Report for Dolezal M

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References (16)

Title : Preparation, in vitro evaluation and molecular modelling of pyridinium-quinolinium\/isoquinolinium non-symmetrical bisquaternary cholinesterase inhibitors - Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
Author(s) : Komloova M , Horova A , Hrabinova M , Jun D , Dolezal M , Vinsova J , Kuca K , Musilek K
Ref : Bioorganic & Medicinal Chemistry Lett , 23 :6663 , 2013
Abstract : Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
ESTHER : Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
PubMedSearch : Komloova_2013_Bioorg.Med.Chem.Lett_23_6663
PubMedID: 24220173

Title : Preparation and in vitro screening of symmetrical bis-isoquinolinium cholinesterase inhibitors bearing various connecting linkage--implications for early Myasthenia gravis treatment - Musilek_2011_Eur.J.Med.Chem_46_811
Author(s) : Musilek K , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Nachon F , Dolezal M , Kuca K
Ref : Eur Journal of Medicinal Chemistry , 46 :811 , 2011
Abstract : Musilek_2011_Eur.J.Med.Chem_46_811
ESTHER : Musilek_2011_Eur.J.Med.Chem_46_811
PubMedSearch : Musilek_2011_Eur.J.Med.Chem_46_811
PubMedID: 21236521

Title : The preparation, in vitro screening and molecular docking of symmetrical bisquaternary cholinesterase inhibitors containing a but-(2E)-en-1,4-diyl connecting linkage - Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
Author(s) : Musilek K , Pavlikova R , Marek J , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Dolezal M , Gunn-Moore F , Kuca K
Ref : J Enzyme Inhib Med Chem , 26 :245 , 2011
Abstract : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
ESTHER : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
PubMedSearch : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245
PubMedID: 21406034

Title : Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage-Preparation, in vitro screening and molecular docking - Musilek_2011_Bioorg.Med.Chem_19_754
Author(s) : Musilek K , Komloova M , Holas O , Horova A , Pohanka M , Gunn-Moore F , Dohnal V , Dolezal M , Kuca K
Ref : Bioorganic & Medicinal Chemistry , 19 :754 , 2011
Abstract : Musilek_2011_Bioorg.Med.Chem_19_754
ESTHER : Musilek_2011_Bioorg.Med.Chem_19_754
PubMedSearch : Musilek_2011_Bioorg.Med.Chem_19_754
PubMedID: 21215642

Title : Design, evaluation and structure-activity relationship studies of the AChE reactivators against organophosphorus pesticides - Musilek_2011_Med.Res.Rev_31_548
Author(s) : Musilek K , Dolezal M , Gunn-Moore F , Kuca K
Ref : Med Res Rev , 31 :548 , 2011
Abstract : Musilek_2011_Med.Res.Rev_31_548
ESTHER : Musilek_2011_Med.Res.Rev_31_548
PubMedSearch : Musilek_2011_Med.Res.Rev_31_548
PubMedID: 20027669

Title : Preparation and in vitro screening of symmetrical bispyridinium cholinesterase inhibitors bearing different connecting linkage-initial study for Myasthenia gravis implications - Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
Author(s) : Musilek K , Komloova M , Zavadova V , Holas O , Hrabinova M , Pohanka M , Dohnal V , Nachon F , Dolezal M , Kuca K , Jung YS
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :1763 , 2010
Abstract : Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
ESTHER : Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
PubMedSearch : Musilek_2010_Bioorg.Med.Chem.Lett_20_1763
PubMedID: 20138518

Title : Structure-activity relationship of quaternary acetylcholinesterase inhibitors - outlook for early myasthenia gravis treatment - Komloova_2010_Curr.Med.Chem_17_1810
Author(s) : Komloova M , Musilek K , Dolezal M , Gunn-Moore F , Kuca K
Ref : Curr Med Chem , 17 :1810 , 2010
Abstract : Komloova_2010_Curr.Med.Chem_17_1810
ESTHER : Komloova_2010_Curr.Med.Chem_17_1810
PubMedSearch : Komloova_2010_Curr.Med.Chem_17_1810
PubMedID: 20345342

Title : RP-HPLC determination of the lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker - Musilek_2008_Anal.Bioanal.Chem_391_367
Author(s) : Musilek K , Jampilek J , Dohnal J , Jun D , Gunn-Moore F , Dolezal M , Kuca K
Ref : Anal Bioanal Chem , 391 :367 , 2008
Abstract : Musilek_2008_Anal.Bioanal.Chem_391_367
ESTHER : Musilek_2008_Anal.Bioanal.Chem_391_367
PubMedSearch : Musilek_2008_Anal.Bioanal.Chem_391_367
PubMedID: 18369602

Title : Synthesis of monooxime-monocarbamoyl bispyridinium compounds bearing (E)-but-2-ene linker and evaluation of their reactivation activity against tabun- and paraoxon-inhibited acetylcholinesterase - Musilek_2008_J.Enzyme.Inhib.Med.Chem_23_70
Author(s) : Musilek K , Holas O , Kuca K , Jun D , Dohnal V , Opletalova V , Dolezal M
Ref : J Enzyme Inhib Med Chem , 23 :70 , 2008
Abstract : Musilek_2008_J.Enzyme.Inhib.Med.Chem_23_70
ESTHER : Musilek_2008_J.Enzyme.Inhib.Med.Chem_23_70
PubMedSearch : Musilek_2008_J.Enzyme.Inhib.Med.Chem_23_70
PubMedID: 18341256

Title : Novel series of bispyridinium compounds bearing a (Z)-but-2-ene linker--synthesis and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase - Musilek_2007_Bioorg.Med.Chem.Lett_17_3172
Author(s) : Musilek K , Holas O , Kuca K , Jun D , Dohnal V , Opletalova V , Dolezal M
Ref : Bioorganic & Medicinal Chemistry Lett , 17 :3172 , 2007
Abstract : Musilek_2007_Bioorg.Med.Chem.Lett_17_3172
ESTHER : Musilek_2007_Bioorg.Med.Chem.Lett_17_3172
PubMedSearch : Musilek_2007_Bioorg.Med.Chem.Lett_17_3172
PubMedID: 17383875

Title : Synthesis of a novel series of non-symmetrical bispyridinium compounds bearing a xylene linker and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase - Musilek_2007_J.Enzyme.Inhib.Med.Chem_22_425
Author(s) : Musilek K , Holas O , Kuca K , Jun D , Dohnal V , Dolezal M
Ref : J Enzyme Inhib Med Chem , 22 :425 , 2007
Abstract : Musilek_2007_J.Enzyme.Inhib.Med.Chem_22_425
ESTHER : Musilek_2007_J.Enzyme.Inhib.Med.Chem_22_425
PubMedSearch : Musilek_2007_J.Enzyme.Inhib.Med.Chem_22_425
PubMedID: 17847708

Title : Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker: preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase - Musilek_2007_Bioorg.Med.Chem_15_6733
Author(s) : Musilek K , Holas O , Jun D , Dohnal V , Gunn-Moore F , Opletalova V , Dolezal M , Kuca K
Ref : Bioorganic & Medicinal Chemistry , 15 :6733 , 2007
Abstract : Musilek_2007_Bioorg.Med.Chem_15_6733
ESTHER : Musilek_2007_Bioorg.Med.Chem_15_6733
PubMedSearch : Musilek_2007_Bioorg.Med.Chem_15_6733
PubMedID: 17764957

Title : Synthesis of the novel series of bispyridinium compounds bearing (E)-but-2-ene linker and evaluation of their reactivation activity against chlorpyrifos-inhibited acetylcholinesterase - Musilek_2006_Bioorg.Med.Chem.Lett_16_622
Author(s) : Musilek K , Kuca K , Jun D , Dohnal V , Dolezal M
Ref : Bioorganic & Medicinal Chemistry Lett , 16 :622 , 2006
Abstract : Musilek_2006_Bioorg.Med.Chem.Lett_16_622
ESTHER : Musilek_2006_Bioorg.Med.Chem.Lett_16_622
PubMedSearch : Musilek_2006_Bioorg.Med.Chem.Lett_16_622
PubMedID: 16288867

Title : Synthesis of asymmetrical bispyridinium compounds bearing cyano-moiety and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase - Musilek_2006_Bioorg.Med.Chem.Lett_16_5673
Author(s) : Musilek K , Holas O , Kuca K , Jun D , Dohnal V , Dolezal M
Ref : Bioorganic & Medicinal Chemistry Lett , 16 :5673 , 2006
Abstract : Musilek_2006_Bioorg.Med.Chem.Lett_16_5673
ESTHER : Musilek_2006_Bioorg.Med.Chem.Lett_16_5673
PubMedSearch : Musilek_2006_Bioorg.Med.Chem.Lett_16_5673
PubMedID: 16934462

Title : [Synthesis of reactivators of phosphorylated acetylcholinesterase of bis-pyridiniumdialdoxime type with a 3-oxapentane connecting chain and their testing in vitro on a model of the enzyme inhibited by chlorpyrifos and methylchlorpyrifos] - Musilek_2006_Ceska.Slov.Farm_55_115
Author(s) : Musilek K , Kuca K , Jun D , Dohnal V , Kim TH , Jung YS , Dolezal M
Ref : Ceska a Slovenska Farmacie , 55 :115 , 2006
Abstract : Musilek_2006_Ceska.Slov.Farm_55_115
ESTHER : Musilek_2006_Ceska.Slov.Farm_55_115
PubMedSearch : Musilek_2006_Ceska.Slov.Farm_55_115
PubMedID: 16838488

Title : Synthesis of a novel series of bispyridinium compounds bearing a xylene linker and evaluation of their reactivation activity against chlorpyrifos-inhibited acetylcholinesterase - Musilek_2005_J.Enzyme.Inhib.Med.Chem_20_409
Author(s) : Musilek K , Kuca K , Jun D , Dohnal V , Dolezal M
Ref : J Enzyme Inhib Med Chem , 20 :409 , 2005
Abstract : Musilek_2005_J.Enzyme.Inhib.Med.Chem_20_409
ESTHER : Musilek_2005_J.Enzyme.Inhib.Med.Chem_20_409
PubMedSearch : Musilek_2005_J.Enzyme.Inhib.Med.Chem_20_409
PubMedID: 16335048