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Mutation Report for: N68A_human-BCHE

N68A_human-BCHE
Gene_Locus|human-BCHE
Mode of mutation|Site directed mutagenesis
Amino Acid change|N68A
Torpedo number|70
Summary|
Comment|p.N68A Asn68Ala (p.N96A Asn96Ala in primary sequence with 28 amino-acids signal peptide) No effect
Kinetic parameters|BW284C51_N68A_human-BCHE,
Butyrylthiocholine_N68A_human-BCHE,
Dibucaine_N68A_human-BCHE,
Solanine_N68A_human-BCHE,
Succinylcholine~Suxamethonium_N68A_human-BCHE,
Tacrine_N68A_human-BCHE


References:
    Title: Overlapping drug interaction sites of human butyrylcholinesterase dissected by site-directed mutagenesis
    Loewenstein-Lichtenstein Y, Glick D, Gluzman N, Sternfeld M, Zakut H, Soreq H
    Ref: Molecular Pharmacology, 50:1423, 1996 : PubMed

            




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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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