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Title : Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes - Augeri_2005_J.Med.Chem_48_5025 |
Author(s) : Augeri DJ , Robl JA , Betebenner DA , Magnin DR , Khanna A , Robertson JG , Wang A , Simpkins LM , Taunk P , Huang Q , Han SP , Abboa-Offei B , Cap M , Xin L , Tao L , Tozzo E , Welzel GE , Egan DM , Marcinkeviciene J , Chang SY , Biller SA , Kirby MS , Parker RA , Hamann LG |
Ref : Journal of Medicinal Chemistry , 48 :5025 , 2005 |
Abstract : Augeri_2005_J.Med.Chem_48_5025 |
ESTHER : Augeri_2005_J.Med.Chem_48_5025 |
PubMedSearch : Augeri_2005_J.Med.Chem_48_5025 |
PubMedID: 16033281 |