2HHA

Name : The structure of DPP4 in complex with an oxadiazole inhibitor

Revelation date : 19-Sep-2006

Family : DPP4N_Peptidase_S9

Gene_locus : human-DPP4

PDB file : ESTHER: header of PDB entry RCSB: Full entry

Comment
Scapin, G.

Ligand :

References (1)

Title : Discovery of potent, selective, and orally bioavailable oxadiazole-based dipeptidyl peptidase IV inhibitors - Xu_2006_Bioorg.Med.Chem.Lett_16_5373
Author(s) : Xu J , Wei L , Mathvink RJ , Edmondson SD , Eiermann GJ , He H , Leone JF , Leiting B , Lyons KA , Marsilio F , Patel RA , Patel SB , Petrov A , Scapin G , Wu JK , Thornberry NA , Weber AE
Ref : Bioorganic & Medicinal Chemistry Lett , 16 :5373 , 2006
Abstract : Xu_2006_Bioorg.Med.Chem.Lett_16_5373
ESTHER : Xu_2006_Bioorg.Med.Chem.Lett_16_5373
PubMedSearch : Xu_2006_Bioorg.Med.Chem.Lett_16_5373
PubMedID: 16919457
Gene_locus related to this paper: human-DPP4

Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server

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