID: 16259317

Title : [A comparison of the efficacy of the reactivators of acetylcholinesterase inhibited with tabun] - Cabal_2005_Ceska.Slov.Farm_54_192
Author(s) : Cabal J , Kuca K , Jun D , Bajgar J , Hrabinova M
Ref : Ceska a Slovenska Farmacie , 54 :192 , 2005
Abstract : Cabal_2005_Ceska.Slov.Farm_54_192
ESTHER : Cabal_2005_Ceska.Slov.Farm_54_192
PubMedSearch : Cabal_2005_Ceska.Slov.Farm_54_192
PubMedID: 16124202

Title : Comparison of in vitro potency of oximes (pralidoxime, obidoxime, HI-6) to reactivate sarin-inhibited acetylcholinesterase in various parts of pig brain - Kuca_2005_J.Appl.Toxicol_25_271
Author(s) : Kuca K , Cabal J , Kassa J , Jun D , Hrabinova M
Ref : J Appl Toxicol , 25 :271 , 2005
Abstract : Kuca_2005_J.Appl.Toxicol_25_271
ESTHER : Kuca_2005_J.Appl.Toxicol_25_271
PubMedSearch : Kuca_2005_J.Appl.Toxicol_25_271
PubMedID: 16021679