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Title : Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9 - Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
Author(s) : Carvalho LAR , Ross B , Fehr L , Bolgi O , Wohrle S , Lum KM , Podlesainski D , Vieira AC , Kiefersauer R , Felix R , Rodrigues T , Lucas SD , Gross O , Geiss-Friedlander R , Cravatt BF , Huber R , Kaiser M , Moreira R |
Ref : Angew Chem Int Ed Engl , : , 2022 |
Abstract : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
ESTHER : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
PubMedSearch : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
PubMedID: 36089535 |
Gene_locus related to this paper: human-DPP8 , human-DPP9 |
Title : 3-Oxo-beta-sultam as a Sulfonylating Chemotype for Inhibition of Serine Hydrolases and Activity-Based Protein Profiling - Carvalho_2020_ACS.Chem.Biol_15_878 |
Author(s) : Carvalho LAR , Almeida VT , Brito JA , Lum KM , Oliveira TF , Guedes RC , Goncalves LM , Lucas SD , Cravatt BF , Archer M , Moreira R |
Ref : ACS Chemical Biology , 15 :878 , 2020 |
Abstract : Carvalho_2020_ACS.Chem.Biol_15_878 |
ESTHER : Carvalho_2020_ACS.Chem.Biol_15_878 |
PubMedSearch : Carvalho_2020_ACS.Chem.Biol_15_878 |
PubMedID: 32176480 |