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| Title : Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors - Simpkins_2007_Bioorg.Med.Chem.Lett_17_6476 |
| Author(s) : Simpkins LM , Bolton S , Pi Z , Sutton JC , Kwon C , Zhao G , Magnin DR , Augeri DJ , Gungor T , Rotella DP , Sun Z , Liu Y , Slusarchyk WS , Marcinkeviciene J , Robertson JG , Wang A , Robl JA , Atwal KS , Zahler RL , Parker RA , Kirby MS , Hamann LG |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :6476 , 2007 |
| Abstract : Simpkins_2007_Bioorg.Med.Chem.Lett_17_6476 |
| ESTHER : Simpkins_2007_Bioorg.Med.Chem.Lett_17_6476 |
| PubMedSearch : Simpkins_2007_Bioorg.Med.Chem.Lett_17_6476 |
| PubMedID: 17937986 |
| Title : Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes - Augeri_2005_J.Med.Chem_48_5025 |
| Author(s) : Augeri DJ , Robl JA , Betebenner DA , Magnin DR , Khanna A , Robertson JG , Wang A , Simpkins LM , Taunk P , Huang Q , Han SP , Abboa-Offei B , Cap M , Xin L , Tao L , Tozzo E , Welzel GE , Egan DM , Marcinkeviciene J , Chang SY , Biller SA , Kirby MS , Parker RA , Hamann LG |
| Ref : Journal of Medicinal Chemistry , 48 :5025 , 2005 |
| Abstract : Augeri_2005_J.Med.Chem_48_5025 |
| ESTHER : Augeri_2005_J.Med.Chem_48_5025 |
| PubMedSearch : Augeri_2005_J.Med.Chem_48_5025 |
| PubMedID: 16033281 |
| Title : Synthesis of novel potent dipeptidyl peptidase IV inhibitors with enhanced chemical stability: interplay between the N-terminal amino acid alkyl side chain and the cyclopropyl group of alpha-aminoacyl-l-cis-4,5-methanoprolinenitrile-based inhibitors - Magnin_2004_J.Med.Chem_47_2587 |
| Author(s) : Magnin DR , Robl JA , Sulsky RB , Augeri DJ , Huang Y , Simpkins LM , Taunk PC , Betebenner DA , Robertson JG , Abboa-Offei BE , Wang A , Cap M , Xin L , Tao L , Sitkoff DF , Malley MF , Gougoutas JZ , Khanna A , Huang Q , Han SP , Parker RA , Hamann LG |
| Ref : Journal of Medicinal Chemistry , 47 :2587 , 2004 |
| Abstract : Magnin_2004_J.Med.Chem_47_2587 |
| ESTHER : Magnin_2004_J.Med.Chem_47_2587 |
| PubMedSearch : Magnin_2004_J.Med.Chem_47_2587 |
| PubMedID: 15115400 |