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| Title : Complete decomposition of poly(ethylene terephthalate) by crude PET hydrolytic enzyme produced in Pichia pastoris - Chen_2024_Chem.Eng.J_481_148418 |
| Author(s) : Chen CC , Li X , Min J , Zeng Z , Ning Z , He H , Long X , Niu D , Peng R , Liu X , Yang Y , Huang JW , Guo RT |
| Ref : Chemical Engineering Journal , 481 :148418 , 2024 |
| Abstract : Chen_2024_Chem.Eng.J_481_148418 |
| ESTHER : Chen_2024_Chem.Eng.J_481_148418 |
| PubMedSearch : Chen_2024_Chem.Eng.J_481_148418 |
| PubMedID: |
| Gene_locus related to this paper: idesa-peth |
| Title : Design of carboxymethylcellulose-conjugated polymeric prodrug micelles for enhanced in vivo performance of docetaxel - Liu_2023_Int.J.Biol.Macromol__127690 |
| Author(s) : Liu Z , Liu Y , Liu H , Lv R , Liu B , Zhao L , Yin T , Zhang Y , He H , Gou J , Tang X , Yang L , Gao S |
| Ref : Int J Biol Macromol , :127690 , 2023 |
| Abstract : Liu_2023_Int.J.Biol.Macromol__127690 |
| ESTHER : Liu_2023_Int.J.Biol.Macromol__127690 |
| PubMedSearch : Liu_2023_Int.J.Biol.Macromol__127690 |
| PubMedID: 37898254 |
| Title : Modulation of oxidative stress and gut microbiota by selenium-containing peptides from Cardamine enshiensis and structural-based characterization - Zhang_2022_Food.Chem_395_133547 |
| Author(s) : Zhang X , Jia L , He H , Yin H , Ming J , Hou T , Xiang J |
| Ref : Food Chem , 395 :133547 , 2022 |
| Abstract : Zhang_2022_Food.Chem_395_133547 |
| ESTHER : Zhang_2022_Food.Chem_395_133547 |
| PubMedSearch : Zhang_2022_Food.Chem_395_133547 |
| PubMedID: 35780669 |
| Title : Detoxification Gene Families at the Genome-Wide Level of Rhus Gall Aphid Schlechtendalia chinensis - He_2022_Genes.(Basel)_13_ |
| Author(s) : He H , Crabbe MJC , Ren Z |
| Ref : Genes (Basel) , 13 : , 2022 |
| Abstract : He_2022_Genes.(Basel)_13_ |
| ESTHER : He_2022_Genes.(Basel)_13_ |
| PubMedSearch : He_2022_Genes.(Basel)_13_ |
| PubMedID: 36140795 |
| Title : Signature of arylacetamide deacetylase expression is associated with prognosis and immune infiltration in ovarian cancer - Feng_2022_Obstet.Gynecol.Sci_65_52 |
| Author(s) : Feng J , He H |
| Ref : Obstet Gynecol Sci , 65 :52 , 2022 |
| Abstract : Feng_2022_Obstet.Gynecol.Sci_65_52 |
| ESTHER : Feng_2022_Obstet.Gynecol.Sci_65_52 |
| PubMedSearch : Feng_2022_Obstet.Gynecol.Sci_65_52 |
| PubMedID: 34902961 |
| Title : Characterization of a Novel Esterase Est33 From an Antarctic Bacterium: A Representative of a New Esterase Family - Liu_2022_Front.Microbiol_13_855658 |
| Author(s) : Liu X , Zhou M , Sun R , Xing S , Wu T , He H , Chen J , Bielicki JK |
| Ref : Front Microbiol , 13 :855658 , 2022 |
| Abstract : Liu_2022_Front.Microbiol_13_855658 |
| ESTHER : Liu_2022_Front.Microbiol_13_855658 |
| PubMedSearch : Liu_2022_Front.Microbiol_13_855658 |
| PubMedID: 35655995 |
| Gene_locus related to this paper: psesp-Est33 |
| Title : TRPV4 Regulates Soman-Induced Status Epilepticus and Secondary Brain Injury via NMDA Receptor and NLRP3 Inflammasome - Wang_2021_Neurosci.Bull__ |
| Author(s) : Wang S , He H , Long J , Sui X , Yang J , Lin G , Wang Q , Wang Y , Luo Y |
| Ref : Neurosci Bull , : , 2021 |
| Abstract : Wang_2021_Neurosci.Bull__ |
| ESTHER : Wang_2021_Neurosci.Bull__ |
| PubMedSearch : Wang_2021_Neurosci.Bull__ |
| PubMedID: 33761112 |
| Title : Identification and Biochemical Characterization of a Novel Hormone-Sensitive Lipase Family Esterase Est19 from the Antarctic Bacterium Pseudomonas sp. E2-15 - Liu_2021_Biomolecules_11_1552 |
| Author(s) : Liu X , Zhou M , Xing S , Wu T , He H , Bielicki JK , Chen J |
| Ref : Biomolecules , 11 :1552 , 2021 |
| Abstract : Liu_2021_Biomolecules_11_1552 |
| ESTHER : Liu_2021_Biomolecules_11_1552 |
| PubMedSearch : Liu_2021_Biomolecules_11_1552 |
| PubMedID: 34827549 |
| Gene_locus related to this paper: psesp-MT761613 |
| Title : Combined effects of polyethylene and organic contaminant on zebrafish (Danio rerio): Accumulation of 9-Nitroanthracene, biomarkers and intestinal microbiota - Zhang_2021_Environ.Pollut_277_116767 |
| Author(s) : Zhang J , Meng H , Kong X , Cheng X , Ma T , He H , Du W , Yang S , Li S , Zhang L |
| Ref : Environ Pollut , 277 :116767 , 2021 |
| Abstract : Zhang_2021_Environ.Pollut_277_116767 |
| ESTHER : Zhang_2021_Environ.Pollut_277_116767 |
| PubMedSearch : Zhang_2021_Environ.Pollut_277_116767 |
| PubMedID: 33640823 |
| Title : Preparation and properties of a dual-function cellulose nanofiber-based bionic biosensor for detecting silver ions and acetylcholinesterase - Wang_2021_J.Hazard.Mater_403_123921 |
| Author(s) : Wang L , Guo W , Zhu H , He H , Wang S |
| Ref : J Hazard Mater , 403 :123921 , 2021 |
| Abstract : Wang_2021_J.Hazard.Mater_403_123921 |
| ESTHER : Wang_2021_J.Hazard.Mater_403_123921 |
| PubMedSearch : Wang_2021_J.Hazard.Mater_403_123921 |
| PubMedID: 33264972 |
| Title : Mori Ramulus (Chin.Ph.)-the Dried Twigs of Morus alba L.\/Part 1: Discovery of Two Novel Coumarin Glycosides from the Anti-Hyperuricemic Ethanol Extract - Yao_2019_Molecules_24_ |
| Author(s) : Yao J , He H , Xue J , Wang J , Jin H , Wu J , Hu J , Wang R , Kuchta K |
| Ref : Molecules , 24 : , 2019 |
| Abstract : Yao_2019_Molecules_24_ |
| ESTHER : Yao_2019_Molecules_24_ |
| PubMedSearch : Yao_2019_Molecules_24_ |
| PubMedID: 30754654 |
| Title : Insecticide Resistance Status and Mechanisms of Anopheles sinensis (Diptera: Culicidae) in Wenzhou, an Important Coastal Port City in China - Chen_2019_J.Med.Entomol_56_803 |
| Author(s) : Chen S , Qin Q , Zhong D , Fang X , He H , Wang L , Dong L , Lin H , Zhang M , Cui L , Yan G |
| Ref : Journal of Medical Entomology , 56 :803 , 2019 |
| Abstract : Chen_2019_J.Med.Entomol_56_803 |
| ESTHER : Chen_2019_J.Med.Entomol_56_803 |
| PubMedSearch : Chen_2019_J.Med.Entomol_56_803 |
| PubMedID: 30715428 |
| Title : Z-Ligustilide Exerted Hormetic Effect on Growth and Detoxification Enzymes of Spodoptera litura Larvae - Yi_2018_Evid.Based.Complement.Alternat.Med_2018_7104513 |
| Author(s) : Yi Y , Dou G , Yu Z , He H , Wang C , Li L , Zhou J , Liu D , Shi J , Li G , Pang L , Yang N , Huang Q , Qi H |
| Ref : Evid Based Complement Alternat Med , 2018 :7104513 , 2018 |
| Abstract : Yi_2018_Evid.Based.Complement.Alternat.Med_2018_7104513 |
| ESTHER : Yi_2018_Evid.Based.Complement.Alternat.Med_2018_7104513 |
| PubMedSearch : Yi_2018_Evid.Based.Complement.Alternat.Med_2018_7104513 |
| PubMedID: 30057645 |
| Title : Influence of Randomly Inserted Feruloyl Esterase A on beta-Glucosidase Activity in Trichoderma reesei - Hou_2017_Appl.Biochem.Biotechnol_183_254 |
| Author(s) : Hou Y , Pan Y , Yan M , He H , Yang Q , Zhong Y |
| Ref : Appl Biochem Biotechnol , 183 :254 , 2017 |
| Abstract : Hou_2017_Appl.Biochem.Biotechnol_183_254 |
| ESTHER : Hou_2017_Appl.Biochem.Biotechnol_183_254 |
| PubMedSearch : Hou_2017_Appl.Biochem.Biotechnol_183_254 |
| PubMedID: 28236194 |
| Title : Characterization of Feruloyl Esterases Produced by the Four Lactobacillus Species: L. amylovorus, L. acidophilus, L. farciminis and L. fermentum, Isolated from Ensiled Corn Stover - Xu_2017_Front.Microbiol_8_941 |
| Author(s) : Xu Z , He H , Zhang S , Guo T , Kong J |
| Ref : Front Microbiol , 8 :941 , 2017 |
| Abstract : Xu_2017_Front.Microbiol_8_941 |
| ESTHER : Xu_2017_Front.Microbiol_8_941 |
| PubMedSearch : Xu_2017_Front.Microbiol_8_941 |
| PubMedID: 28626449 |
| Title : The discovery of novel 5,6,5- and 5,5,6-tricyclic pyrrolidines as potent and selective DPP-4 inhibitors - Cox_2016_Bioorg.Med.Chem.Lett_26_2622 |
| Author(s) : Cox JM , Chu HD , Kuethe JT , Gao YD , Scapin G , Eiermann G , He H , Li X , Lyons KA , Metzger J , Petrov A , Wu JK , Xu S , Sinha-Roy R , Weber AE , Biftu T |
| Ref : Bioorganic & Medicinal Chemistry Lett , 26 :2622 , 2016 |
| Abstract : Cox_2016_Bioorg.Med.Chem.Lett_26_2622 |
| ESTHER : Cox_2016_Bioorg.Med.Chem.Lett_26_2622 |
| PubMedSearch : Cox_2016_Bioorg.Med.Chem.Lett_26_2622 |
| PubMedID: 27106708 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Two nematicidal furocoumarins from Ficus carica L. leaves and their physiological effects on pine wood nematode (Bursaphelenchus xylophilus) - Guo_2015_Nat.Prod.Res__1 |
| Author(s) : Guo Q , Du G , He H , Xu H , Guo D , Li R |
| Ref : Nat Prod Res , :1 , 2015 |
| Abstract : Guo_2015_Nat.Prod.Res__1 |
| ESTHER : Guo_2015_Nat.Prod.Res__1 |
| PubMedSearch : Guo_2015_Nat.Prod.Res__1 |
| PubMedID: 26479900 |
| Title : Discovery of the lomaiviticin biosynthetic gene cluster in Salinispora pacifica - Janso_2014_Tetrahedron_70_4156 |
| Author(s) : Janso JE , Haltli BA , Eustaquio AS , Kulowski K , Waldman AJ , Zha L , Nakamura H , Bernan VS , He H , Carter GT , Koehn FE , Balskus EP |
| Ref : Tetrahedron , 70 :4156 , 2014 |
| Abstract : Janso_2014_Tetrahedron_70_4156 |
| ESTHER : Janso_2014_Tetrahedron_70_4156 |
| PubMedSearch : Janso_2014_Tetrahedron_70_4156 |
| PubMedID: 25045187 |
| Gene_locus related to this paper: 9actn-a0a059uc17 |
| Title : Leonurus japonicus Houtt.: ethnopharmacology, phytochemistry and pharmacology of an important traditional Chinese medicine - Shang_2014_J.Ethnopharmacol_152_14 |
| Author(s) : Shang X , Pan H , Wang X , He H , Li M |
| Ref : J Ethnopharmacol , 152 :14 , 2014 |
| Abstract : Shang_2014_J.Ethnopharmacol_152_14 |
| ESTHER : Shang_2014_J.Ethnopharmacol_152_14 |
| PubMedSearch : Shang_2014_J.Ethnopharmacol_152_14 |
| PubMedID: 24412548 |
| Title : Omarigliptin (MK-3102): a novel long-acting DPP-4 inhibitor for once-weekly treatment of type 2 diabetes - Biftu_2014_J.Med.Chem_57_3205 |
| Author(s) : Biftu T , Sinha-Roy R , Chen P , Qian X , Feng D , Kuethe JT , Scapin G , Gao YD , Yan Y , Krueger D , Bak A , Eiermann G , He J , Cox J , Hicks J , Lyons K , He H , Salituro G , Tong S , Patel S , Doss G , Petrov A , Wu J , Xu SS , Sewall C , Zhang X , Zhang B , Thornberry NA , Weber AE |
| Ref : Journal of Medicinal Chemistry , 57 :3205 , 2014 |
| Abstract : Biftu_2014_J.Med.Chem_57_3205 |
| ESTHER : Biftu_2014_J.Med.Chem_57_3205 |
| PubMedSearch : Biftu_2014_J.Med.Chem_57_3205 |
| PubMedID: 24660890 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Age-dependent loss of cholinergic neurons in learning and memory-related brain regions and impaired learning in SAMP8 mice with trigeminal nerve damage - He_2014_Neural.Regen.Res_9_1985 |
| Author(s) : He Y , Zhu J , Huang F , Qin L , Fan W , He H |
| Ref : Neural Regen Res , 9 :1985 , 2014 |
| Abstract : He_2014_Neural.Regen.Res_9_1985 |
| ESTHER : He_2014_Neural.Regen.Res_9_1985 |
| PubMedSearch : He_2014_Neural.Regen.Res_9_1985 |
| PubMedID: 25598781 |
| Title : Discovery and optimization of orally active cyclohexane-based prolylcarboxypeptidase (PrCP) inhibitors - Debenham_2013_Bioorg.Med.Chem.Lett_23_6228 |
| Author(s) : Debenham JS , Graham TH , Verras A , Zhang Y , Clements MJ , Kuethe JT , Madsen-Duggan C , Liu W , Bhatt UR , Chen D , Chen Q , Garcia-Calvo M , Geissler WM , He H , Li X , Lisnock J , Shen Z , Tong X , Tung EC , Wiltsie J , Xu S , Hale JJ , Pinto S , Shen DM |
| Ref : Bioorganic & Medicinal Chemistry Lett , 23 :6228 , 2013 |
| Abstract : Debenham_2013_Bioorg.Med.Chem.Lett_23_6228 |
| ESTHER : Debenham_2013_Bioorg.Med.Chem.Lett_23_6228 |
| PubMedSearch : Debenham_2013_Bioorg.Med.Chem.Lett_23_6228 |
| PubMedID: 24157366 |
| Title : The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors - Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
| Author(s) : Graham TH , Shen HC , Liu W , Xiong Y , Verras A , Bleasby K , Bhatt UR , Chabin RM , Chen D , Chen Q , Garcia-Calvo M , Geissler WM , He H , Lassman ME , Shen Z , Tong X , Tung EC , Xie D , Xu S , Colletti SL , Tata JR , Hale JJ , Pinto S , Shen DM |
| Ref : Bioorganic & Medicinal Chemistry Lett , 22 :658 , 2012 |
| Abstract : Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
| ESTHER : Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
| PubMedSearch : Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
| PubMedID: 22079761 |
| Gene_locus related to this paper: human-PRCP |
| Title : A survey of Rhipicephalus microplus populations for mutations associated with pyrethroid resistance - Chen_2009_J.Econ.Entomol_102_373 |
| Author(s) : Chen AC , He H , Temeyer KB , Jones S , Green P , Barker SC |
| Ref : J Econ Entomol , 102 :373 , 2009 |
| Abstract : Chen_2009_J.Econ.Entomol_102_373 |
| ESTHER : Chen_2009_J.Econ.Entomol_102_373 |
| PubMedSearch : Chen_2009_J.Econ.Entomol_102_373 |
| PubMedID: 19253657 |
| Title : Absorption, metabolism, and excretion of [14C]vildagliptin, a novel dipeptidyl peptidase 4 inhibitor, in humans - He_2009_Drug.Metab.Dispos_37_536 |
| Author(s) : He H , Tran P , Yin H , Smith H , Batard Y , Wang L , Einolf H , Gu H , Mangold JB , Fischer V , Howard D |
| Ref : Drug Metabolism & Disposition: The Biological Fate of Chemicals , 37 :536 , 2009 |
| Abstract : He_2009_Drug.Metab.Dispos_37_536 |
| ESTHER : He_2009_Drug.Metab.Dispos_37_536 |
| PubMedSearch : He_2009_Drug.Metab.Dispos_37_536 |
| PubMedID: 19074975 |
| Title : Disposition of vildagliptin, a novel dipeptidyl peptidase 4 inhibitor, in rats and dogs - He_2009_Drug.Metab.Dispos_37_545 |
| Author(s) : He H , Tran P , Yin H , Smith H , Flood D , Kramp R , Filipeck R , Fischer V , Howard D |
| Ref : Drug Metabolism & Disposition: The Biological Fate of Chemicals , 37 :545 , 2009 |
| Abstract : He_2009_Drug.Metab.Dispos_37_545 |
| ESTHER : He_2009_Drug.Metab.Dispos_37_545 |
| PubMedSearch : He_2009_Drug.Metab.Dispos_37_545 |
| PubMedID: 19074976 |
| Title : Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors - Edmondson_2009_Bioorg.Med.Chem.Lett_19_4097 |
| Author(s) : Edmondson SD , Mastracchio A , Cox JM , Eiermann GJ , He H , Lyons KA , Patel RA , Patel SB , Petrov A , Scapin G , Wu JK , Xu S , Zhu B , Thornberry NA , Roy RS , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 19 :4097 , 2009 |
| Abstract : Edmondson_2009_Bioorg.Med.Chem.Lett_19_4097 |
| ESTHER : Edmondson_2009_Bioorg.Med.Chem.Lett_19_4097 |
| PubMedSearch : Edmondson_2009_Bioorg.Med.Chem.Lett_19_4097 |
| PubMedID: 19539471 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Discovery of potent and selective dipeptidyl peptidase IV inhibitors derived from beta-aminoamides bearing subsituted triazolopiperazines - Kim_2008_J.Med.Chem_51_589 |
| Author(s) : Kim D , Kowalchick JE , Brockunier LL , Parmee ER , Eiermann GJ , Fisher MH , He H , Leiting B , Lyons K , Scapin G , Patel SB , Petrov A , Pryor KD , Roy RS , Wu JK , Zhang X , Wyvratt MJ , Zhang BB , Zhu L , Thornberry NA , Weber AE |
| Ref : Journal of Medicinal Chemistry , 51 :589 , 2008 |
| Abstract : Kim_2008_J.Med.Chem_51_589 |
| ESTHER : Kim_2008_J.Med.Chem_51_589 |
| PubMedSearch : Kim_2008_J.Med.Chem_51_589 |
| PubMedID: 18201067 |
| Title : Fluoroolefins as amide bond mimics in dipeptidyl peptidase IV inhibitors - Edmondson_2008_Bioorg.Med.Chem.Lett_18_2409 |
| Author(s) : Edmondson SD , Wei L , Xu J , Shang J , Xu S , Pang J , Chaudhary A , Dean DC , He H , Leiting B , Lyons KA , Patel RA , Patel SB , Scapin G , Wu JK , Beconi MG , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 18 :2409 , 2008 |
| Abstract : Edmondson_2008_Bioorg.Med.Chem.Lett_18_2409 |
| ESTHER : Edmondson_2008_Bioorg.Med.Chem.Lett_18_2409 |
| PubMedSearch : Edmondson_2008_Bioorg.Med.Chem.Lett_18_2409 |
| PubMedID: 18331795 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Imidazopiperidine amides as dipeptidyl peptidase IV inhibitors for the treatment of diabetes - Chen_2007_Bioorg.Med.Chem.Lett_17_5853 |
| Author(s) : Chen P , Caldwell CG , Mathvink RJ , Leiting B , Marsilio F , Patel RA , Wu JK , He H , Lyons KA , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :5853 , 2007 |
| Abstract : Chen_2007_Bioorg.Med.Chem.Lett_17_5853 |
| ESTHER : Chen_2007_Bioorg.Med.Chem.Lett_17_5853 |
| PubMedSearch : Chen_2007_Bioorg.Med.Chem.Lett_17_5853 |
| PubMedID: 17869513 |
| Title : Design, synthesis, and biological evaluation of triazolopiperazine-based beta-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors - Kowalchick_2007_Bioorg.Med.Chem.Lett_17_5934 |
| Author(s) : Kowalchick JE , Leiting B , Pryor KD , Marsilio F , Wu JK , He H , Lyons KA , Eiermann GJ , Petrov A , Scapin G , Patel RA , Thornberry NA , Weber AE , Kim D |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :5934 , 2007 |
| Abstract : Kowalchick_2007_Bioorg.Med.Chem.Lett_17_5934 |
| ESTHER : Kowalchick_2007_Bioorg.Med.Chem.Lett_17_5934 |
| PubMedSearch : Kowalchick_2007_Bioorg.Med.Chem.Lett_17_5934 |
| PubMedID: 17827003 |
| Gene_locus related to this paper: human-DPP4 |
| Title : 4-arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV - Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| Author(s) : Kaelin DE , Smenton AL , Eiermann GJ , He H , Leiting B , Lyons KA , Patel RA , Patel SB , Petrov A , Scapin G , Wu JK , Thornberry NA , Weber AE , Duffy JL |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :5806 , 2007 |
| Abstract : Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| ESTHER : Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| PubMedSearch : Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| PubMedID: 17851076 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Optimization of 1,4-diazepan-2-one containing dipeptidyl peptidase IV inhibitors for the treatment of type 2 diabetes - Liang_2007_Bioorg.Med.Chem.Lett_17_1903 |
| Author(s) : Liang GB , Qian X , Feng D , Biftu T , Eiermann G , He H , Leiting B , Lyons K , Petrov A , Sinha-Roy R , Zhang B , Wu J , Zhang X , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :1903 , 2007 |
| Abstract : Liang_2007_Bioorg.Med.Chem.Lett_17_1903 |
| ESTHER : Liang_2007_Bioorg.Med.Chem.Lett_17_1903 |
| PubMedSearch : Liang_2007_Bioorg.Med.Chem.Lett_17_1903 |
| PubMedID: 17291750 |
| Title : Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: close analogs of JANUVIA (sitagliptin phosphate) - Kim_2007_Bioorg.Med.Chem.Lett_17_3373 |
| Author(s) : Kim D , Kowalchick JE , Edmondson SD , Mastracchio A , Xu J , Eiermann GJ , Leiting B , Wu JK , Pryor KD , Patel RA , He H , Lyons KA , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :3373 , 2007 |
| Abstract : Kim_2007_Bioorg.Med.Chem.Lett_17_3373 |
| ESTHER : Kim_2007_Bioorg.Med.Chem.Lett_17_3373 |
| PubMedSearch : Kim_2007_Bioorg.Med.Chem.Lett_17_3373 |
| PubMedID: 17434732 |
| Title : (3R)-4-[(3R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoyl]-3-(2,2,2-trifluoroethyl)- 1,4-diazepan-2-one, a selective dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes - Biftu_2007_Bioorg.Med.Chem.Lett_17_49 |
| Author(s) : Biftu T , Feng D , Qian X , Liang GB , Kieczykowski G , Eiermann G , He H , Leiting B , Lyons K , Petrov A , Sinha-Roy R , Zhang B , Scapin G , Patel S , Gao YD , Singh S , Wu J , Zhang X , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :49 , 2007 |
| Abstract : Biftu_2007_Bioorg.Med.Chem.Lett_17_49 |
| ESTHER : Biftu_2007_Bioorg.Med.Chem.Lett_17_49 |
| PubMedSearch : Biftu_2007_Bioorg.Med.Chem.Lett_17_49 |
| PubMedID: 17055272 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Rational design of a novel, potent, and orally bioavailable cyclohexylamine DPP-4 inhibitor by application of molecular modeling and X-ray crystallography of sitagliptin - Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
| Author(s) : Biftu T , Scapin G , Singh S , Feng D , Becker JW , Eiermann G , He H , Lyons K , Patel S , Petrov A , Sinha-Roy R , Zhang B , Wu J , Zhang X , Doss GA , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :3384 , 2007 |
| Abstract : Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
| ESTHER : Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
| PubMedSearch : Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
| PubMedID: 17433672 |
| Gene_locus related to this paper: human-DPP4 |
| Title : 4-aminophenylalanine and 4-aminocyclohexylalanine derivatives as potent, selective, and orally bioavailable inhibitors of dipeptidyl peptidase IV - Duffy_2007_Bioorg.Med.Chem.Lett_17_2879 |
| Author(s) : Duffy JL , Kirk BA , Wang L , Eiermann GJ , He H , Leiting B , Lyons KA , Patel RA , Patel SB , Petrov A , Scapin G , Wu JK , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :2879 , 2007 |
| Abstract : Duffy_2007_Bioorg.Med.Chem.Lett_17_2879 |
| ESTHER : Duffy_2007_Bioorg.Med.Chem.Lett_17_2879 |
| PubMedSearch : Duffy_2007_Bioorg.Med.Chem.Lett_17_2879 |
| PubMedID: 17350841 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors - Cox_2007_Bioorg.Med.Chem.Lett_17_4579 |
| Author(s) : Cox JM , Harper B , Mastracchio A , Leiting B , Sinha Roy R , Patel RA , Wu JK , Lyons KA , He H , Xu S , Zhu B , Thornberry NA , Weber AE , Edmondson SD |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :4579 , 2007 |
| Abstract : Cox_2007_Bioorg.Med.Chem.Lett_17_4579 |
| ESTHER : Cox_2007_Bioorg.Med.Chem.Lett_17_4579 |
| PubMedSearch : Cox_2007_Bioorg.Med.Chem.Lett_17_4579 |
| PubMedID: 17562364 |
| Title : Discovery of potent, selective, and orally bioavailable oxadiazole-based dipeptidyl peptidase IV inhibitors - Xu_2006_Bioorg.Med.Chem.Lett_16_5373 |
| Author(s) : Xu J , Wei L , Mathvink RJ , Edmondson SD , Eiermann GJ , He H , Leone JF , Leiting B , Lyons KA , Marsilio F , Patel RA , Patel SB , Petrov A , Scapin G , Wu JK , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 16 :5373 , 2006 |
| Abstract : Xu_2006_Bioorg.Med.Chem.Lett_16_5373 |
| ESTHER : Xu_2006_Bioorg.Med.Chem.Lett_16_5373 |
| PubMedSearch : Xu_2006_Bioorg.Med.Chem.Lett_16_5373 |
| PubMedID: 16919457 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitors - Xu_2006_Bioorg.Med.Chem.Lett_16_1346 |
| Author(s) : Xu J , Wei L , Mathvink R , Edmondson SD , Mastracchio A , Eiermann GJ , He H , Leone JF , Leiting B , Lyons KA , Marsilio F , Patel RA , Petrov A , Wu JK , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 16 :1346 , 2006 |
| Abstract : Xu_2006_Bioorg.Med.Chem.Lett_16_1346 |
| ESTHER : Xu_2006_Bioorg.Med.Chem.Lett_16_1346 |
| PubMedSearch : Xu_2006_Bioorg.Med.Chem.Lett_16_1346 |
| PubMedID: 16332437 |
| Title : (2S,3S)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-N,N-dimethyl-4-oxo-2-(4-[1,2,4]tr iazolo[1,5-a]-pyridin-6-ylphenyl)butanamide: a selective alpha-amino amide dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes - Edmondson_2006_J.Med.Chem_49_3614 |
| Author(s) : Edmondson SD , Mastracchio A , Mathvink RJ , He J , Harper B , Park YJ , Beconi M , Di Salvo J , Eiermann GJ , He H , Leiting B , Leone JF , Levorse DA , Lyons K , Patel RA , Patel SB , Petrov A , Scapin G , Shang J , Roy RS , Smith A , Wu JK , Xu S , Zhu B , Thornberry NA , Weber AE |
| Ref : Journal of Medicinal Chemistry , 49 :3614 , 2006 |
| Abstract : Edmondson_2006_J.Med.Chem_49_3614 |
| ESTHER : Edmondson_2006_J.Med.Chem_49_3614 |
| PubMedSearch : Edmondson_2006_J.Med.Chem_49_3614 |
| PubMedID: 16759103 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors - Xu_2005_Bioorg.Med.Chem.Lett_15_2533 |
| Author(s) : Xu J , Wei L , Mathvink R , He J , Park YJ , He H , Leiting B , Lyons KA , Marsilio F , Patel RA , Wu JK , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :2533 , 2005 |
| Abstract : Xu_2005_Bioorg.Med.Chem.Lett_15_2533 |
| ESTHER : Xu_2005_Bioorg.Med.Chem.Lett_15_2533 |
| PubMedSearch : Xu_2005_Bioorg.Med.Chem.Lett_15_2533 |
| PubMedID: 15863311 |
| Title : Dipeptidyl peptidase IV inhibitors derived from beta-aminoacylpiperidines bearing a fused thiazole, oxazole, isoxazole, or pyrazole - Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
| Author(s) : Ashton WT , Sisco RM , Dong H , Lyons KA , He H , Doss GA , Leiting B , Patel RA , Wu JK , Marsilio F , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :2253 , 2005 |
| Abstract : Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
| ESTHER : Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
| PubMedSearch : Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
| PubMedID: 15837304 |
| Title : Dipeptidyl peptidase IV inhibition for the treatment of type 2 diabetes: potential importance of selectivity over dipeptidyl peptidases 8 and 9 - Lankas_2005_Diabetes_54_2988 |
| Author(s) : Lankas GR , Leiting B , Roy RS , Eiermann GJ , Beconi MG , Biftu T , Chan CC , Edmondson S , Feeney WP , He H , Ippolito DE , Kim D , Lyons KA , Ok HO , Patel RA , Petrov AN , Pryor KA , Qian X , Reigle L , Woods A , Wu JK , Zaller D , Zhang X , Zhu L , Weber AE , Thornberry NA |
| Ref : Diabetes , 54 :2988 , 2005 |
| Abstract : Lankas_2005_Diabetes_54_2988 |
| ESTHER : Lankas_2005_Diabetes_54_2988 |
| PubMedSearch : Lankas_2005_Diabetes_54_2988 |
| PubMedID: 16186403 |
| Title : (2R)-4-oxo-4-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin-7(8H)- yl]-1-(2,4,5-trifluorophenyl)butan-2-amine: a potent, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes - Kim_2005_J.Med.Chem_48_141 |
| Author(s) : Kim D , Wang L , Beconi M , Eiermann GJ , Fisher MH , He H , Hickey GJ , Kowalchick JE , Leiting B , Lyons K , Marsilio F , McCann ME , Patel RA , Petrov A , Scapin G , Patel SB , Roy RS , Wu JK , Wyvratt MJ , Zhang BB , Zhu L , Thornberry NA , Weber AE |
| Ref : Journal of Medicinal Chemistry , 48 :141 , 2005 |
| Abstract : Kim_2005_J.Med.Chem_48_141 |
| ESTHER : Kim_2005_J.Med.Chem_48_141 |
| PubMedSearch : Kim_2005_J.Med.Chem_48_141 |
| PubMedID: 15634008 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Discovery of potent and selective orally bioavailable beta-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors - Edmondson_2005_Bioorg.Med.Chem.Lett_15_3048 |
| Author(s) : Edmondson SD , Mastracchio A , Duffy JL , Eiermann GJ , He H , Ita I , Leiting B , Leone JF , Lyons KA , Makarewicz AM , Patel RA , Petrov A , Wu JK , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :3048 , 2005 |
| Abstract : Edmondson_2005_Bioorg.Med.Chem.Lett_15_3048 |
| ESTHER : Edmondson_2005_Bioorg.Med.Chem.Lett_15_3048 |
| PubMedSearch : Edmondson_2005_Bioorg.Med.Chem.Lett_15_3048 |
| PubMedID: 15908206 |
| Title : Potent and selective proline derived dipeptidyl peptidase IV inhibitors - Edmondson_2004_Bioorg.Med.Chem.Lett_14_5151 |
| Author(s) : Edmondson SD , Mastracchio A , Beconi M , Colwell LF, Jr. , Habulihaz B , He H , Kumar S , Leiting B , Lyons KA , Mao A , Marsilio F , Patel RA , Wu JK , Zhu L , Thornberry NA , Weber AE , Parmee ER |
| Ref : Bioorganic & Medicinal Chemistry Lett , 14 :5151 , 2004 |
| Abstract : Edmondson_2004_Bioorg.Med.Chem.Lett_14_5151 |
| ESTHER : Edmondson_2004_Bioorg.Med.Chem.Lett_14_5151 |
| PubMedSearch : Edmondson_2004_Bioorg.Med.Chem.Lett_14_5151 |
| PubMedID: 15380217 |
| Title : 4-Amino cyclohexylglycine analogues as potent dipeptidyl peptidase IV inhibitors - Parmee_2004_Bioorg.Med.Chem.Lett_14_43 |
| Author(s) : Parmee ER , He J , Mastracchio A , Edmondson SD , Colwell L , Eiermann G , Feeney WP , Habulihaz B , He H , Kilburn R , Leiting B , Lyons K , Marsilio F , Patel RA , Petrov A , Di Salvo J , Wu JK , Thornberry NA , Weber AE |
| Ref : Bioorganic & Medicinal Chemistry Lett , 14 :43 , 2004 |
| Abstract : Parmee_2004_Bioorg.Med.Chem.Lett_14_43 |
| ESTHER : Parmee_2004_Bioorg.Med.Chem.Lett_14_43 |
| PubMedSearch : Parmee_2004_Bioorg.Med.Chem.Lett_14_43 |
| PubMedID: 14684294 |
| Title : Identification of a point mutation in an esterase gene in different populations of the southern cattle tick, Boophilus microplus - Hernandez_2000_Insect.Biochem.Mol.Biol_30_969 |
| Author(s) : Hernandez R , He H , Chen AC , Waghela SD , Wayne Ivie G , George JE , Gale Wagner G |
| Ref : Insect Biochemistry & Molecular Biology , 30 :969 , 2000 |
| Abstract : Hernandez_2000_Insect.Biochem.Mol.Biol_30_969 |
| ESTHER : Hernandez_2000_Insect.Biochem.Mol.Biol_30_969 |
| PubMedSearch : Hernandez_2000_Insect.Biochem.Mol.Biol_30_969 |
| PubMedID: 10899463 |
| Gene_locus related to this paper: boomi-este08 , boomi-este13 |
| Title : Cloning and sequencing of a putative acetylcholinesterase cDNA from Boophilus microplus (Acari: Ixodidae) - Hernandez_1999_J.Med.Entomol_36_764 |
| Author(s) : Hernandez R , He H , Chen AC , Ivie GW , George JE , Wagner GG |
| Ref : Journal of Medical Entomology , 36 :764 , 1999 |
| Abstract : Hernandez_1999_J.Med.Entomol_36_764 |
| ESTHER : Hernandez_1999_J.Med.Entomol_36_764 |
| PubMedSearch : Hernandez_1999_J.Med.Entomol_36_764 |
| PubMedID: 10593078 |
| Gene_locus related to this paper: boomi-ACHE2 |