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Title : Design, Synthesis, and Evaluation of Reversible and Irreversible Monoacylglycerol Lipase Positron Emission Tomography (PET) Tracers Using a Tail Switching Strategy on a Piperazinyl Azetidine Skeleton - Chen_2019_J.Med.Chem_62_3336 |
Author(s) : Chen Z , Mori W , Deng X , Cheng R , Ogasawara D , Zhang G , Schafroth MA , Dahl K , Fu H , Hatori A , Shao T , Zhang Y , Yamasaki T , Zhang X , Rong J , Yu Q , Hu K , Fujinaga M , Xie L , Kumata K , Gou Y , Chen J , Gu S , Bao L , Wang L , Collier TL , Vasdev N , Shao Y , Ma JA , Cravatt BF , Fowler C , Josephson L , Zhang MR , Liang SH |
Ref : Journal of Medicinal Chemistry , 62 :3336 , 2019 |
Abstract : Chen_2019_J.Med.Chem_62_3336 |
ESTHER : Chen_2019_J.Med.Chem_62_3336 |
PubMedSearch : Chen_2019_J.Med.Chem_62_3336 |
PubMedID: 30829483 |
Gene_locus related to this paper: human-MGLL |
Title : In Vitro and in Vivo Evaluation of (11)C-Labeled Azetidinecarboxylates for Imaging Monoacylglycerol Lipase by PET Imaging Studies - Cheng_2018_J.Med.Chem_61_2278 |
Author(s) : Cheng R , Mori W , Ma L , Alhouayek M , Hatori A , Zhang Y , Ogasawara D , Yuan G , Chen Z , Zhang X , Shi H , Yamasaki T , Xie L , Kumata K , Fujinaga M , Nagai Y , Minamimoto T , Svensson M , Wang L , Du Y , Ondrechen MJ , Vasdev N , Cravatt BF , Fowler C , Zhang MR , Liang SH |
Ref : Journal of Medicinal Chemistry , 61 :2278 , 2018 |
Abstract : Cheng_2018_J.Med.Chem_61_2278 |
ESTHER : Cheng_2018_J.Med.Chem_61_2278 |
PubMedSearch : Cheng_2018_J.Med.Chem_61_2278 |
PubMedID: 29481079 |