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Title : Highly Selective Inhibitors of Dipeptidyl Peptidase 9 (DPP9) Derived from the Clinically Used DPP4-Inhibitor Vildagliptin - Benramdane_2023_J.Med.Chem__ |
Author(s) : Benramdane S , De Loose J , Filippi N , Espadinha M , Beyens O , Rymenant YV , Dirkx L , Bozdag M , Feijens PB , Augustyns K , Caljon G , De Winter H , De Meester I , Van der Veken P |
Ref : Journal of Medicinal Chemistry , : , 2023 |
Abstract : Benramdane_2023_J.Med.Chem__ |
ESTHER : Benramdane_2023_J.Med.Chem__ |
PubMedSearch : Benramdane_2023_J.Med.Chem__ |
PubMedID: 37721854 |
Title : Vildagliptin-Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8\/9-Specific Lead - Benramdane_2022_ChemMedChem__e202200097 |
Author(s) : Benramdane S , De Loose J , Beyens O , Van Rymenant Y , Vliegen G , Augustyns K , De Winter H , De Meester I , Van der Veken P |
Ref : ChemMedChem , :e202200097 , 2022 |
Abstract : Benramdane_2022_ChemMedChem__e202200097 |
ESTHER : Benramdane_2022_ChemMedChem__e202200097 |
PubMedSearch : Benramdane_2022_ChemMedChem__e202200097 |
PubMedID: 35760756 |
Title : Spectrophores as one-dimensional descriptors calculated from three-dimensional atomic properties: applications ranging from scaffold hopping to multi-target virtual screening - Gladysz_2018_J.Cheminform_10_9 |
Author(s) : Gladysz R , Dos Santos FM , Langenaeker W , Thijs G , Augustyns K , De Winter H |
Ref : J Cheminform , 10 :9 , 2018 |
Abstract : Gladysz_2018_J.Cheminform_10_9 |
ESTHER : Gladysz_2018_J.Cheminform_10_9 |
PubMedSearch : Gladysz_2018_J.Cheminform_10_9 |
PubMedID: 29516311 |
Title : Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling - Rea_2017_Eur.J.Med.Chem_139_482 |
Author(s) : Rea D , Van Elzen R , De Winter H , Van Goethem S , Landuyt B , Luyten W , Schoofs L , Van der Veken P , Augustyns K , De Meester I , Fulop V , Lambeir AM |
Ref : Eur Journal of Medicinal Chemistry , 139 :482 , 2017 |
Abstract : Rea_2017_Eur.J.Med.Chem_139_482 |
ESTHER : Rea_2017_Eur.J.Med.Chem_139_482 |
PubMedSearch : Rea_2017_Eur.J.Med.Chem_139_482 |
PubMedID: 28826083 |
Gene_locus related to this paper: porgi-DPP |