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Title : Combining Experimental and Computational Methods to Produce Conjugates of Anticholinesterase and Antioxidant Pharmacophores with Linker Chemistries Affecting Biological Activities Related to Treatment of Alzheimer's Disease - Makhaeva_2024_Molecules_29_321 |
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serkov IV , Proshin AN , Soldatova YV , Poletaeva DA , Faingold, II , Mumyatova VA , Terentiev AA , Radchenko EV , Palyulin VA , Bachurin SO , Richardson RJ |
Ref : Molecules , 29 :321 , 2024 |
Abstract : Makhaeva_2024_Molecules_29_321 |
ESTHER : Makhaeva_2024_Molecules_29_321 |
PubMedSearch : Makhaeva_2024_Molecules_29_321 |
PubMedID: 38257233 |
Title : Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit beta-amyloid self-aggregation: potential therapeutic agents for Alzheimer's disease - Makhaeva_2023_Front.Pharmacol_14_1219980 |
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serebryakova OG , Shchepochkin AV , Averkov MA , Utepova IA , Demina NS , Radchenko EV , Palyulin VA , Fisenko VP , Bachurin SO , Chupakhin ON , Charushin VN , Richardson RJ |
Ref : Front Pharmacol , 14 :1219980 , 2023 |
Abstract : Makhaeva_2023_Front.Pharmacol_14_1219980 |
ESTHER : Makhaeva_2023_Front.Pharmacol_14_1219980 |
PubMedSearch : Makhaeva_2023_Front.Pharmacol_14_1219980 |
PubMedID: 37654616 |
Title : Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease - Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Grishchenko MV , Lushchekina SV , Astakhova TY , Serebryakova OG , Timokhina EN , Zhilina EF , Shchegolkov EV , Ulitko MV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ |
Ref : Int J Mol Sci , 24 :2285 , 2023 |
Abstract : Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
ESTHER : Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
PubMedSearch : Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
PubMedID: 36768608 |
Title : Conjugates of Tacrine with Salicylamide as Promising Multitarget Agents for Alzheimer's Disease - Grishchenko_2022_ChemMedChem__e202200080 |
Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Rudakova EV , Boltneva NP , Kovaleva NV , Serebryakova OG , Lushchekina SV , Astakhova TY , Zhilina EF , Shchegolkov EV , Richardson RJ , Saloutin VI |
Ref : ChemMedChem , :e202200080 , 2022 |
Abstract : Grishchenko_2022_ChemMedChem__e202200080 |
ESTHER : Grishchenko_2022_ChemMedChem__e202200080 |
PubMedSearch : Grishchenko_2022_ChemMedChem__e202200080 |
PubMedID: 35322571 |
Title : New Multifunctional Agents for Potential Alzheimer's Disease Treatment Based on Tacrine Conjugates with 2-Arylhydrazinylidene-1,3-Diketones - Elkina_2022_Biomolecules_12_ |
Author(s) : Elkina NA , Grishchenko MV , Shchegolkov EV , Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Radchenko EV , Palyulin VA , Zhilina EF , Perminova AN , Lapshin LS , Burgart YV , Saloutin VI , Richardson RJ |
Ref : Biomolecules , 12 : , 2022 |
Abstract : Elkina_2022_Biomolecules_12_ |
ESTHER : Elkina_2022_Biomolecules_12_ |
PubMedSearch : Elkina_2022_Biomolecules_12_ |
PubMedID: 36358901 |
Title : Bis-Amiridines as Acetylcholinesterase and Butyrylcholinesterase Inhibitors: N-Functionalization Determines the Multitarget Anti-Alzheimer's Activity Profile - Makhaeva_2022_Molecules_27_ |
Author(s) : Makhaeva GF , Kovaleva NV , Boltneva NP , Rudakova EV , Lushchekina SV , Astakhova TY , Serkov IV , Proshin AN , Radchenko EV , Palyulin VA , Korabecny J , Soukup O , Bachurin SO , Richardson RJ |
Ref : Molecules , 27 : , 2022 |
Abstract : Makhaeva_2022_Molecules_27_ |
ESTHER : Makhaeva_2022_Molecules_27_ |
PubMedSearch : Makhaeva_2022_Molecules_27_ |
PubMedID: 35164325 |
Title : New Hybrids of 4-Amino-2,3-polymethylene-quinoline and p-Tolylsulfonamide as Dual Inhibitors of Acetyl- and Butyrylcholinesterase and Potential Multifunctional Agents for Alzheimer's Disease Treatment - Makhaeva_2020_Molecules_25_3915 |
Author(s) : Makhaeva GF , Kovaleva NV , Boltneva NP , Lushchekina SV , Astakhova TY , Rudakova EV , Proshin AN , Serkov IV , Radchenko EV , Palyulin VA , Bachurin SO , Richardson RJ |
Ref : Molecules , 25 :3915 , 2020 |
Abstract : Makhaeva_2020_Molecules_25_3915 |
ESTHER : Makhaeva_2020_Molecules_25_3915 |
PubMedSearch : Makhaeva_2020_Molecules_25_3915 |
PubMedID: 32867324 |