Report for Mukhin AG

General

Full name : Mukhin Alexey G

First name : Alexey G

Mail : Center for Nicotine and Smoking Cessation Research, Duke University Medical Center, 2424 Erwin Road, Suite 201, Durham, NC 27705

Zip Code :

City :

Country : USA

Email : a.mukhin@duke.edu

Phone :

Fax :

Website :

Directory :

References (24)

Title : Brain nicotinic acetylcholine receptor availability and response to smoking cessation treatment: a randomized trial - Brody_2014_JAMA.Psychiatry_71_797
Author(s) : Brody AL , Mukhin AG , Mamoun MS , Luu T , Neary M , Liang L , Shieh J , Sugar CA , Rose JE , Mandelkern MA
Ref : JAMA Psychiatry , 71 :797 , 2014
Abstract : Brody_2014_JAMA.Psychiatry_71_797
ESTHER : Brody_2014_JAMA.Psychiatry_71_797
PubMedSearch : Brody_2014_JAMA.Psychiatry_71_797
PubMedID: 24850280

Title : Up-regulation of nicotinic acetylcholine receptors in menthol cigarette smokers - Brody_2013_Int.J.Neuropsychopharmacol_16_957
Author(s) : Brody AL , Mukhin AG , La Charite J , Ta K , Farahi J , Sugar CA , Mamoun MS , Vellios E , Archie M , Kozman M , Phuong J , Arlorio F , Mandelkern MA
Ref : Int J Neuropsychopharmacol , 16 :957 , 2013
Abstract : Brody_2013_Int.J.Neuropsychopharmacol_16_957
ESTHER : Brody_2013_Int.J.Neuropsychopharmacol_16_957
PubMedSearch : Brody_2013_Int.J.Neuropsychopharmacol_16_957
PubMedID: 23171716

Title : Treatment for tobacco dependence: effect on brain nicotinic acetylcholine receptor density - Brody_2013_Neuropsychopharmacology_38_1548
Author(s) : Brody AL , Mukhin AG , Stephanie S , Mamoun MS , Kozman M , Phuong J , Neary M , Luu T , Mandelkern MA
Ref : Neuropsychopharmacology , 38 :1548 , 2013
Abstract : Brody_2013_Neuropsychopharmacology_38_1548
ESTHER : Brody_2013_Neuropsychopharmacology_38_1548
PubMedSearch : Brody_2013_Neuropsychopharmacology_38_1548
PubMedID: 23429692

Title : Effect of secondhand smoke on occupancy of nicotinic acetylcholine receptors in brain - Brody_2011_Arch.Gen.Psychiatry_68_953
Author(s) : Brody AL , Mandelkern MA , London ED , Khan A , Kozman D , Costello MR , Vellios EE , Archie MM , Bascom R , Mukhin AG
Ref : Arch Gen Psychiatry , 68 :953 , 2011
Abstract : Brody_2011_Arch.Gen.Psychiatry_68_953
ESTHER : Brody_2011_Arch.Gen.Psychiatry_68_953
PubMedSearch : Brody_2011_Arch.Gen.Psychiatry_68_953
PubMedID: 21536968

Title : Brain nicotinic acetylcholine receptor occupancy: effect of smoking a denicotinized cigarette - Brody_2009_Int.J.Neuropsychopharmacol_12_305
Author(s) : Brody AL , Mandelkern MA , Costello MR , Abrams AL , Scheibal D , Farahi J , London ED , Olmstead RE , Rose JE , Mukhin AG
Ref : Int J Neuropsychopharmacol , 12 :305 , 2009
Abstract : Brody_2009_Int.J.Neuropsychopharmacol_12_305
ESTHER : Brody_2009_Int.J.Neuropsychopharmacol_12_305
PubMedSearch : Brody_2009_Int.J.Neuropsychopharmacol_12_305
PubMedID: 18706128

Title : Baseline expression of alpha4beta2* nicotinic acetylcholine receptors predicts motivation to self-administer nicotine - Le_2009_Biol.Psychiatry_65_714
Author(s) : Le Foll B , Chefer SI , Kimes AS , Shumway D , Stein EA , Mukhin AG , Goldberg SR
Ref : Biological Psychiatry , 65 :714 , 2009
Abstract : Le_2009_Biol.Psychiatry_65_714
ESTHER : Le_2009_Biol.Psychiatry_65_714
PubMedSearch : Le_2009_Biol.Psychiatry_65_714
PubMedID: 19095220

Title : Cigarette smoking saturates brain alpha 4 beta 2 nicotinic acetylcholine receptors - Brody_2006_Arch.Gen.Psychiatry_63_907
Author(s) : Brody AL , Mandelkern MA , London ED , Olmstead RE , Farahi J , Scheibal D , Jou J , Allen V , Tiongson E , Chefer SI , Koren AO , Mukhin AG
Ref : Arch Gen Psychiatry , 63 :907 , 2006
Abstract : Brody_2006_Arch.Gen.Psychiatry_63_907
ESTHER : Brody_2006_Arch.Gen.Psychiatry_63_907
PubMedSearch : Brody_2006_Arch.Gen.Psychiatry_63_907
PubMedID: 16894067

Title : The biology of tobacco and nicotine: bench to bedside - Dennis_2005_Cancer.Epidemiol.Biomarkers.Prev_14_764
Author(s) : Dennis PA , Van Waes C , Gutkind JS , Kellar KJ , Vinson C , Mukhin AG , Spitz MR , Bailey-Wilson JE , Yeh GC , Anderson LM , Wiest JS
Ref : Cancer Epidemiol Biomarkers Prev , 14 :764 , 2005
Abstract : Dennis_2005_Cancer.Epidemiol.Biomarkers.Prev_14_764
ESTHER : Dennis_2005_Cancer.Epidemiol.Biomarkers.Prev_14_764
PubMedSearch : Dennis_2005_Cancer.Epidemiol.Biomarkers.Prev_14_764
PubMedID: 15824140

Title : In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for alpha4beta2* nicotinic acetylcholine receptors - Gundisch_2005_Synapse_55_89
Author(s) : Gundisch D , Koren AO , Horti AG , Pavlova OA , Kimes AS , Mukhin AG , London ED
Ref : Synapse , 55 :89 , 2005
Abstract : Gundisch_2005_Synapse_55_89
ESTHER : Gundisch_2005_Synapse_55_89
PubMedSearch : Gundisch_2005_Synapse_55_89
PubMedID: 15529332

Title : Pharmacological and toxicological evaluation of 2-fluoro-3-(2(S)-azetidinylmethoxy)pyridine (2-F-A-85380), a ligand for imaging cerebral nicotinic acetylcholine receptors with positron emission tomography - Vaupel_2005_J.Pharmacol.Exp.Ther_312_355
Author(s) : Vaupel DB , Tella SR , Huso DL , Wagner VO, 3rd , Mukhin AG , Chefer SI , Horti AG , London ED , Koren AO , Kimes AS
Ref : Journal of Pharmacology & Experimental Therapeutics , 312 :355 , 2005
Abstract : Vaupel_2005_J.Pharmacol.Exp.Ther_312_355
ESTHER : Vaupel_2005_J.Pharmacol.Exp.Ther_312_355
PubMedSearch : Vaupel_2005_J.Pharmacol.Exp.Ther_312_355
PubMedID: 15331657

Title : 2-[18F]F-A-85380: PET imaging of brain nicotinic acetylcholine receptors and whole body distribution in humans - Kimes_2003_FASEB.J_17_1331
Author(s) : Kimes AS , Horti AG , London ED , Chefer SI , Contoreggi C , Ernst M , Friello P , Koren AO , Kurian V , Matochik JA , Pavlova O , Vaupel DB , Mukhin AG
Ref : FASEB Journal , 17 :1331 , 2003
Abstract : Kimes_2003_FASEB.J_17_1331
ESTHER : Kimes_2003_FASEB.J_17_1331
PubMedSearch : Kimes_2003_FASEB.J_17_1331
PubMedID: 12759330

Title : Quantification of nicotinic acetylcholine receptors in human brain using [123I]5-I-A-85380 SPET - Fujita_2003_Eur.J.Nucl.Med.Mol.Imaging_30_1620
Author(s) : Fujita M , Ichise M , van Dyck CH , Zoghbi SS , Tamagnan G , Mukhin AG , Bozkurt A , Seneca N , Tipre D , DeNucci CC , Iida H , Vaupel DB , Horti AG , Koren AO , Kimes AS , London ED , Seibyl JP , Baldwin RM , Innis RB
Ref : Eur J Nucl Med Mol Imaging , 30 :1620 , 2003
Abstract : Fujita_2003_Eur.J.Nucl.Med.Mol.Imaging_30_1620
ESTHER : Fujita_2003_Eur.J.Nucl.Med.Mol.Imaging_30_1620
PubMedSearch : Fujita_2003_Eur.J.Nucl.Med.Mol.Imaging_30_1620
PubMedID: 14523584

Title : Graphical analysis of 2-[18F]FA binding to nicotinic acetylcholine receptors in rhesus monkey brain - Chefer_2003_Synapse_48_25
Author(s) : Chefer SI , London ED , Koren AO , Pavlova OA , Kurian V , Kimes AS , Horti AG , Mukhin AG
Ref : Synapse , 48 :25 , 2003
Abstract : Chefer_2003_Synapse_48_25
ESTHER : Chefer_2003_Synapse_48_25
PubMedSearch : Chefer_2003_Synapse_48_25
PubMedID: 12557269

Title : Conditional expression in corticothalamic efferents reveals a developmental role for nicotinic acetylcholine receptors in modulation of passive avoidance behavior - King_2003_J.Neurosci_23_3837
Author(s) : King SL , Marks MJ , Grady SR , Caldarone BJ , Koren AO , Mukhin AG , Collins AC , Picciotto MR
Ref : Journal of Neuroscience , 23 :3837 , 2003
Abstract : King_2003_J.Neurosci_23_3837
ESTHER : King_2003_J.Neurosci_23_3837
PubMedSearch : King_2003_J.Neurosci_23_3837
PubMedID: 12736354

Title : Whole-body biodistribution, radiation absorbed dose, and brain SPET imaging with [123i]5-i-A-85380 in healthy human subjects - Fujita_2002_Eur.J.Nucl.Med.Mol.Imaging_29_183
Author(s) : Fujita M , Seibyl JP , Vaupel DB , Tamagnan G , Early M , Zoghbi SS , Baldwin RM , Horti AG , Kore NA , Mukhin AG , Khan S , Bozkurt A , Kimes AS , London ED , Innis RB
Ref : Eur J Nucl Med Mol Imaging , 29 :183 , 2002
Abstract : Fujita_2002_Eur.J.Nucl.Med.Mol.Imaging_29_183
ESTHER : Fujita_2002_Eur.J.Nucl.Med.Mol.Imaging_29_183
PubMedSearch : Fujita_2002_Eur.J.Nucl.Med.Mol.Imaging_29_183
PubMedID: 11926380

Title : Development of ligands for in vivo imaging of cerebral nicotinic receptors - Sihver_2000_Behav.Brain.Res_113_143
Author(s) : Sihver W , Nordberg A , Langstrom B , Mukhin AG , Koren AO , Kimes AS , London ED
Ref : Behavioural Brain Research , 113 :143 , 2000
Abstract : Sihver_2000_Behav.Brain.Res_113_143
ESTHER : Sihver_2000_Behav.Brain.Res_113_143
PubMedSearch : Sihver_2000_Behav.Brain.Res_113_143
PubMedID: 10942041

Title : 6-[18F]fluoro-A-85380, a novel radioligand for in vivo imaging of central nicotinic acetylcholine receptors - Horti_2000_Life.Sci_67_463
Author(s) : Horti AG , Chefer SI , Mukhin AG , Koren AO , Gundisch D , Links JM , Kurian V , Dannals RF , London ED
Ref : Life Sciences , 67 :463 , 2000
Abstract : Horti_2000_Life.Sci_67_463
ESTHER : Horti_2000_Life.Sci_67_463
PubMedSearch : Horti_2000_Life.Sci_67_463
PubMedID: 11003056

Title : 5-Iodo-A-85380, an alpha4beta2 subtype-selective ligand for nicotinic acetylcholine receptors - Mukhin_2000_Mol.Pharmacol_57_642
Author(s) : Mukhin AG , Gundisch D , Horti AG , Koren AO , Tamagnan G , Kimes AS , Chambers J , Vaupel DB , King SL , Picciotto MR , Innis RB , London ED
Ref : Molecular Pharmacology , 57 :642 , 2000
Abstract : Mukhin_2000_Mol.Pharmacol_57_642
ESTHER : Mukhin_2000_Mol.Pharmacol_57_642
PubMedSearch : Mukhin_2000_Mol.Pharmacol_57_642
PubMedID: 10692507

Title : High affinity binding of [3H]epibatidine to rat brain membranes - Gnadisch_1999_Neuroreport_10_1631
Author(s) : Gnadisch D , London ED , Terry P , Hill GR , Mukhin AG
Ref : Neuroreport , 10 :1631 , 1999
Abstract : Gnadisch_1999_Neuroreport_10_1631
ESTHER : Gnadisch_1999_Neuroreport_10_1631
PubMedSearch : Gnadisch_1999_Neuroreport_10_1631
PubMedID: 10501548

Title : 2-[18F]F-A-85380: a PET radioligand for alpha4beta2 nicotinic acetylcholine receptors - Chefer_1999_Neuroreport_10_2715
Author(s) : Chefer SI , Horti AG , Koren AO , Gundisch D , Links JM , Kurian V , Dannals RF , Mukhin AG , London ED
Ref : Neuroreport , 10 :2715 , 1999
Abstract : Chefer_1999_Neuroreport_10_2715
ESTHER : Chefer_1999_Neuroreport_10_2715
PubMedSearch : Chefer_1999_Neuroreport_10_2715
PubMedID: 10511429

Title : Radiosynthesis and preliminary evaluation of 5-[123\/125I]iodo-3-(2(S)-azetidinylmethoxy)pyridine: a radioligand for nicotinic acetylcholine receptors - Horti_1999_Nucl.Med.Biol_26_175
Author(s) : Horti AG , Koren AO , Lee KS , Mukhin AG , Vaupel DB , Kimes AS , Stratton M , London ED
Ref : Nucl Med Biol , 26 :175 , 1999
Abstract : Horti_1999_Nucl.Med.Biol_26_175
ESTHER : Horti_1999_Nucl.Med.Biol_26_175
PubMedSearch : Horti_1999_Nucl.Med.Biol_26_175
PubMedID: 10100216

Title : 2-, 5-, and 6-Halo-3-(2(S)-azetidinylmethoxy)pyridines: synthesis, affinity for nicotinic acetylcholine receptors, and molecular modeling - Koren_1998_J.Med.Chem_41_3690
Author(s) : Koren AO , Horti AG , Mukhin AG , Gundisch D , Kimes AS , Dannals RF , London ED
Ref : Journal of Medicinal Chemistry , 41 :3690 , 1998
Abstract : Koren_1998_J.Med.Chem_41_3690
ESTHER : Koren_1998_J.Med.Chem_41_3690
PubMedSearch : Koren_1998_J.Med.Chem_41_3690
PubMedID: 9733494

Title : In vivo studies with [125I]5-I-A-85380, a nicotinic acetylcholine receptor radioligand - Vaupel_1998_Neuroreport_9_2311
Author(s) : Vaupel DB , Mukhin AG , Kimes AS , Horti AG , Koren AO , London ED
Ref : Neuroreport , 9 :2311 , 1998
Abstract : Vaupel_1998_Neuroreport_9_2311
ESTHER : Vaupel_1998_Neuroreport_9_2311
PubMedSearch : Vaupel_1998_Neuroreport_9_2311
PubMedID: 9694220

Title : In vivo imaging of brain nicotinic acetylcholine receptors with 5-[123I]iodo-A-85380 using single photon emission computed tomography - Chefer_1998_Life.Sci_63_PL355
Author(s) : Chefer SI , Horti AG , Lee KS , Koren AO , Jones DW , Gorey JG , Links JM , Mukhin AG , Weinberger DR , London ED
Ref : Life Sciences , 63 :PL355 , 1998
Abstract : Chefer_1998_Life.Sci_63_PL355
ESTHER : Chefer_1998_Life.Sci_63_PL355
PubMedSearch : Chefer_1998_Life.Sci_63_PL355
PubMedID: 9870715