Report for Bak A

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References (5)

Title : Synthesis and Hybrid SAR Property Modeling of Novel Cholinesterase Inhibitors - Kos_2021_Int.J.Mol.Sci_22_
Author(s) : Kos J , Kozik V , Pindjakova D , Jankech T , Smolinski A , Stepankova S , Hosek J , Oravec M , Jampilek J , Bak A
Ref : Int J Mol Sci , 22 : , 2021
Abstract : Kos_2021_Int.J.Mol.Sci_22_
ESTHER : Kos_2021_Int.J.Mol.Sci_22_
PubMedSearch : Kos_2021_Int.J.Mol.Sci_22_
PubMedID: 33810550

Title : Novel Benzene-Based Carbamates for AChE\/BChE Inhibition: Synthesis and Ligand\/Structure-Oriented SAR Study - Bak_2019_Int.J.Mol.Sci_20_1524
Author(s) : Bak A , Kozik V , Kozakiewicz D , Gajcy K , Strub DJ , Swietlicka A , Stepankova S , Imramovsky A , Polanski J , Smolinski A , Jampilek J
Ref : Int J Mol Sci , 20 :1524 , 2019
Abstract : Bak_2019_Int.J.Mol.Sci_20_1524
ESTHER : Bak_2019_Int.J.Mol.Sci_20_1524
PubMedSearch : Bak_2019_Int.J.Mol.Sci_20_1524
PubMedID: 30934674

Title : SAR-mediated Similarity Assessment of the Property Profile for New, Silicon-Based AChE\/BChE Inhibitors - Bak_2019_Int.J.Mol.Sci_20_5385
Author(s) : Bak A , Pizova H , Kozik V , Vorcakova K , Kos J , Treml J , Odehnalova K , Oravec M , Imramovsky A , Bobal P , Smolinski A , Travnicek Z , Jampilek J
Ref : Int J Mol Sci , 20 :5385 , 2019
Abstract : Bak_2019_Int.J.Mol.Sci_20_5385
ESTHER : Bak_2019_Int.J.Mol.Sci_20_5385
PubMedSearch : Bak_2019_Int.J.Mol.Sci_20_5385
PubMedID: 31671776

Title : Proline-Based Carbamates as Cholinesterase Inhibitors - Pizova_2017_Molecules_22_
Author(s) : Pizova H , Havelkova M , Stepankova S , Bak A , Kauerova T , Kozik V , Oravec M , Imramovsky A , Kollar P , Bobal P , Jampilek J
Ref : Molecules , 22 : , 2017
Abstract : Pizova_2017_Molecules_22_
ESTHER : Pizova_2017_Molecules_22_
PubMedSearch : Pizova_2017_Molecules_22_
PubMedID: 29135926

Title : Omarigliptin (MK-3102): a novel long-acting DPP-4 inhibitor for once-weekly treatment of type 2 diabetes - Biftu_2014_J.Med.Chem_57_3205
Author(s) : Biftu T , Sinha-Roy R , Chen P , Qian X , Feng D , Kuethe JT , Scapin G , Gao YD , Yan Y , Krueger D , Bak A , Eiermann G , He J , Cox J , Hicks J , Lyons K , He H , Salituro G , Tong S , Patel S , Doss G , Petrov A , Wu J , Xu SS , Sewall C , Zhang X , Zhang B , Thornberry NA , Weber AE
Ref : Journal of Medicinal Chemistry , 57 :3205 , 2014
Abstract : Biftu_2014_J.Med.Chem_57_3205
ESTHER : Biftu_2014_J.Med.Chem_57_3205
PubMedSearch : Biftu_2014_J.Med.Chem_57_3205
PubMedID: 24660890
Gene_locus related to this paper: human-DPP4