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Title : Rational design of a novel, potent, and orally bioavailable cyclohexylamine DPP-4 inhibitor by application of molecular modeling and X-ray crystallography of sitagliptin - Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
Author(s) : Biftu T , Scapin G , Singh S , Feng D , Becker JW , Eiermann G , He H , Lyons K , Patel S , Petrov A , Sinha-Roy R , Zhang B , Wu J , Zhang X , Doss GA , Thornberry NA , Weber AE |
Ref : Bioorganic & Medicinal Chemistry Lett , 17 :3384 , 2007 |
Abstract : Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
ESTHER : Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
PubMedSearch : Biftu_2007_Bioorg.Med.Chem.Lett_17_3384 |
PubMedID: 17433672 |
Gene_locus related to this paper: human-DPP4 |
Title : Dipeptidyl peptidase IV inhibitors derived from beta-aminoacylpiperidines bearing a fused thiazole, oxazole, isoxazole, or pyrazole - Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
Author(s) : Ashton WT , Sisco RM , Dong H , Lyons KA , He H , Doss GA , Leiting B , Patel RA , Wu JK , Marsilio F , Thornberry NA , Weber AE |
Ref : Bioorganic & Medicinal Chemistry Lett , 15 :2253 , 2005 |
Abstract : Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
ESTHER : Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
PubMedSearch : Ashton_2005_Bioorg.Med.Chem.Lett_15_2253 |
PubMedID: 15837304 |