5I7U
Name : Human DPP4 in complex with a novel tricyclic hetero-cycle inhibitor
Revelation date : 08-Jun-2016
Family : DPP4N_Peptidase_S9
Gene_locus : human-DPP4
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Scapin, G
Ligand :
References (1)
| Title : Discovery of Novel Tricyclic Heterocycles as Potent and Selective DPP-4 Inhibitors for the Treatment of Type 2 Diabetes - Wu_2016_ACS.Med.Chem.Lett_7_498 |
| Author(s) : Wu WL , Hao J , Domalski M , Burnett DA , Pissarnitski D , Zhao Z , Stamford A , Scapin G , Gao YD , Soriano A , Kelly TM , Yao Z , Powles MA , Chen S , Mei H , Hwa J |
| Ref : ACS Med Chem Lett , 7 :498 , 2016 |
| Abstract : Wu_2016_ACS.Med.Chem.Lett_7_498 |
| ESTHER : Wu_2016_ACS.Med.Chem.Lett_7_498 |
| PubMedSearch : Wu_2016_ACS.Med.Chem.Lett_7_498 |
| PubMedID: 27190600 |
| Gene_locus related to this paper: human-DPP4 |
Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server
