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Title : Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE Inhibitor - Catto_2020_ACS.Med.Chem.Lett_11_869 |
Author(s) : Catto M , Pisani L , De la Mora E , Belviso BD , Mangiatordi GF , Pinto A , Palma A , Denora N , Caliandro R , Colletier JP , Silman I , Nicolotti O , Altomare CD |
Ref : ACS Med Chem Lett , 11 :869 , 2020 |
Abstract : Catto_2020_ACS.Med.Chem.Lett_11_869 |
ESTHER : Catto_2020_ACS.Med.Chem.Lett_11_869 |
PubMedSearch : Catto_2020_ACS.Med.Chem.Lett_11_869 |
PubMedID: 32435398 |
Title : Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease - Chalupova_2019_Eur.J.Med.Chem_168_491 |
Author(s) : Chalupova K , Korabecny J , Bartolini M , Monti B , Lamba D , Caliandro R , Pesaresi A , Brazzolotto X , Gastellier AJ , Nachon F , Pejchal J , Jarosova M , Hepnarova V , Jun D , Hrabinova M , Dolezal R , Karasova JZ , Mzik M , Kristofikova Z , Misik J , Muckova L , Jost P , Soukup O , Benkova M , Setnicka V , Habartova L , Chvojkova M , Kleteckova L , Vales K , Mezeiova E , Uliassi E , Valis M , Nepovimova E , Bolognesi ML , Kuca K |
Ref : Eur Journal of Medicinal Chemistry , 168 :491 , 2019 |
Abstract : Chalupova_2019_Eur.J.Med.Chem_168_491 |
ESTHER : Chalupova_2019_Eur.J.Med.Chem_168_491 |
PubMedSearch : Chalupova_2019_Eur.J.Med.Chem_168_491 |
PubMedID: 30851693 |
Gene_locus related to this paper: torca-ACHE |
Title : Kinetic and structural studies on the interactions of Torpedo californica acetylcholinesterase with two donepezil-like rigid analogues - Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
Author(s) : Caliandro R , Pesaresi A , Cariati L , Procopio A , Oliverio M , Lamba D |
Ref : J Enzyme Inhib Med Chem , 33 :794 , 2018 |
Abstract : Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
ESTHER : Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
PubMedSearch : Caliandro_2018_J.Enzyme.Inhib.Med.Chem_33_794 |
PubMedID: 29651884 |
Gene_locus related to this paper: torca-ACHE |